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1
المؤلفون: Graeme Bainbridge, Nicole Caspers, Andrew Robertson, Jeffrey A. Pfefferkorn, Yuntao Song, Lisa Dillon, Catherine Sekerke, Jeffrey C. Hanselman, Chulho Choi, Gina Lu, Valerie Askew, Zhiwu Lin, Alexander Pavlovsky, Bharat K. Trivedi, Bruce Auerbach, Scott D. Larsen, Melissa S. Harris
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:4531-4537
مصطلحات موضوعية: Clinical Biochemistry, Pharmaceutical Science, Hyperlipidemias, Reductase, Biochemistry, Chemical synthesis, Mice, Structure-Activity Relationship, In vivo, Drug Discovery, Animals, Structure–activity relationship, Pyrroles, Molecular Biology, chemistry.chemical_classification, Molecular Structure, biology, Chemistry, Organic Chemistry, Hydroxymethylglutaryl-CoA reductase, Cholesterol, Enzyme, Enzyme inhibitor, Drug Design, HMG-CoA reductase, biology.protein, Molecular Medicine, lipids (amino acids, peptides, and proteins), Hydroxymethylglutaryl-CoA Reductase Inhibitors
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2
المؤلفون: Jeffrey A. Pfefferkorn, Lisa Dillon, Larry D. Bratton, Bruce Auerbach, Bharat K. Trivedi, Jeffrey C. Hanselman, Scott D. Larsen, Andrew Robertson, Catherine Sekerke, Gina Lu, Paul C. Unangst, Chulho Choi, Karl Olsen
المصدر: Bioorganic & Medicinal Chemistry. 15:5576-5589
مصطلحات موضوعية: Male, Stereochemistry, Clinical Biochemistry, Substituent, Pharmaceutical Science, Reductase, Ligands, Biochemistry, Chemical synthesis, Rats, Sprague-Dawley, chemistry.chemical_compound, Drug Discovery, Animals, Pyrroles, Molecular Biology, Alkyl, Pyrrole, chemistry.chemical_classification, Molecular Structure, biology, Organic Chemistry, Hydroxymethylglutaryl-CoA reductase, Rats, Cholesterol, Liver, chemistry, HMG-CoA reductase, Lipophilicity, Microsomes, Liver, biology.protein, Molecular Medicine, Hydroxymethylglutaryl CoA Reductases, Hydroxymethylglutaryl-CoA Reductase Inhibitors
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3
المؤلفون: Yuntao Song, Jeffrey C. Hanselman, Xue-Min Cheng, Scott D. Larsen, Zhiwu Lin, Bharat K. Trivedi, Graeme Bainbridge, Alexander Pavlovsky, Larry D. Bratton, Andrew Robertson, Paul C. Unangst, Jeffrey A. Pfefferkorn, Melissa S. Harris, Lisa Dillon, Bruce Auerbach, Erasga Noe Ouano, Chitase Lee, Chulho Choi, Karl Olsen, Catherine Sekerke, Toni Jo Poel, Nicole Caspers, Matthias Eberstadt, Kuai Lin Sun, Steven R. Miller, Roderick Joseph Sorenson, Gina Lu, Valerie Askew, Thomas E. Mertz, Huifen Chen
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:4538-4544
مصطلحات موضوعية: Models, Molecular, Statin, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Hyperlipidemias, Reductase, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Cricetinae, Drug Discovery, medicine, Animals, Structure–activity relationship, Pyrroles, Rosuvastatin Calcium, Molecular Biology, chemistry.chemical_classification, Sulfonamides, Dose-Response Relationship, Drug, Molecular Structure, biology, Organic Chemistry, Hydroxymethylglutaryl-CoA reductase, Fluorobenzenes, Pyrimidines, Enzyme, Liver, chemistry, Enzyme inhibitor, Drug Design, HMG-CoA reductase, biology.protein, Molecular Medicine, Hydroxymethylglutaryl-CoA Reductase Inhibitors
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4
المؤلفون: Jay R. Luly, Kenneth G. Carson, David J Heilig, Wen Song Yue, Shixin Qin, Jie Jack Li, David T. Connor, Joseph Edwin Low, Roberta A Glynn, Bharat K. Trivedi, Qing Ye, Stephen W. Hunt, Steven R. Miller, Bruce D. Roth, Weixing Yang
المصدر: Bioorganic & Medicinal Chemistry. 11:3777-3790
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Anti-Inflammatory Agents, Pharmaceutical Science, Antineoplastic Agents, Diamines, Biochemistry, Chemical synthesis, Receptors, Interleukin-8A, Structure-Activity Relationship, Quinoxalines, Drug Discovery, Humans, Structure–activity relationship, Interleukin 8, Receptor, Molecular Biology, Bicyclic molecule, Chemistry, Chemotaxis, Organic Chemistry, Interleukin-8 receptor, Small molecule, In vitro, Molecular Medicine, Calcium
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5Addition reactions of allyl stannanes to an indolo[2′,3′:3,4]pyrido[1,2-b]isoquinoline imminium salt
المؤلفون: David T. Connor, Bruce D. Roth, Paul C. Unangst, Larry D. Bratton, Bharat K. Trivedi, J. Ronald Rubin
المصدر: Journal of Heterocyclic Chemistry. 37:1081-1087
مصطلحات موضوعية: chemistry.chemical_classification, Addition reaction, Organic Chemistry, chemistry.chemical_element, Salt (chemistry), Medicinal chemistry, Adduct, chemistry.chemical_compound, chemistry, Reagent, Yield (chemistry), Proton NMR, Isoquinoline, Tin
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6
المؤلفون: Bruce D. Roth, Jie Jack Li, J. Ronald Rubin, Bharat K. Trivedi
المصدر: Tetrahedron Letters. 39:6111-6114
مصطلحات موضوعية: chemistry.chemical_classification, Organic Chemistry, Alkaloid synthesis, Iminium, Salt (chemistry), Biochemistry, Enamine, chemistry.chemical_compound, chemistry, Acetyl chloride, Reagent, Drug Discovery, Robinson annulation, Organic chemistry
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7
المؤلفون: N. Suman-Chauhan, Louise Webdale, Bharat K. Trivedi, Terri S. Purchase, Bruce D. Roth, Bradley Dean Tait, Michael W. Wilson, C.E. Augelli-Szafran
المصدر: Bioorganic & Medicinal Chemistry Letters. 7:2009-2014
مصطلحات موضوعية: chemistry.chemical_classification, Indole test, Stereochemistry, medicine.drug_class, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Biological activity, Receptor antagonist, Biochemistry, Chemical synthesis, CI-988, chemistry, Heterocyclic compound, Drug Discovery, medicine, Molecular Medicine, Moiety, Molecular Biology
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8
المؤلفون: R. L. Stanfield, K. L. Hamelehle, Brian R. Krause, Bharat K. Trivedi, A. D. Essenburg, Ann Holmes, Terri S. Purchase, MaryKay Shaw Hes
المصدر: Bioorganic & Medicinal Chemistry. 5:739-747
مصطلحات موضوعية: Magnetic Resonance Spectroscopy, Stereochemistry, Hypercholesterolemia, Clinical Biochemistry, Rat model, Sterol O-acyltransferase, Administration, Oral, Pharmaceutical Science, Biochemistry, Fluorides, Structure-Activity Relationship, chemistry.chemical_compound, Total cholesterol, Drug Discovery, Benzene Derivatives, Animals, Urea, Structure–activity relationship, Molecular Biology, Total plasma, Chemistry, Cholesterol, Anticholesteremic Agents, Organic Chemistry, Diet, Rats, Cholesterol blood, Disease Models, Animal, Molecular Medicine, Rabbits, Sterol O-Acyltransferase
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9
المؤلفون: Alan Daugherty, Kathryn Welch, Richard D. Dyer, Joseph A. Cornicelli, Thomas M.A. Bocan, Sandra M. Sendobry, Bharat K. Trivedi, Steven J. Feinmark, Norman L. Colbry, Bradley Dean Tait
المصدر: British Journal of Pharmacology. 120:1199-1206
مصطلحات موضوعية: Pharmacology, medicine.medical_specialty, Antioxidant, biology, Cholesterol, medicine.medical_treatment, Arteriosclerosis, medicine.disease, chemistry.chemical_compound, Endocrinology, ABAP, chemistry, Enzyme inhibitor, In vivo, Internal medicine, medicine, biology.protein, computer, Ex vivo, Lipoprotein, computer.programming_language
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10
المؤلفون: Louise Webdale, Bharat K. Trivedi, Janak K. Padia, N. Suman-Chauhan, H. Chilvers, Robert D. Pinnock, P. Daum
المصدر: Bioorganic & Medicinal Chemistry Letters. 7:805-810
مصطلحات موضوعية: Quinazoline derivatives, Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Asperlicin, Biochemistry, Combinatorial chemistry, Chemical synthesis, chemistry.chemical_compound, One pot reaction, Drug Discovery, Molecular Medicine, Receptor, Molecular Biology, Cholecystokinin