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المؤلفون: NaHong Qiu, Birgit Molitor, Justine Badée, Gabriele Cruciani, Stephen Fowler, Nicolo Milani
المصدر: Drug Metabolism and Disposition. 48:176-186
مصطلحات موضوعية: UGT 2B10, N-GLUCURONIDATION, UGT1A4, COMMON, Glucuronidation, Pharmaceutical Science, NICOTINE, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, UDP-GLUCURONOSYLTRANSFERASE ENZYMES, In vivo, DRUG-INTERACTION, Humans, Glucuronosyltransferase, Pharmacology, chemistry.chemical_classification, Virtual screening, Polymorphism, Genetic, Drug interaction, In vitro, COTININE, Phenotype, Enzyme, Pharmaceutical Preparations, chemistry, Biochemistry, 030220 oncology & carcinogenesis, Microsomes, Liver, Microsome, INHIBITORS, 1A4
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3840194123b98eedc0b7f47330c3519a
https://doi.org/10.1124/dmd.119.089482 -
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المؤلفون: Rolf Michels, Kerstin Rickert, Birgit Molitor, Joachim Scheele, Petra Wagner
المصدر: Open Dialogue for Psychosis ISBN: 9781351199599
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::a18d6c679738f2f27d56cbc398c9b0ed
https://doi.org/10.4324/9781351199599-10 -
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المؤلفون: Luca Docci, Florian Klammers, Aynur Ekiciler, Birgit Molitor, Kenichi Umehara, Isabelle Walter, Stephan Krähenbühl, Neil Parrott, Stephen Fowler
المصدر: The AAPS Journal. 22
مصطلحات موضوعية: Pharmaceutical Science
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المؤلفون: Stephen Fowler, Luca Docci, Kenichi Umehara, Aynur Ekiciler, Neil Parrott, Birgit Molitor, Florian Klammers, Isabelle Walter, Stephan Krähenbühl
المصدر: The AAPS journal. 22(6)
مصطلحات موضوعية: Male, Primary Cell Culture, Pharmaceutical Science, Plasma protein binding, Pharmacology, 030226 pharmacology & pharmacy, Models, Biological, 03 medical and health sciences, Mice, 0302 clinical medicine, Glucuronides, Pharmacokinetics, In vivo, Animals, Humans, Glucuronosyltransferase, chemistry.chemical_classification, biology, Chemistry, Cytochrome P450, Metabolism, Fibroblasts, In vitro, Coculture Techniques, Hepatobiliary Elimination, Enzyme, Liver, 030220 oncology & carcinogenesis, biology.protein, Hepatocytes, Female, Drug metabolism
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المؤلفون: Josephine Schmaler, Mohammed Ullah, Franziska Boess, Birgit Molitor, Aynur Ekiciler, Alexandre Durrwell, Isabelle Walter, Brian Leonard, Nicole A. Kratochwil, Giorgio Ottaviani, Russell Jones, Charles Alexandre Tournillac, Florian Klammers, Yuyan Jin, Neil Parrott, Martina B. Mueller, Dan Turley, Stephen Fowler, Michaela Marschmann, Pierre-Alexis Gonsard, Miriam Triyatni
المصدر: Journal of Pharmacology and Experimental Therapeutics. 365:237-248
مصطلحات موضوعية: 0301 basic medicine, Hepatitis B virus, Physiologically based pharmacokinetic modelling, Time Factors, Pharmacology, Antiviral Agents, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, Cytochrome P-450 Enzyme System, Pharmacokinetics, medicine, Humans, Distribution (pharmacology), Drug Interactions, Tissue Distribution, Enzyme inducer, ADME, Dose-Response Relationship, Drug, biology, Chemistry, Cytochrome P450, Biological Transport, In vitro, Kinetics, 030104 developmental biology, Liver, Hepatocytes, biology.protein, Molecular Medicine, Ritonavir, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f58a3bb7e1d0e52e6b59ad6ff7a653e7
https://doi.org/10.1124/jpet.117.245712 -
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المؤلفون: Andrea Treyer, Mohammed Ullah, Birgit Molitor, Per Artursson, Stephen Fowler, Neil Parrott
المصدر: The AAPS Journal
مصطلحات موضوعية: Male, Drug-drug interaction, Pharmacology toxicology, Pharmaceutical Science, Pharmacy, Pharmacology and Toxicology, Pharmacology, 030226 pharmacology & pharmacy, Models, Biological, Pharmaceutical Sciences, 03 medical and health sciences, 0302 clinical medicine, Drug Development, Cytochrome P-450 CYP2D6 Inhibitors, Medicine, Humans, Drug Interactions, Pharmaceutical sciences, unbound drug concentrations, Cells, Cultured, intracellular bioavailability, business.industry, Drug discovery, Farmakologi och toxikologi, Farmaceutiska vetenskaper, Enzyme inhibition, Pharmaceutical Preparations, scaling factor, 030220 oncology & carcinogenesis, Hepatocytes, Microsomes, Liver, physiologically based pharmacokinetic modeling, Cytochrome P-450 CYP3A Inhibitors, Female, business, Intracellular, drug-drug interaction, Research Article
وصف الملف: application/pdf
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المؤلفون: Birgit Molitor, Simon Detzner, Tim Tetaz, Arno Friedlein, Jean-Luc Mary
المصدر: Journal of chromatography. A. 1218(35)
مصطلحات موضوعية: Gene isoform, Cytochrome, Apolipoproteins M, Biochemistry, Analytical Chemistry, law.invention, law, Cell Line, Tumor, medicine, Animals, Humans, Protein Isoforms, Horses, Prontosil, Chromatography, biology, Apolipoprotein A-I, Chemistry, Hydrophilic interaction chromatography, Organic Chemistry, Cytochromes c, Proteins, General Medicine, Lipocalins, APOM, Apolipoproteins, Solubility, biology.protein, Recombinant DNA, lipids (amino acids, peptides, and proteins), Hydrophobic and Hydrophilic Interactions, medicine.drug, Chromatography, Liquid
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المؤلفون: Sandrine Simon, Nicole A. Kratochwil, Johanna Walther, Christoph Funk, Claudia McGinnis, Aynur Ekiciler, Thierry Lavé, Miriam Triyatni, Christophe Meille, Isabelle Walter, Neil Parrott, Florian Klammers, Birgit Molitor, Brian Leonard, Stephen Fowler, Franz Schuler, Hassan Javanbakht
المصدر: The AAPS Journal. 19(2):534-550
مصطلحات موضوعية: 0301 basic medicine, CYP2D6, Time Factors, Pharmaceutical Science, Pharmacology, Biology, 030226 pharmacology & pharmacy, Models, Biological, 03 medical and health sciences, 0302 clinical medicine, In vivo, medicine, Humans, Pharmacokinetics, chemistry.chemical_classification, Transporter, Hep G2 Cells, In vitro, Coculture Techniques, Enzymes, 030104 developmental biology, Enzyme, medicine.anatomical_structure, chemistry, Cytochrome P-450 CYP2D6, Liver, Nonlinear Dynamics, Pharmaceutical Preparations, Cell culture, Hepatocyte, Hepatocytes, Drug metabolism
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d91e7923231330205cba35662a26d35f