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1دورية أكاديمية
المؤلفون: Erik Ylipää, Swapnil Chavan, Maria Bånkestad, Johan Broberg, Björn Glinghammar, Ulf Norinder, Ian Cotgreave
المصدر: Current Research in Toxicology, Vol 5, Iss , Pp 100121- (2023)
مصطلحات موضوعية: Deep Learning, Graph-neural Network, hERG Channel, Random Forest, Recurrent-neural Network, Support-vector Machines, Toxicology. Poisons, RA1190-1270
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Marcin Buler, Thomas Naessens, Johan Mattsson, Yannick Morias, Magnus Söderberg, Philip Robbins, Lillevi Kärrberg, Tor S. Svensson, Petra Thulin, Björn Glinghammar, Richard C. Scarpulla, Ulf Andersson
المصدر: FASEB BioAdvances, Vol 2, Iss 8, Pp 453-463 (2020)
مصطلحات موضوعية: cytokine expression, drug‐induced liver injury, hepatic inflammation, PPRC1, PRC, Biology (General), QH301-705.5
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2573-9832
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المؤلفون: Andrej Emanuel Cotman, Martina Durcik, Davide Benedetto Tiz, Federica Fulgheri, Daniela Secci, Maša Sterle, Štefan Možina, Žiga Skok, Nace Zidar, Anamarija Zega, Janez Ilaš, Lucija Peterlin Mašič, Tihomir Tomašič, Diarmaid Hughes, Douglas L. Huseby, Sha Cao, Linnéa Garoff, Talía Berruga Fernández, Paraskevi Giachou, Lisa Crone, Ivailo Simoff, Richard Svensson, Bryndis Birnir, Sergiy V. Korol, Zhe Jin, Francisca Vicente, Maria C. Ramos, Mercedes de la Cruz, Björn Glinghammar, Lena Lenhammar, Sara R. Henderson, Julia E. A. Mundy, Anthony Maxwell, Clare E. M. Stevenson, David M. Lawson, Guido V. Janssen, Geert Jan Sterk, Danijel Kikelj
المساهمون: Medicinal chemistry, AIMMS
المصدر: Journal of medicinal chemistry, vol. 66, no. 2, 2023.
Journal of medicinal chemistry, str. 1380-1425 : Ilustr., Vol. 66, no. 2, 2023
COBISS-ID: 512806681
Journal of medicinal chemistry, 66(2), 1380-1425. American Chemical Society
Cotman, A E, Durcik, M, Benedetto Tiz, D, Fulgheri, F, Secci, D, Sterle, M, Možina, Š, Skok, Ž, Zidar, N, Zega, A, Ilaš, J, Peterlin Mašič, L, Tomašič, T, Hughes, D, Huseby, D L, Cao, S, Garoff, L, Berruga Fernández, T, Giachou, P, Crone, L, Simoff, I, Svensson, R, Birnir, B, Korol, S V, Jin, Z, Vicente, F, Ramos, M C, De La Cruz, M, Glinghammar, B, Lenhammar, L, Henderson, S R, Mundy, J E A, Maxwell, A, Stevenson, C E M, Lawson, D M, Janssen, G V, Sterk, G J & Kikelj, D 2023, ' Discovery and Hit-to-Lead Optimization of Benzothiazole Scaffold-Based DNA Gyrase Inhibitors with Potent Activity against Acinetobacter baumannii and Pseudomonas aeruginosa ', Journal of medicinal chemistry, vol. 66, no. 2, pp. 1380-1425 . https://doi.org/10.1021/acs.jmedchem.2c01597مصطلحات موضوعية: antibacterial activity, bacteria, genetics, inhibitors, solubility, zaviralci, topnost, bakterijska rezistenca, solubility, Bakterijska rezistenca, Topnost, Läkemedelskemi, udc:615, bakterije, Bakterije, antibacterial activity, genetika, Drug Discovery, inhibitors, Molecular Medicine, antibakterijsko delovanje, zaviralci, genetics, antibakterijsko delovanje, Genetika, Medicinal Chemistry, bacteria, udc:615.015.8
وصف الملف: application/pdf; text/url
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المؤلفون: Nadilly Bonagas, Nina M. S. Gustafsson, Martin Henriksson, Petra Marttila, Robert Gustafsson, Elisée Wiita, Sanjay Borhade, Alanna C. Green, Karl S. A. Vallin, Antonio Sarno, Richard Svensson, Camilla Göktürk, Therese Pham, Ann-Sofie Jemth, Olga Loseva, Victoria Cookson, Nicole Kiweler, Lars Sandberg, Azita Rasti, Judith E. Unterlass, Martin Haraldsson, Yasmin Andersson, Emma R. Scaletti, Christoffer Bengtsson, Cynthia B. J. Paulin, Kumar Sanjiv, Eldar Abdurakhmanov, Linda Pudelko, Ben Kunz, Matthieu Desroses, Petar Iliev, Katarina Färnegårdh, Andreas Krämer, Neeraj Garg, Maurice Michel, Sara Häggblad, Malin Jarvius, Christina Kalderén, Amanda Bögedahl Jensen, Ingrid Almlöf, Stella Karsten, Si Min Zhang, Maria Häggblad, Anders Eriksson, Jianping Liu, Björn Glinghammar, Natalia Nekhotiaeva, Fredrik Klingegård, Tobias Koolmeister, Ulf Martens, Sabin Llona-Minguez, Ruth Moulson, Helena Nordström, Vendela Parrow, Leif Dahllund, Birger Sjöberg, Irene L. Vargas, Duy Duc Vo, Johan Wannberg, Stefan Knapp, Hans E. Krokan, Per I. Arvidsson, Martin Scobie, Johannes Meiser, Pål Stenmark, Ulrika Warpman Berglund, Evert J. Homan, Thomas Helleday
المصدر: Nature Cancer
مصطلحات موضوعية: Methylenetetrahydrofolate Dehydrogenase (NADP), Cancer och onkologi, Leukemia, Myeloid, Acute, Cancer Research, Oncology, Cellbiologi, Aminohydrolases, Hydrolases, Cancer and Oncology, Humans, Cell Biology, Multifunctional Enzymes, Thymidine
وصف الملف: application/pdf
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المؤلفون: Martina Durcik, Andrej Emanuel Cotman, Žan Toplak, Štefan Možina, Žiga Skok, Petra Eva Szili, Márton Czikkely, Elvin Maharramov, Thu Hien Vu, Maria Vittoria Piras, Nace Zidar, Janez Ilaš, Anamarija Zega, Jurij Trontelj, Luis A. Pardo, Diarmaid Hughes, Douglas Huseby, Tália Berruga-Fernández, Sha Cao, Ivailo Simoff, Richard Svensson, Sergiy V. Korol, Zhe Jin, Francisca Vicente, Maria C. Ramos, Julia E. A. Mundy, Anthony Maxwell, Clare E. M. Stevenson, David M. Lawson, Björn Glinghammar, Eva Sjöström, Martin Bohlin, Joanna Oreskär, Sofie Alvér, Guido V. Janssen, Geert Jan Sterk, Danijel Kikelj, Csaba Pal, Tihomir Tomašič, Lucija Peterlin Mašič
المساهمون: Medicinal chemistry, AIMMS
المصدر: Durcik, M, Cotman, A E, Toplak, Ž, Možina, Š, Skok, Ž, Szili, P E, Czikkely, M, Maharramov, E, Vu, T H, Piras, M V, Zidar, N, Ilaš, J, Zega, A, Trontelj, J, Pardo, L A, Hughes, D, Huseby, D, Berruga-Fernández, T, Cao, S, Simoff, I, Svensson, R, Korol, S V, Jin, Z, Vicente, F, Ramos, M C, Mundy, J E A, Maxwell, A, Stevenson, C E M, Lawson, D M, Glinghammar, B, Sjöström, E, Bohlin, M, Oreskär, J, Alvér, S, Janssen, G V, Sterk, G J, Kikelj, D, Pal, C, Tomašič, T & Peterlin Mašič, L 2023, ' New Dual Inhibitors of Bacterial Topoisomerases with Broad-Spectrum Antibacterial Activity and In Vivo Efficacy against Vancomycin-Intermediate Staphylococcus aureus ', Journal of medicinal chemistry, vol. 66, no. 6, pp. 3968-3994 . https://doi.org/10.1021/acs.jmedchem.2c01905
Journal of medicinal chemistry, 66(6), 3968-3994. American Chemical Society
Journal of Medicinal Chemistry
Journal of medicinal chemistry, str. 3968-3994 : Ilustr., Vol. 66, iss. 6, 2023
COBISS-ID: 512806681
Journal of medicinal chemistry, vol. 66, no. 6, pp. 3968-3994, 2023.مصطلحات موضوعية: Infectious Medicine, topoizomeraza IV, bakterijska rezistenca, nanomolarni inhibitorji benzotiazola, Farmacevtska kemija, Infektionsmedicin, peptides and proteins, antibakterijsko delovanje, zaviralci, nanomolarni inhibitorji benzotiazola, topoizomeraza IV, Microbiology in the medical area, Bakterije, antibacterial activity, SDG 3 - Good Health and Well-being, inhibitors, Drug Discovery, Mikrobiologi inom det medicinska området, genetics, antibakterijsko delovanje, bacteria, zaviralci, Bakterijska rezistenca, Läkemedelskemi, antibacterial activity, bacteria, inhibitors, udc:615, inhibition, bakterije, farmacevtska kemija, Molecular Medicine, Medicinal Chemistry, udc:615.015.8
وصف الملف: application/pdf; text/url
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المؤلفون: Nadilly Bonagas, Nina Gustafsson, Martin Henriksson, Petra Marttila, Robert Gustafsson, Elisée Wiita, Sanjay Borhade, Alanna Green, Karl Vallin, Antonio Sarno, Richard Svensson, Camilla Göktürk, Therese Pham, Ann-Sofie Jemth, Olga Loseva, Victoria Cookson, Nicole Kiweler, Lars Sandberg, Azita Rasti, Judith Unterlass, Martin Haraldsson, Yasmin Andersson, Emma Scaletti, Christoffer Bengtsson, Cynthia Paulin, Kumar Sanjiv, Eldar Abdurakhmanov, Linda Pudelko, Ben Kunz, Matthieu Desroses, Petar Iliev, Katarina Färnegårdh, Andreas Krämer, Neeraj Garg, Maurice Michel, Sara Häggblad, Malin Jarvius, Christina Kalderén, Amanda Bögedahl Jensen, Ingrid Almlöf, Stella Karsten, Si Min Zhang, Maria Häggblad, Anders Eriksson, Jianping Liu, Björn Glinghammar, Natalia Nekhotiaeva, Fredrik Klingegård, Tobias Koolmeister, Ulf Martens, Sabin Llona-Minguez, Ruth Moulson, Helena Nordström, Vendela Parrow, Leif Dahllund, Birger Sjöberg, Irene Vargas, Duy Duc Vo, Johan Wannberg, Stefan Knapp, Hans Krokan, Per Arvidsson, Martin Scobie, Johannes Meiser, Pål Stenmark, Ulrika Warpman Berglund, Evert Homan, Thomas Helleday
مصطلحات موضوعية: hemic and lymphatic diseases
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::032514cb5181fdda8fdfefd73848c5d0
https://doi.org/10.21203/rs.3.pex-1730/v1 -
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المؤلفون: Richard C. Scarpulla, Björn Glinghammar, Johan Mattsson, Ulf Andersson, Tor Svensson, Thomas Naessens, Marcin Buler, Lillevi Kärrberg, Yannick Morias, Petra Thulin, Philip Robbins, Magnus Söderberg
المصدر: FASEB BioAdvances
FASEB BioAdvances, Vol 2, Iss 8, Pp 453-463 (2020)مصطلحات موضوعية: Cancer Research, animal structures, Physiology, Inflammation, PPRC1, Biochemistry, Genetics and Molecular Biology (miscellaneous), Coactivator, medicine, cytokine expression, STAT1, lcsh:QH301-705.5, Research Articles, Liver injury, Gene knockdown, CD40, hepatic inflammation, biology, Chemistry, Monocyte, medicine.disease, Cell biology, medicine.anatomical_structure, lcsh:Biology (General), biology.protein, STAT protein, Molecular Medicine, medicine.symptom, drug‐induced liver injury, PRC, Research Article
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المؤلفون: Björn Dahl, Björn Glinghammar, Krister Bamberg, Petra Thulin, Marcin Buler
المصدر: International Journal of Molecular Medicine. 38:961-968
مصطلحات موضوعية: Male, 0301 basic medicine, Blotting, Western, Gene Expression, Peroxisome proliferator-activated receptor, Biology, Xenobiotics, 03 medical and health sciences, 0302 clinical medicine, Species Specificity, Cell Line, Tumor, Sequence Homology, Nucleic Acid, Genetics, medicine, Animals, Humans, PPAR alpha, Luciferase, Amino Acid Sequence, Sulfones, Rats, Wistar, Luciferases, Promoter Regions, Genetic, Cells, Cultured, chemistry.chemical_classification, Liver injury, Reporter gene, Base Sequence, Sequence Homology, Amino Acid, Oncogene, Alanine Transaminase, Promoter, General Medicine, medicine.disease, Molecular biology, 030104 developmental biology, chemistry, 030220 oncology & carcinogenesis, Toxicity, Hepatocytes, Female, Propionates, Alanine Aminotransferase 1
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المؤلفون: Tommy B. Andersson, Gabriella Brolén, Anna Jonebring, Johanna Sagemark, Xue-Qing Li, Björn Glinghammar, Anna-Karin Sjögren, Maria Liljevald, Ian A. Cotgreave
المصدر: Archives of Toxicology. 88:1427-1437
مصطلحات موضوعية: Male, Programmed cell death, Cell type, Health, Toxicology and Mutagenesis, Cellular differentiation, Foreskin, Induced Pluripotent Stem Cells, Cell, Apoptosis, Biology, Toxicology, Cell Line, Toxicity Tests, medicine, Humans, Staurosporine, Induced pluripotent stem cell, Cells, Cultured, Acetaminophen, Cryopreservation, Principal Component Analysis, Cell Differentiation, General Medicine, Fibroblasts, Cell biology, medicine.anatomical_structure, Hepatocytes, Hepatic stellate cell, Chemical and Drug Induced Liver Injury, medicine.drug
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المؤلفون: Björn Glinghammar, Getnet Yimer, Lars Lindquist, B. Kevin Park, Gunnar Nordahl, Eyasu Makonnen, Alison H. Harrill, Paul B. Watkins, Marcus Gry, Ina Schuppe-Koistinen, Stig Linder, Björn Ekblom, Daniel J. Antoine, Petra Thulin, Eleni Aklillu, Getachew Aderaye, C. Mikael Mattsson
المصدر: Liver International. 34:367-378
مصطلحات موضوعية: Drug, Liver injury, Keratin-18, Hepatology, business.industry, media_common.quotation_subject, Alanine Transaminase, Enzyme-Linked Immunosorbent Assay, Gold standard (test), Pharmacology, medicine.disease, Sensitivity and Specificity, Peptide Fragments, Keratin 18, Cohort Studies, MicroRNAs, microRNA, Humans, Medicine, Chemical and Drug Induced Liver Injury, Alanine aminotransferase, business, Biomarkers, Predictive biomarker, media_common