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المؤلفون: Shu Fu Lin, Li-Wei Teng, Ya-Chi Huang, Shyh-Fong Chen, Guan-Ru Huang, Chih-Lin Chang, Pi-Chen Hsu, Min-Sian Huang, Yu-Sheng Gao, Ya-Wen Chan, Jiann-Jyh Huang, Sheng-Chuan Yang, Bo-Han Jian, Yann-Yu Lu, Yu-Fen Chen, Tzu-Hao Lo, Shih-Hsien Chuang, Wen-Yun Hsueh, Po-Hsun Huang, Hsin-Yi Huang, Lien-Hsiang Chang, Win-Yin Wei, Ying-Chou Chen, Her-Sheng Lin, Shan-Yen Chou, Ta-Tung Yuan, Yu-Ting Chao, Ying-Shuan E. Lee, Yi-Feng Kao, Yu-Hsiang Lin, Jo-Chu Lin, Hung-Huang Liu, Shao-Yun Wang, Chin-Hung Lai, Shin-Yi Huang
المصدر: Journal of Medicinal Chemistry. 64:1435-1453
مصطلحات موضوعية: 0303 health sciences, biology, Nitrile, Stereochemistry, Topoisomerase, Substrate (chemistry), 01 natural sciences, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, chemistry.chemical_compound, Cascade reaction, chemistry, Mechanism of action, Docking (molecular), Drug Discovery, biology.protein, medicine, Molecular Medicine, Structure–activity relationship, Dimethylformamide, medicine.symptom, 030304 developmental biology
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المؤلفون: Wen-Yun, Hsueh, Ying-Shuan E, Lee, Min-Sian, Huang, Chin-Hung, Lai, Yu-Sheng, Gao, Jo-Chu, Lin, Yu-Fen, Chen, Chih-Lin, Chang, Shan-Yen, Chou, Shyh-Fong, Chen, Yann-Yu, Lu, Lien-Hsiang, Chang, Shu Fu, Lin, Yu-Hsiang, Lin, Pi-Chen, Hsu, Win-Yin, Wei, Ya-Chi, Huang, Yi-Feng, Kao, Li-Wei, Teng, Hung-Huang, Liu, Ying-Chou, Chen, Ta-Tung, Yuan, Ya-Wen, Chan, Po-Hsun, Huang, Yu-Ting, Chao, Shin-Yi, Huang, Bo-Han, Jian, Hsin-Yi, Huang, Sheng-Chuan, Yang, Tzu-Hao, Lo, Guan-Ru, Huang, Shao-Yun, Wang, Her-Sheng, Lin, Shih-Hsien, Chuang, Jiann-Jyh, Huang
المصدر: Journal of medicinal chemistry. 64(3)
مصطلحات موضوعية: Male, Models, Molecular, Mice, Nude, Antineoplastic Agents, Quinolones, Xenograft Model Antitumor Assays, Catalysis, Rats, Molecular Docking Simulation, Rats, Sprague-Dawley, Mice, Structure-Activity Relationship, DNA Topoisomerases, Type I, Drug Design, Nitriles, Animals, Humans, Female, Drug Screening Assays, Antitumor, Topoisomerase I Inhibitors, Copper