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1دورية أكاديمية
المؤلفون: Maria Luisa Introvigne, Trevor J. Beardsley, Micah C. Fernando, David A. Leonard, Bradley J. Wallar, Susan D. Rudin, Magdalena A. Taracila, Philip N. Rather, Jennifer M. Colquhoun, Shaina Song, Francesco Fini, Kristine M. Hujer, Andrea M. Hujer, Fabio Prati, Rachel A. Powers, Robert A. Bonomo, Emilia Caselli
المصدر: Antibiotics, Vol 12, Iss 4, p 644 (2023)
مصطلحات موضوعية: antibiotic resistance, β-lactamases, Acinetobacter baumannii, boronic acids, cross-class inhibitors, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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المؤلفون: Sara J. Barlow, Robert A. Bonomo, Rachel A. Powers, Fabio Prati, Kali A. Smolen, Magdalena A. Taracila, Bradley J. Wallar, Emilia Caselli, Brandy N. Curtis
المصدر: Antimicrob Agents Chemother
مصطلحات موضوعية: Stereochemistry, Ceftazidime, beta-Lactamases, 03 medical and health sciences, Hydrolysis, chemistry.chemical_compound, Transition state analog, Mechanisms of Resistance, Amide, medicine, Side chain, Pharmacology (medical), Acinetobacter, Acinetobacter baumannii, boronic acid transition state analog inhibitor, ceftazidime, cephalosporinase, lactamase, 030304 developmental biology, Cephalosporinase, Pharmacology, 0303 health sciences, 030306 microbiology, Hydrogen bond, Boronic Acids, Anti-Bacterial Agents, Infectious Diseases, chemistry, Oxyanion hole, beta-Lactamase Inhibitors, Boronic acid, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::48bf2b0fb3eb0a52d0b3f34fb1ae5132
https://pubmed.ncbi.nlm.nih.gov/32988830 -
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المؤلفون: Emilia, Caselli, Francesco, Fini, Maria Luisa, Introvigne, Mattia, Stucchi, Magdalena A, Taracila, Erin R, Fish, Kali A, Smolen, Philip N, Rather, Rachel A, Powers, Bradley J, Wallar, Robert A, Bonomo, Fabio, Prati
المصدر: ACS Infectious Diseases
مصطلحات موضوعية: Acinetobacter baumannii, Structure-Activity Relationship, boronic acids, Acinetobacter, β-lactamase inhibitors, click chemistry, amide bioisostere, beta-Lactamase Inhibitors, beta-Lactamases, Article, Cephalosporinase
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المؤلفون: Bradley J. Wallar, Rachel A. Powers, Francesco Fini, Philip N. Rather, Fabio Prati, Erin R. Fish, Maria Luisa Introvigne, Robert A. Bonomo, Mattia Stucchi, Kali A. Smolen, Magdalena A. Taracila, Emilia Caselli
مصطلحات موضوعية: 0301 basic medicine, Amide binding, boronic acids, Acinetobacter, Stereochemistry, β-lactamase inhibitors, 030106 microbiology, Triazole, amide bioisostere, Enzyme binding, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, Infectious Diseases, chemistry, Amide, click chemistry, Side chain, Structure–activity relationship, Bioisostere, Boronic acid
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::216e83087d08f3162ebae8cbb64b0670
https://hdl.handle.net/11380/1208053 -
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المؤلفون: Thomas H. Clarke, Derrick E. Fouts, Magdalena A. Taracila, Pratap Venepally, David A. Leonard, Bradley J. Wallar, Paul G. Higgins, Rachel A. Powers, Philip N. Rather, Lauren Brinkac, Robert A. Bonomo, Steven H. Marshall, Andrew R Mack, Kristine M. Hujer, Barry N. Kreiswirth, Fabio Prati, Christopher Greco, Emilia Caselli, Andrea M. Hujer
المصدر: Diagnostic Microbiology and Infectious Disease
مصطلحات موضوعية: Acinetobacter baumannii, 0301 basic medicine, Microbiology (medical), 030106 microbiology, OXA carbapenemase, beta-Lactam Resistance, beta-Lactamases, Microbiology, carbapenemase, 03 medical and health sciences, 0302 clinical medicine, Bacterial Proteins, Carbapenem resistant Acinetobacter baumannii, Humans, 030212 general & internal medicine, Allele, OXA β-lactamase, OXA-23, biology, OXA-82, β lactamases, ADC β-lactamase, OXA-172, General Medicine, Antimicrobial, biology.organism_classification, Infectious Diseases, Carbapenems, Original Article, carbapenem resistant Acinetobacter baumannii, Genome, Bacterial, Acinetobacter Infections
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c3b5484c7966f3e402e6bf859770e686
https://doi.org/10.1016/j .diagmicrobio.2020.115242 -
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المؤلفون: Rachel A. Powers, Kali A. Smolen, Fabio Prati, Alexandra A. Bouza, Magdalena A. Taracila, Emilia Caselli, Robert A. Bonomo, Francesco Fini, Hollister C. Swanson, Bradley J. Wallar, Chiara Romagnoli
مصطلحات موضوعية: 0301 basic medicine, Models, Molecular, carboxylate, Stereochemistry, Protein Conformation, boronic acid, 030106 microbiology, Crystallography, X-Ray, Article, 03 medical and health sciences, chemistry.chemical_compound, Amide, Structure–activity relationship, Carboxylate, Cephalosporinase, Binding Sites, biology, Acinetobacter, Molecular Structure, Chemistry, enzyme plasticity, Active site, structure activity relationship study, structure activity relationship, β-lactamase, biology.organism_classification, Boronic Acids, click chemistry, Infectious Diseases, 030104 developmental biology, biology.protein, Click chemistry, beta-Lactamase Inhibitors, Lead compound, Boronic acid, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f75682e8ee3ed7686321fca1b7b6a5ad
https://europepmc.org/articles/PMC5987196/ -
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المؤلفون: Rachel A. Powers, Chiara Romagnoli, Kali A. Smolen, Magdalena A. Taracila, Fabio Prati, Hollister C. Swanson, Emilia Caselli, Robert A. Bonomo, Alison L. VanDine, Alexandra A. Bouza, Bradley J. Wallar
المصدر: ACS infectious diseases. 4(3)
مصطلحات موضوعية: 0301 basic medicine, Models, Molecular, Circular dichroism, Stereochemistry, Protein Conformation, ADC-7, Acinetobacter, boronic acid, cephalosporinase, transition state analog inhibitors, β-lactamase, 030106 microbiology, Crystallography, X-Ray, Article, 03 medical and health sciences, chemistry.chemical_compound, Transition state analog, Beta-Lactamase Inhibitors, Cephalosporinase, Trifluoromethyl, Binding Sites, biology, Chemistry, Circular Dichroism, biology.organism_classification, Boronic Acids, Acinetobacter baumannii, Multiple drug resistance, body regions, 030104 developmental biology, Infectious Diseases, Biochemistry, beta-Lactamase Inhibitors, Boronic acid, Protein Binding
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المؤلفون: Nicholas W. Florek, Emilia Caselli, Hollister C. Swanson, Robert A. Bonomo, Bradley J. Wallar, Fabio Prati, Magdalena A. Taracila, Rachel A. Powers, Chiara Romagnoli
المصدر: Biochemistry
مصطلحات موضوعية: Acinetobacter baumannii, Models, Molecular, antibiotic resistance, boronic acids, medicine.drug_class, Stereochemistry, medicine.medical_treatment, Static Electricity, Cephalosporin, Crystallography, X-Ray, Biochemistry, Biophysical Phenomena, beta-Lactam Resistance, Article, BETA-LACTAMASE, chemistry.chemical_compound, Bacterial Proteins, Catalytic Domain, Acinetobacter baumanii, Hydrolase, Antimicrobial chemotherapy, medicine, Beta-Lactamase Inhibitors, Cephalosporinase, chemistry.chemical_classification, Molecular Structure, biology, biology.organism_classification, Boronic Acids, body regions, Kinetics, Enzyme, chemistry, Drug Design, Beta-lactamase, Thermodynamics, beta-Lactamase Inhibitors, Boronic acid
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المؤلفون: Jessica A. Schoenherr, Susan M. Kitchen, Brittany N. Stropich, Holly A. Holman, Arthur S. Alberts, Bradley J. Wallar
المصدر: Journal of Biological Chemistry. 281:4300-4307
مصطلحات موضوعية: Molecular Sequence Data, Formins, macromolecular substances, GTPase, Inhibitory postsynaptic potential, Biochemistry, Mice, Animals, Homeostasis, Amino Acid Sequence, Cytoskeleton, Molecular Biology, Actin, chemistry.chemical_classification, biology, Effector, NADPH Dehydrogenase, Cell Biology, Actins, Protein Structure, Tertiary, Amino acid, Cell biology, Crystallography, chemistry, NIH 3T3 Cells, biology.protein, Carrier Proteins, Microtubule-Associated Proteins
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::f19afad71cfa77aaaf6dcd6934613999
https://doi.org/10.1074/jbc.m510277200 -
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المؤلفون: Philippe Chavrier, Jun Peng, Florence Niedergang, Bradley J. Wallar, Emma Colucci-Guyon, Arthur S. Alberts
المصدر: Current Biology. 15:2007-2012
مصطلحات موضوعية: Phagocytic cup, RHOA, Phagocytosis, Blotting, Western, Fluorescent Antibody Technique, Formins, Macrophage-1 Antigen, chemical and pharmacologic phenomena, macromolecular substances, Complement receptor, General Biochemistry, Genetics and Molecular Biology, Cell Line, Mice, 03 medical and health sciences, Animals, RNA, Small Interfering, 030304 developmental biology, 0303 health sciences, Agricultural and Biological Sciences(all), biology, Biochemistry, Genetics and Molecular Biology(all), Effector, Macrophages, 030302 biochemistry & molecular biology, hemic and immune systems, Actins, Cell biology, Macrophage-1 antigen, Microscopy, Electron, Scanning, biology.protein, MDia1, Carrier Proteins, General Agricultural and Biological Sciences