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1
المؤلفون: Thomas Hollenbeck, Christine Tumanut, Donald S. Karanewsky, Robert Epple, Michael J. Roberts, Hong Liu, Michael Hornsby, Glen Spraggon, David H. Woodmansee, Brian T. Masick, Tove Tuntland, Jonathan Chang, David C. Tully, Jun Li, Jennifer A. Williams, Jennifer L. Harris, Phil B. Alper, Perry Gordon, Arnab K. Chatterjee
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:5112-5117
مصطلحات موضوعية: Male, Stereochemistry, Peptidomimetic, Clinical Biochemistry, Administration, Oral, Biological Availability, Pharmaceutical Science, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Ethers, Cyclic, Amide, Drug Discovery, Animals, Humans, Protease Inhibitors, Rats, Wistar, Molecular Biology, Cathepsin S, chemistry.chemical_classification, Binding Sites, Molecular Structure, biology, Organic Chemistry, Aromatic amine, Active site, Amides, Cathepsins, Rats, Zinc, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Molecular Medicine
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2
المؤلفون: Nicholas James Devereux, Anne-Marie D’Souza, Valerie Boissel, Vidal Agnes, Mark Nash, Ardem Patapoutian, Ryan West, J. Martin Verkuyl, Andrew M. Schumacher, Brian T. Masick, Victoria Head, H. Michael Petrassi, Rowan Stringer, Lisa Ann Rooney, Natalie Stoakley, Moh Panesar, David C. Tully, Jianmin Lao, Matt Petrus
المصدر: Journal of medicinal chemistry. 57(12)
مصطلحات موضوعية: Male, Indazoles, Stereochemistry, Freund's Adjuvant, Anti-Inflammatory Agents, Administration, Oral, Biological Availability, Nerve Tissue Proteins, CHO Cells, Ring (chemistry), chemistry.chemical_compound, Structure-Activity Relationship, Cricetulus, Transient Receptor Potential Channels, Species Specificity, In vivo, Drug Discovery, Animals, Humans, Plant Oils, Rats, Wistar, IC50, TRPA1 Cation Channel, TRPC Cation Channels, Indazole, Analgesics, Trifluoromethyl, Antagonist, Hit to lead, In vitro, Mice, Inbred C57BL, chemistry, Hyperalgesia, Molecular Medicine, Calcium Channels, Mustard Plant
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3
المؤلفون: Jennifer L. Harris, Takashi Nakai, Jun Li, Bradley J. Backes, H. Michael Petrassi, Christine Tumanut, Brian T. Masick, Jennifer A. Williams, Jared Ek
المصدر: Bioorganicmedicinal chemistry letters. 15(12)
مصطلحات موضوعية: Models, Molecular, Proteases, Proteolysis, medicine.medical_treatment, Clinical Biochemistry, Molecular Sequence Data, Pharmaceutical Science, Cleavage (embryo), Biochemistry, Substrate Specificity, Serine, Thrombin, Coumarins, Drug Discovery, medicine, Combinatorial Chemistry Techniques, Humans, Computer Simulation, Amino Acid Sequence, Threonine, Molecular Biology, Fluorescent Dyes, Protease, medicine.diagnostic_test, Chemistry, Caspase 3, Organic Chemistry, Caspases, Molecular Medicine, Oligopeptides, medicine.drug, Cysteine