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1
المؤلفون: Renato Skerlj, Tuya Ba, Ernest J. McEachern, Elyse Bourque, Ian Baird, Dominique Schols, Wilson Trevor R, Renee Mosi, Jonathan Langille, Yuanxi Zhou, Bryon Carpenter, Michael Bey, Simon P. Fricker, Dana Huskens, Duane Veale, Rebecca S.Y. Wong, Gary Bridger, Curtis Harwig, Veronique Bodart, Ron MacFarland, Markus Metz, Sanjay Danthi
المصدر: ACS Medicinal Chemistry Letters. 3:216-221
مصطلحات موضوعية: congenital, hereditary, and neonatal diseases and abnormalities, biology, business.industry, Purkinje fibers, Organic Chemistry, hERG, Human immunodeficiency virus (HIV), Pharmacology, medicine.disease_cause, Biochemistry, Bioavailability, Chemokine receptor, medicine.anatomical_structure, Drug Discovery, Lipophilicity, biology.protein, Medicine, Action potential duration, cardiovascular diseases, business, Ion channel
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2
المؤلفون: Renato T. Skerlj, Jason B. Crawford, Gary Bridger, Wilson Trevor R, Jenny Ji, Bryon Carpenter, Gang Chen
المصدر: Organic Process Research & Development. 16:109-116
مصطلحات موضوعية: Stereochemistry, Longest linear sequence, Chemistry, Organic Chemistry, CCR5 receptor antagonist, Physical and Theoretical Chemistry, Laboratory scale, Combinatorial chemistry
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3
المؤلفون: Tong-Shuang Li, Simon P. Fricker, Gang Chen, Renato Skerlj, David Bogucki, Markus Metz, Gary Bridger, Susan Nan, Rebecca S.Y. Wong, Dominique Schols, Jean Labrecque, Gloria Lau, Marilyn C. Darkes, Bryon Carpenter
المصدر: Virology. 413(2):231-243
مصطلحات موضوعية: Models, Molecular, Receptors, CCR5, Protein Conformation, Vicriviroc, viruses, Aplaviroc, Drug design, CCR5 receptor antagonist, Computational biology, Biology, Maraviroc, chemistry.chemical_compound, HIV Fusion Inhibitors, Virology, High-Throughput Screening Assays, medicine, Homology modeling, Binding site characterization, virus diseases, Reproducibility of Results, Stereoisomerism, Virus Internalization, Molecular biology, Small molecule, Small molecule antagonists, Antifusogenic assay, chemistry, Mutagenesis, CCR5 Receptor Antagonists, Mutation, HIV-1, Mutagenesis, Site-Directed, CCR5, medicine.drug
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4
المؤلفون: Jason B. Crawford, Gang Chen, Ernie Mceachern, Gary Bridger, Curtis Harwig, Atsma Bern, Alan Kaller, Renato Skerlj, Ian Baird, Wilson Trevor R, Bryon Carpenter, David Gauthier
المصدر: Organic Process Research & Development. 12:823-830
مصطلحات موضوعية: Organic Chemistry, Imine, chemistry.chemical_element, Zinc, Borohydride, CXCR4, Reductive amination, Chemokine Receptor Antagonist, chemistry.chemical_compound, Sodium borohydride, chemistry, Reagent, Organic chemistry, Physical and Theoretical Chemistry
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5
المؤلفون: Curtis Harwig, Dominique Schols, Gang Chen, Wen Yang, Duane Veale, Susan Nan, Simon P. Fricker, Alan Kaller, Danielle Guay, Jason M. Crawford, Michael Satori, Markus Metz, Yongbao Zhu, Helen Yee, Maria Krumpak, Elyse Bourque, Wilson Trevor R, David Bogucki, Bryon Carpenter, Michael Bey, David C. Leitch, Ron MacFarland, David Gauthier, Ian Baird, Rebecca Wong, Renato T. Skerlj, Jonathan Langille, Yuanxi Zhou, Gary Bridger, Renee Mosi, Ernest J. McEachern, Tuya Ba, Tong-Shuang Li, Krystyna Vocadlo, Veronique Bodart
المصدر: Journal of medicinal chemistry. 56(20)
مصطلحات موضوعية: Receptors, CCR5, Anti-HIV Agents, Cell Survival, hERG, Human immunodeficiency virus (HIV), CHO Cells, Pharmacology, medicine.disease_cause, Imidazolidines, Virus Replication, Benzoates, Chemokine receptor, Structure-Activity Relationship, Cricetulus, Piperidines, In vivo, Cricetinae, Drug Discovery, medicine, Animals, Humans, Cells, Cultured, Cardiotoxicity, biology, Molecular Structure, Chemistry, Imidazoles, In vitro, Receptor selectivity, HEK293 Cells, Biochemistry, Models, Chemical, Drug Design, Lipophilicity, CCR5 Receptor Antagonists, Host-Pathogen Interactions, biology.protein, HIV-1, Leukocytes, Mononuclear, Molecular Medicine
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6دورية أكاديمية
المؤلفون: Jason B. Crawford, Gang Chen, Bryon Carpenter, Trevor Wilson, Jenny Ji, Renato T. Skerlj, Gary J. Bridger
المصدر: Organic Process Research & Development; Jan2012, Vol. 16 Issue 1, p109-116, 8p