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1دورية أكاديمية
المؤلفون: Brent R. Lyda, Gregory P. Leary, Jill Farnsworth, Benjamin Seaver, Derek Silvius, Michael P. Kavanaugh, C. Sean Esslinger, Nicholas R. Natale
المصدر: Molecules, Vol 29, Iss 10, p 2330 (2024)
مصطلحات موضوعية: solute carrier superfamily (SLC), alkoxy hydroxy-pyrrolidine carboxylic acids (AHPCs), computational homology model, SLC1A4 (ASCT1), SLC1A5 (ASCT2), electrophysiology, Organic chemistry, QD241-441
وصف الملف: electronic resource
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المؤلفون: Brent R. Lyda, Gregory P. Leary, Jill Farnsworth, Derek Silvius, Benjamin Seaver, C. Sean Esslinger, Nicholas R. Natale, Michael P. Kavanaugh
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::16821e2ba966c8cf06206d75570da98d
https://doi.org/10.1101/2021.12.14.470456 -
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المؤلفون: Ben Seaver, Mariusz P. Gajewski, C. Sean Esslinger
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:4163-4166
مصطلحات موضوعية: Models, Molecular, Stereochemistry, Xenopus, Clinical Biochemistry, Triazole, Pharmaceutical Science, Endogeny, Ligands, Biochemistry, Article, chemistry.chemical_compound, Drug Discovery, Neutral amino acid transport, Side chain, Animals, Amino Acids, Molecular Biology, chemistry.chemical_classification, Hydrogen bond, Organic Chemistry, Hydrogen Bonding, Biological activity, General Medicine, Triazoles, Ligand (biochemistry), Rats, Amino acid, Amino Acid Transport Systems, Neutral, chemistry, Molecular Probes, Molecular Medicine
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المؤلفون: Michael P. Kavanaugh, Erin O’Brien, Shailesh Agarwal, Joseph F. Rhoderick, A. Richard Chamberlin, C. Sean Esslinger, Richard J. Bridges, Hans P. Koch, John M. Gerdes, Alicia N. Awes, Erin S. Davis, David J. Poulsen, Teri Mavencamp, Paul A. Wilson
المصدر: Neuropharmacology. 49:850-861
مصطلحات موضوعية: Models, Molecular, Neurotransmitter transporter, Patch-Clamp Techniques, Stereochemistry, Amino Acid Transport System X-AG, Xenopus, Gene Expression, Context (language use), Transfection, Tritium, Membrane Potentials, Mice, Cellular and Molecular Neuroscience, Animals, Cell Line, Transformed, Neurons, Pharmacology, chemistry.chemical_classification, Aspartic Acid, Dose-Response Relationship, Drug, biology, Glutamate receptor, Transporter, biology.organism_classification, Electric Stimulation, Amino acid, Excitatory Amino Acid Transporter 1, Excitatory Amino Acid Transporter 3, Excitatory Amino Acid Transporter 2, chemistry, Biochemistry, Oocytes, Excitatory postsynaptic potential, Pharmacophore
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المؤلفون: Richard J. Bridges, C. Sean Esslinger
المصدر: Pharmacology & Therapeutics. 107:271-285
مصطلحات موضوعية: Central Nervous System, Pharmacology, chemistry.chemical_classification, Glutamate receptor, Glutamic Acid, AMPA receptor, Biology, Neurotransmission, Synaptic Transmission, Amino acid, Glutamate Plasma Membrane Transport Proteins, chemistry, Biochemistry, Excitatory Amino Acid Agonists, Excitatory postsynaptic potential, Animals, Humans, NMDA receptor, Pharmacology (medical), Synaptic signaling, Receptor, Excitatory Amino Acid Antagonists
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المؤلفون: R D Bartlett, Charles M. Thompson, Christina N. Carrigan, C. Sean Esslinger, Kimberly A. Cybulski, Richard J. Bridges, Pakamas Tongcharoensirikul
المصدر: Journal of Medicinal Chemistry. 45:2260-2276
مصطلحات موضوعية: Male, Telencephalon, Glutamic Acid, In Vitro Techniques, Synaptic vesicle, Chemical synthesis, Rats, Sprague-Dawley, Structure-Activity Relationship, chemistry.chemical_compound, ATP hydrolysis, Drug Discovery, Animals, Neurotransmitter, chemistry.chemical_classification, Quinoline, Glutamate receptor, In vitro, Rats, Kinetics, Dicarboxylic acid, chemistry, Biochemistry, Quinolines, Molecular Medicine, Synaptic Vesicles, Carrier Proteins
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المؤلفون: Michael P. Kavanaugh, Richard J. Bridges, Charles M. Thompson, C. Sean Esslinger, A. Richard Chamberlin, Hans P. Koch, Dean P. Philips
المصدر: ChemInform. 30
مصطلحات موضوعية: biology, Biochemistry, Excitatory amino-acid transporter, Chemistry, biology.protein, General Medicine
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مصطلحات موضوعية: Models, Molecular, Magnetic Resonance Spectroscopy, Molecular model, Stereochemistry, Clinical Biochemistry, Excitatory Amino Acid Transporter 3, Pharmaceutical Science, Biochemistry, Chemical synthesis, Article, Mass Spectrometry, Cell Line, Structure-Activity Relationship, Drug Discovery, Aspartic acid, Structure–activity relationship, Animals, Binding site, Molecular Biology, Neurons, Aspartic Acid, Chemistry, Organic Chemistry, Glutamate receptor, Molecular Medicine, Pharmacophore
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::c30b9135ca6d48f59928b3f3259c335a
https://europepmc.org/articles/PMC2631431/ -
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المصدر: Bioorganicmedicinal chemistry. 10(11)
مصطلحات موضوعية: Neurotransmitter transporter, Models, Molecular, Pyrrolidines, Molecular model, Stereochemistry, Amino Acid Transport System X-AG, Clinical Biochemistry, Carboxylic Acids, Molecular Conformation, Pharmaceutical Science, macromolecular substances, In Vitro Techniques, Biochemistry, Methylation, Pyrrolidine, chemistry.chemical_compound, Prosencephalon, Drug Discovery, medicine, Animals, Dicarboxylic Acids, Molecular Biology, Chemistry, Organic Chemistry, Glutamate receptor, Substrate (chemistry), Computational Biology, hemic and immune systems, Membrane transport, Transport inhibitor, Rats, Kinetics, Mechanism of action, Excitatory Amino Acid Transporter 2, Models, Chemical, Cyclization, Molecular Medicine, Indicators and Reagents, medicine.symptom, Synaptosomes
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المؤلفون: Hans P. Koch, A. Richard Chamberlin, C. Sean Esslinger, Michael P. Kavanaugh, Dean P. Philips, Charles M. Thompson, Richard J. Bridges
المصدر: Bioorganicmedicinal chemistry letters. 8(21)
مصطلحات موضوعية: Male, Pyrrolidines, Intramolecular reaction, Stereochemistry, Amino Acid Transport System X-AG, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Glutamic Acid, Biochemistry, Chemical synthesis, Pyrrolidine, Rats, Sprague-Dawley, chemistry.chemical_compound, Drug Discovery, Animals, Dicarboxylic Acids, Molecular Biology, Bicyclic molecule, Organic Chemistry, Glutamate receptor, Substrate (chemistry), Glutamic acid, Rats, chemistry, Intramolecular force, Molecular Medicine, ATP-Binding Cassette Transporters