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المؤلفون: Fulci, C, Rotili, Dante, De Luca, A, Stella, L, Morozzo Della Rocca, B, Forgione, M, Di Paolo, V, Mai, Antonello, Falconi, M, Quintieri, L, Caccuri, Am, 7, .
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 32, Iss 1, Pp 240-247 (2017)
Europe PubMed Central
Journal of Enzyme Inhibition and Medicinal Chemistryمصطلحات موضوعية: Models, Molecular, 0301 basic medicine, TRAF2, Tripeptide, GSTP1, chemistry.chemical_compound, 0302 clinical medicine, Models, Drug Discovery, GSTP1-1, Enzyme Inhibitors, Oxazoles, Ultraviolet, Tumor, Chemistry, General Medicine, Biochemistry, Spectrophotometry, 030220 oncology & carcinogenesis, medicine.symptom, Lead compound, Research Article, Stereochemistry, In silico, NBDHEX, Enzyme-Linked Immunosorbent Assay, Fluorescence, Cell Line, GSH, nitrobenzoxadiazoles, 03 medical and health sciences, Cell Line, Tumor, medicine, Humans, Nitrobenzoxadiazoles, Glutathione S-Transferase pi, Spectrometry, Fluorescence, Spectrophotometry, Ultraviolet, Pharmacology, Drug Discovery3003 Pharmaceutical Science, Settore BIO/10, Spectrometry, lcsh:RM1-950, Molecular, Glutathione, In vitro, 030104 developmental biology, lcsh:Therapeutics. Pharmacology, Mechanism of action
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المؤلفون: De Luca, A, Rotili, D, Carpanese, D, Lenoci, A, Calderan, L, Scimeca, M, Mai, A, Bonanno, E, Rosato, A, Geroni, C, Quintieri, L, Caccuri, Am, DE LUCA, A
المصدر: Scopus-Elsevier
Europe PubMed Central
Oncotargetمصطلحات موضوعية: Oral, Administration, Oral, Apoptosis, Human Melanoma Xenografts, Pharmacology, Settore MED/08 - Anatomia Patologica, Cell Line, chemistry.chemical_compound, Mice, Random Allocation, c-Jun N-terminal Kinase, Animals, Cell Line, Tumor, Cell Proliferation, Enzyme Inhibitors, Female, Glutathione S-Transferase pi, Humans, Melanoma, Oxadiazoles, Xenograft Model Antitumor Assays, In vivo, Settore BIO/10, Glutathione Transferase P1-1, 6-((7-nitrobenzo[c][1,2,5]oxadiazoles, Tumor, Chemistry, Cell growth, Glutathione, In vitro, Oncology, Cell culture, Settore CHIM/09 - Farmaceutico Tecnologico Applicativo, Administration, Target protein, Research Paper
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::83de4a0b9e91142fc8eb82414bab32fc
http://hdl.handle.net/11577/3181848 -
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المؤلفون: DE LUCA, A, Graziani, G, Rotili, D, Muzi, A, Mai, A, Leonetti, C, Artuso, S, Bonanno, E, Tentori, L, Caccuri, Am
مصطلحات موضوعية: Settore BIO/14
URL الوصول: https://explore.openaire.eu/search/publication?articleId=od______3667::d80080a31b3ac6dd7d24da9e5d68fc5c
http://hdl.handle.net/2108/170908 -
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المؤلفون: DE MARIA F, PEDERSEN JZ, CACCURI AM, TURELLA P, STELLA L, LO BELLO M, FEDERICI G, RICCI G., ANTONINI, GIOVANNI
المساهمون: DE MARIA, F, Pedersen, Jz, Caccuri, Am, Antonini, Giovanni, Turella, P, Stella, L, LO BELLO, M, Federici, G, Ricci, G.
مصطلحات موضوعية: Settore BIO/10
URL الوصول: https://explore.openaire.eu/search/publication?articleId=dedup_wf_001::30309d8fbb6357c5a3874d2b197d583b
http://hdl.handle.net/2108/100290 -
5
المؤلفون: Caccuri, Am, Antonini, G, Ascenzi, P, Nicotra, M, Nuccetelli, M, Mazzetti, A, Federici, G, LO BELLO, M, Ricci, G
المساهمون: Caccuri, Am, Antonini, Giovanni, Ascenzi, Paolo, Nicotra, M, Nuccetelli, M, Mazzetti, Ap, Federici, G, LO BELLO, M, Ricci, G.
المصدر: The Journal of biological chemistry. 274(27)
مصطلحات موضوعية: Models, Molecular, chemical, site-directed, physiological, adaptation, Adaptation, Physiological, Glutathione, Isoenzymes, models, Amino Acid Substitution, Glutathione S-Transferase pi, Models, Chemical, Mutagenesis, Site-Directed, mutagenesis, site-directed, glutathione s-transferase PI, models, molecular, glutathione, isoenzymes, glutathione transferase, tyrosine, models, chemical, adaptation, physiological, protein binding, amino acid substitution, Tyrosine, molecular, Settore BIO/10, mutagenesis, Glutathione Transferase, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::0162e66fcfcdbc1ab3a9bc85706b5b66
https://pubmed.ncbi.nlm.nih.gov/10383436 -
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المؤلفون: Pedersen, Jz, DE MARIA, F, Turella, P, Federici, G, Mattei, M, Fabrini, R, Dawood, Kf, Massimi, Mara, Caccuri, Am, Ricci, G.
مصطلحات موضوعية: Male, Rats, Sprague-Dawley, Glutathione S-Transferase pi, Iron, Hepatocytes, Animals, Humans, Nitrogen Oxides, Settore BIO/10, Nitric Oxide, Cells, Cultured, Glutathione Transferase, Rats
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::bd31e63af6a351b7118cbe44d7186f7e
http://hdl.handle.net/2108/21125 -
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المؤلفون: Caccuri AM, ASCENZI, Paolo, Parker MW, Oakley AJ, Chiessi E, Nuccetelli M, Battistoni A, Bellizia A, Ricci G., ANTONINI, GIOVANNI
المساهمون: Caccuri, Am, Ascenzi, Paolo, Antonini, Giovanni, Parker, Mw, Oakley, Aj, Chiessi, E, Nuccetelli, M, Battistoni, A, Bellizia, A, Ricci, G.
مصطلحات موضوعية: structural, isoenzymes, mathematics, binding sites, Models, Theoretical, recombinant proteins, Protein Structure, Secondary, Models, Structural, models, thermodynamics, dinitrochlorobenzene, kinetics, glutathione transferase, protein structure, glutathione, point mutation, Settore BIO/10, secondary, humans, theoretical, protein structure, secondary, models, structural, 4-chloro-7-nitrobenzofurazan, models, theoretical
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::52f625d00b06cf4c719aacd8be16dbcc
http://hdl.handle.net/2108/69223 -
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المؤلفون: Turella, P, Filomeni, G, Dupuis, M, Ciriolo, Mr, Molinari, A, De Maria, F, Tombesi, M, Cianfriglia, M, Federici, G, Ricci, G, Caccuri, Am
المصدر: The Journal of biological chemistry. 281(33)
مصطلحات موضوعية: Cytotoxicity, LC 50, Drug Resistance, Apoptosis, stress activated protein kinase, glycoprotein P, Piperazines, caspase 3, drug uptake, Enzyme Inhibitors, multidrug resistance protein 1, enzyme inhibition, Glutathione Transferase, 3 benzoxadiazol 4 ylthio)hexanol, Oxadiazoles, Tumor, Leukemia, Cell Death, article, transferase inhibitor, 6 (7 nitro 2, Drug Resistance, Multiple, unclassified drug, enzyme activity, Mitochondria, drug distribution, Membrane permeability, Phenotype, priority journal, Caspases, Acute Disease, Biomedical engineering, leukemia cell line, Multiple, drug transport, Leukemia, T-Cell, Cells, caspase, gene overexpression, Antineoplastic Agents, Tumor cells, Cell Line, in vivo study, Drug products, Enzyme inhibition, Patient treatment, Toxicity, Tumors, Leukemia cells, 6 (7 nitro 2,1,3 benzoxadiazol 4 ylthio)hexanol, glutathione transferase, glutathione transferase P1, apoptosis, cell death, controlled study, cytotoxicity, drug inhibition, drug mechanism, drug penetration, drug sensitivity, human, human cell, membrane permeability, protein expression, tumor cell line, tumor resistance, Biological Transport, Cell Line, Tumor, Drug Resistance, Neoplasm, Humans, Kinetics, P-Glycoprotein, ATP Binding Cassette Transporter, Subfamily B, Member 1, Settore BIO/10, T-Cell, Neoplasm
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::ab2d361d38d3a97b44882ca3d692ca78
https://pubmed.ncbi.nlm.nih.gov/16769721 -
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المؤلفون: Ricci, G, De Maria, F, Antonini, G, Turella, P, Bullo, A, Stella, L, Filomeni, G, Federici, G, Caccuri, Am
المصدر: The Journal of biological chemistry. 280(28)
مصطلحات موضوعية: Models, Molecular, Time Factors, Protein Conformation, Drug Resistance, Tumor cell lines, stress activated protein kinase, cancer cell culture, Spectroscopic analysis, enzyme inhibitor complex, Piperazines, Models, Suicide inhibitor, Enzyme Inhibitors, enzyme inhibition, antineoplastic agent, Glutathione Transferase, 3 benzoxadiazol 4 ylthio)hexanol, Microscopy, Oxadiazoles, Tumor, 6 mercapto 1 hexanol, glutathione transferase m2 2, glutathione transferase P1 1, apoptosis, article, Temperature, 7 nitro 2, Cells, Dissociation, Drug products, Molecules, Proteins, Tumors, Human glutathione S-transferases, Protein pumps, Derivatives, 6 (7 nitro 2,1,3 benzoxadiazol 4 ylthio)hexanol, 7 nitro 2,1,3 benzoxadiazole derivative, enzyme inhibitor, glutathione transferase, glutathione transferase A1, hexanol, multidrug resistance protein, oxadiazole derivative, thiol derivative, unclassified drug, dissociation, drug accumulation, drug conjugation, drug mechanism, drug structure, enzyme active site, enzyme binding, enzyme inhibitor interaction, human, human cell, IC 50, molecular stability, priority journal, spectroscopy, tumor cell, Antineoplastic Agents, Binding Sites, Cell Line, Tumor, Dose-Response Relationship, Drug, Drug Design, Drug Resistance, Multiple, Hexanols, Humans, K562 Cells, Kinetics, Microscopy, Fluorescence, Models, Chemical, Peptides, Protein Binding, Spectrometry, Fluorescence, Spectrophotometry, Sulfhydryl Compounds, 6 (7 nitro 2, Drug, Multiple, Chemical, Fluorescence, Cell Line, Dose-Response Relationship, Settore BIO/10, Spectrometry, Molecular, 3 benzoxadiazole derivative
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid_dedup__::dd08ce2e4c6b4a44eaf9b8cacb0e6c83
https://pubmed.ncbi.nlm.nih.gov/15888444