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المصدر: Inducing Targeted Protein Degradation. :313-336
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::69068f34af5e23613f10407689898f88
https://doi.org/10.1002/9783527836208.ch12 -
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المؤلفون: Janneke Keemink, Carina Cantrill, William Riboulet, Stella Jurmanović, Ivana Pavlovski, Caterina Bissantz
المصدر: Molecular Pharmaceutics.
مصطلحات موضوعية: Drug Discovery, Pharmaceutical Science, Molecular Medicine
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المؤلفون: Claudia Senn, Carina Cantrill, Holger Fischer, Franz Schuler, Li Yu, Mohammed Ullah
المصدر: Journal of Pharmacology and Experimental Therapeutics. 376:322-329
مصطلحات موضوعية: 0301 basic medicine, Drug Evaluation, Preclinical, Clinical Chemistry Tests, 03 medical and health sciences, 0302 clinical medicine, In vivo, Drug Discovery, Animals, ATP Binding Cassette Transporter, Subfamily B, Member 1, Transcellular, P-glycoprotein, Pharmacology, biology, Chemistry, Transporter, In vitro, Rats, Transport protein, Protein Transport, 030104 developmental biology, Permeability (electromagnetism), Biophysics, biology.protein, Molecular Medicine, Efflux, 030217 neurology & neurosurgery
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e4e159e338ca1c2160568d8fbd905d75
https://doi.org/10.1124/jpet.120.000158 -
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المؤلفون: Harvey J. Clewell, Thomas G. Osimitz, R.J. Price, Marjory Moreau, J. Brian Houston, Miyoung Yoon, Moire R. Creek, Carina Cantrill, Larry G. Higgins, Brian G. Lake, Mary P. Scott
المصدر: Xenobiotica. 51:40-50
مصطلحات موضوعية: Pharmacology, endocrine system, Chemistry, Health, Toxicology and Mutagenesis, Kinetics, General Medicine, Metabolism, Toxicology, 030226 pharmacology & pharmacy, Biochemistry, In vitro, 03 medical and health sciences, chemistry.chemical_compound, Cytosol, 0302 clinical medicine, Deltamethrin, 030220 oncology & carcinogenesis, parasitic diseases, Microsome, medicine, Cis–trans isomerism, Permethrin, medicine.drug
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المؤلفون: Mohammed Ullah, Kenichi Umehara, Carina Cantrill, Florian Klammers, Aynur Ekiciler, Neil Parrott, Stephen Fowler, Elisa Di Lenarda, Matthias B. Wittwer
المصدر: Drug Metabolism and Disposition. 48:849-860
مصطلحات موضوعية: Male, Metabolic Clearance Rate, Primary Cell Culture, Pharmaceutical Science, Computational biology, Models, Biological, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, Drug Development, In vivo, Drug Discovery, Humans, Cells, Cultured, Selection (genetic algorithm), Pharmacology, Chemistry, Drug discovery, In vitro toxicology, Uptake transporters, Coculture Techniques, In vitro, Metabolic enzymes, 030220 oncology & carcinogenesis, Hepatocytes, Female, Hepatic Elimination
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e8e02ed211aab3a6527b03d7c3d99af9
https://doi.org/10.1124/dmd.120.000133 -
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المؤلفون: Roger J, Price, Mary P, Scott, Carina, Cantrill, Larry G, Higgins, Marjory, Moreau, Miyoung, Yoon, Harvey J, Clewell, Moire R, Creek, Thomas G, Osimitz, J Brian, Houston, Brian G, Lake
المصدر: Xenobiotica; the fate of foreign compounds in biological systems. 51(1)
مصطلحات موضوعية: Male, Carboxylesterase, Rats, Rats, Sprague-Dawley, Kinetics, Cytosol, Cytochrome P-450 Enzyme System, Liver, Nitriles, Pyrethrins, Hepatocytes, Microsomes, Liver, Animals, Humans, Permethrin
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المؤلفون: Carina Cantrill, Caroline Rynn, Prasoon Chaturvedi, Matthias B. Wittwer, Isabelle Walter, Jeannine Petrig Schaffland
المصدر: Drug discovery today. 25(6)
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, Computer science, Drug discovery, Computational biology, Myotonin-Protein Kinase, Small Molecule Libraries, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, 030220 oncology & carcinogenesis, Neoplasms, Drug Discovery, Animals, Humans
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المؤلفون: Carina Cantrill, Arto Urtti, Paulina Jakubiak, Rubén Alvarez-Sánchez
المصدر: Molecular pharmaceutics. 16(12)
مصطلحات موضوعية: Octanols, Pharmaceutical Science, 02 engineering and technology, Pharmacology, Eye, 030226 pharmacology & pharmacy, Cell Line, Melanin, 03 medical and health sciences, 0302 clinical medicine, Melanin binding, Pharmacokinetics, Tandem Mass Spectrometry, Drug Discovery, Distribution (pharmacology), Animals, Humans, ATP Binding Cassette Transporter, Subfamily B, Member 1, In vitro in vivo, Rats, Wistar, Melanins, integumentary system, Chemistry, Half-life, Blood Proteins, 021001 nanoscience & nanotechnology, Small molecule, In vitro, 3. Good health, Rats, Kinetics, Molecular Medicine, sense organs, 0210 nano-technology, Chromatography, Liquid, Half-Life, Protein Binding
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المؤلفون: Carina Cantrill, J. Brian Houston
المصدر: Journal of Pharmaceutical Sciences. 106:2815-2825
مصطلحات موضوعية: Male, Quinidine, Atorvastatin, Pharmaceutical Science, Pharmacology, 030226 pharmacology & pharmacy, Rats, Sprague-Dawley, 03 medical and health sciences, 0302 clinical medicine, medicine, Animals, Humans, Cells, Cultured, biology, Chemistry, Multidrug resistance-associated protein 2, Membrane Transport Proteins, Biological Transport, Repaglinide, Hepatobiliary Elimination, Organic anion-transporting polypeptide, medicine.anatomical_structure, Liver, Pharmaceutical Preparations, 030220 oncology & carcinogenesis, Hepatocyte, Hepatocytes, biology.protein, Efflux, Saquinavir, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ad0e58a62fa5d8368a02809b1caf674f
https://doi.org/10.1016/j.xphs.2017.04.056 -
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المؤلفون: A. David Rodrigues, Manthena V.S. Varma, Sweta Modi, Carina Cantrill, Ayşe Ufuk, Mark Niosi, Tom De Bruyn, Yi An Bi, Rachel E. Kosa, J. Brian Houston, Aleksandra Galetin, Larry M. Tremaine
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 46(7)
مصطلحات موضوعية: Adult, Metabolic Clearance Rate, Pharmaceutical Science, Organic Anion Transporters, Pharmacology, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, In vivo, medicine, Animals, Humans, Pitavastatin, biology, Chemistry, Cerivastatin, Transporter, Biological Transport, In vitro, Orders of magnitude (mass), Organic anion-transporting polypeptide, Kinetics, Macaca fascicularis, medicine.anatomical_structure, Liver, Pharmaceutical Preparations, 030220 oncology & carcinogenesis, Hepatocyte, biology.protein, Hepatocytes, Female, Hydroxymethylglutaryl-CoA Reductase Inhibitors, Peptides, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d8e815acb044ed7774f8725c3f309670
https://pubmed.ncbi.nlm.nih.gov/29720472