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1
المؤلفون: Benjamin Bader, Sabine Zitzmann-Kolbe, Carl Friedrich Nising, Ulrich Lücking, Qi Wang, Hartmut Rehwinkel, Florian Bartels, Qiuwen Wang, Markus Berger, Antje Margret Wengner, Lars Wortmann, Dieter Moosmayer, Philipp Buchgraber, Hans Briem, Dominik Mumberg, Knut Eis, Uwe Eberspächer, Stefanie Hammer, Christoph A. Schatz, Gerhard Siemeister, Philip Lienau, Ulf Bömer
المصدر: Journal of Medicinal Chemistry. 64:12723-12737
مصطلحات موضوعية: DNA repair, Cell, Antineoplastic Agents, DNA-Activated Protein Kinase, Cell cycle phase, Mice, Phosphatidylinositol 3-Kinases, Structure-Activity Relationship, chemistry.chemical_compound, Cell Line, Tumor, Drug Discovery, medicine, Animals, Humans, Protein kinase A, Cell Proliferation, Molecular Structure, Chemistry, TOR Serine-Threonine Kinases, Drug Synergism, medicine.disease, Xenograft Model Antitumor Assays, In vitro, Rats, medicine.anatomical_structure, Gene Expression Regulation, Ataxia-telangiectasia, Hepatocytes, Cancer research, Molecular Medicine, Drug Therapy, Combination, Homologous recombination, DNA
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2
المؤلفون: Niels Böhnke, Markus Berger, Nils Griebenow, Antje Rottmann, Michael Erkelenz, Stefanie Hammer, Sandra Berndt, Judith Günther, Antje M. Wengner, Beatrix Stelte-Ludwig, Christoph Mahlert, Simone Greven, Lisa Dietz, Hannah Jörißen, Naomi Barak, Ulf Bömer, Roman C. Hillig, Uwe Eberspaecher, Jörg Weiske, Anja Giese, Dominik Mumberg, Carl Friedrich Nising, Hilmar Weinmann, Anette Sommer
المصدر: Bioconjugate chemistry. 33(6)
مصطلحات موضوعية: Pharmacology, B7 Antigens, Immunoconjugates, Organic Chemistry, Biomedical Engineering, Pharmaceutical Science, Bioengineering, Antineoplastic Agents, Xenograft Model Antitumor Assays, Mice, Structure-Activity Relationship, Cell Line, Tumor, Neoplasms, Animals, Humans, Nicotinamide Phosphoribosyltransferase, Biotechnology
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3
المؤلفون: Andrea Hägebarth, Carl Friedrich Nising, Philip Lienau, Julien Lefranc, Benjamin Bader, Clara D. Christ, Volker K Schulze, Clara Lemos, Simon Holton, Tobias Heinrich, Ulf Bömer, Franz von Nussbaum, Hans Briem, Ekaterina Nevedomskaya, Simon J. Baumgart, Dominik Mumberg, Bernard Haendler, Marcus Bauser, Lara Kuhnke
المصدر: Cellular Oncology. 44:581-594
مصطلحات موضوعية: Male, 0301 basic medicine, Cancer Research, Antineoplastic Agents, AMP-Activated Protein Kinases, 03 medical and health sciences, Prostate cancer, 0302 clinical medicine, Cell Line, Tumor, Lipid droplet, medicine, Humans, Enzyme Inhibitors, Protein kinase A, Chemistry, Kinase, Prostatic Neoplasms, AMPK, Lipid metabolism, General Medicine, medicine.disease, Androgen receptor, 030104 developmental biology, Oncology, 030220 oncology & carcinogenesis, Cancer research, Molecular Medicine, Chromatin immunoprecipitation, Signal Transduction
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4
المؤلفون: Carl Friedrich Nising
المصدر: Forschung & Lehre.
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::bf361186d26c177791b3c9aa7305b188
https://doi.org/10.37307/j.0945-5604.2022.01.14 -
5
المؤلفون: Volker Schulze, Franz von Nussbaum, Clara Lemos, Philip Lienau, Ulf Bömer, Clara Christ, Marcus Bauser, Carl Friedrich Nising, Simon J. Baumgart, Simon Holton, Tobias Heinrich, Hans Briem, Benjamin Bader, Bernard Haendler, Julien Lefranc, Andrea Hägebarth, Dominik Mumberg, Ekaterina Nevedomskaya, Lara Kuhnke
مصطلحات موضوعية: Prostate cancer, Androgen dependent, business.industry, medicine, Cancer research, AMPK, medicine.disease, business, Bay
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::de28afe92f682da433e5d167b7b11ea8
https://doi.org/10.21203/rs.3.rs-47637/v1 -
6
المؤلفون: Antje Margret Wengner, Hans Briem, Stefan Gradl, Srinivasan Rengachari, Tobias Heinrich, Carl Friedrich Nising, Detlef Stöckigt, Franz von Nussbaum, Ulf Bömer, Julien Lefranc, Benjamin Bader, Anne Mengel, Dominik Mumberg, Roman C. Hillig, Volker K Schulze, Florian Prinz, Daniel Panne, József Bálint, Horst Irlbacher
المصدر: Journal of medicinal chemistry. 63(2)
مصطلحات موضوعية: Models, Molecular, Protein Serine-Threonine Kinases, Crystallography, X-Ray, 01 natural sciences, Substrate Specificity, Serine, 03 medical and health sciences, Structure-Activity Relationship, TANK-binding kinase 1, Drug Discovery, Structure–activity relationship, Humans, Threonine, Phosphorylation, Protein Kinase Inhibitors, 030304 developmental biology, 0303 health sciences, Binding Sites, Kinase, Drug discovery, Chemistry, 0104 chemical sciences, High-Throughput Screening Assays, I-kappa B Kinase, 010404 medicinal & biomolecular chemistry, Cancer research, Molecular Medicine, Benzimidazoles, Interferon regulatory factors
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7
المؤلفون: Carl Friedrich Nising, Brice Sautier, Lars Wortmann
المصدر: Angewandte Chemie International Edition. 55:15982-15988
مصطلحات موضوعية: 0301 basic medicine, Chemistry, Pharmaceutical, Druggability, Antineoplastic Agents, General Chemistry, Medicinal chemistry, Catalysis, 03 medical and health sciences, 030104 developmental biology, Neoplasms, Signaling proteins, Political science, ras Proteins, Humans, Critical assessment
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8
المؤلفون: Lars Wortmann, Brice Sautier, Carl Friedrich Nising
المصدر: Angewandte Chemie. 128:16215-16221
مصطلحات موضوعية: 0301 basic medicine, 03 medical and health sciences, 030104 developmental biology, General Medicine
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9
المؤلفون: Christoph Schatz, Frank Dittmer, Joachim Schuhmacher, Stefanie Hammer, Charlotte Christine Kopitz, Manuela Braun, Beatrix Stelte-Ludwig, Anette Sommer, Sabine Wittemer-Rump, Bertolt Kreft, Simone Greven, Hung Huynh, Heiner Apeler, Carl Friedrich Nising, Hans-Georg Lerchen, Christoph Mahlert, Axel Harrenga, Karl Ziegelbauer, Rolf Jautelat, Frank Reetz, Ruprecht Zierz
المصدر: Cancer Research. 76:6331-6339
مصطلحات موضوعية: musculoskeletal diseases, 0301 basic medicine, congenital, hereditary, and neonatal diseases and abnormalities, Cancer Research, Antibody-drug conjugate, Immunoconjugates, medicine.drug_class, Pharmacology, Biology, Antibodies, Monoclonal, Humanized, Monoclonal antibody, Mice, 03 medical and health sciences, 0302 clinical medicine, In vivo, Cell Line, Tumor, Neoplasms, medicine, Animals, Humans, Cytotoxic T cell, Potency, Aminobenzoates, Receptor, Fibroblast Growth Factor, Type 2, Mice, Inbred BALB C, integumentary system, Antibodies, Monoclonal, Cancer, medicine.disease, Xenograft Model Antitumor Assays, stomatognathic diseases, 030104 developmental biology, Oncology, Fibroblast growth factor receptor, 030220 oncology & carcinogenesis, embryonic structures, Monoclonal, Female, Oligopeptides
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5f282dd79ad32afbccf3ff32c85dd67f
https://doi.org/10.1158/0008-5472.can-16-0180 -
10
المؤلفون: Franziska Siegel, Carl Friedrich Nising, Franz von Nussbaum, Ulf Boemer, Herbert Himmel, Detlev Suelzle, Marcus Bauser, Uwe Eberspaecher, Simon Holton, Joerg Weiske, Florian Prinz, Ralf Lesche, Clara Lemos, Dominik Mumberg, Dieter Moosmayer, Knut Eis, Andrea Haegebarth, Stefan Prechtl, Barbara Nicke, Duy Nguyen, Lars Wortmann, Christian Lechner, Katrin Nowak-Reppel
المصدر: Journal of medicinal chemistry. 62(2)
مصطلحات موضوعية: 0301 basic medicine, Transcription, Genetic, Pyridines, Cell, Drug Evaluation, Preclinical, Apoptosis, Crystallography, X-Ray, Cell Line, 03 medical and health sciences, Structure-Activity Relationship, 0302 clinical medicine, Protein structure, RNA interference, Drug Discovery, medicine, Structure–activity relationship, Humans, Binding site, Protein Kinase Inhibitors, Mitogen-Activated Protein Kinase 7, Cell Proliferation, Binding Sites, Kinase, Chemistry, Cell Differentiation, Small molecule, Cell biology, Protein Structure, Tertiary, Molecular Docking Simulation, 030104 developmental biology, medicine.anatomical_structure, Pyrimidines, Cell culture, 030220 oncology & carcinogenesis, Molecular Medicine, Half-Life, Signal Transduction