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1دورية أكاديمية
المؤلفون: Christine Huynh, Swen Seeland, Jerome Segrestaa, Carmela Gnerre, Jens Hogeback, Henriette E. Meyer zu Schwabedissen, Jasper Dingemanse, Patricia N. Sidharta
المصدر: Frontiers in Pharmacology, Vol 13 (2022)
مصطلحات موضوعية: CXCR7, ADME, accelerator mass spectrometry, microtracer, CYP3A4, 14C-ACT-1004-1239, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Alexander Treiber, Stephane Delahaye, Swen Seeland, Carmela Gnerre
المصدر: Pharmacology Research & Perspectives, Vol 8, Iss 4, Pp n/a-n/a (2020)
مصطلحات موضوعية: endothelin receptor antagonist, macitentan, P450 induction, species differences, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2052-1707
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3دورية أكاديمية
المؤلفون: Carmela Gnerre, Gertrud U. Schuster, Adrian Roth, Christoph Handschin, Lisen Johansson, Renate Looser, Paolo Parini, Michael Podvinec, Kirsten Robertsson, Jan-Åke Gustafsson, Urs A. Meyer
المصدر: Journal of Lipid Research, Vol 46, Iss 8, Pp 1633-1642 (2005)
مصطلحات موضوعية: liver X receptor, pregnane X receptor, constitutive androstane receptor, metabolism, cytochrome P450 3a11, cytochrome P450 2b10, Biochemistry, QD415-436
وصف الملف: electronic resource
Relation: http://www.sciencedirect.com/science/article/pii/S002222752032962X; https://doaj.org/toc/0022-2275
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4
المؤلفون: Hamed Aissaoui, Martin Holdener, Carmela Gnerre, Kerstin Niggemann, Stefan Reber, Sylvia Richard, Romain Siegrist, Christoph Boss
المصدر: ChemMedChem. 18
مصطلحات موضوعية: Pharmacology, Organic Chemistry, Drug Discovery, Molecular Medicine, General Pharmacology, Toxicology and Pharmaceutics, Biochemistry
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5
المؤلفون: Sylvia Richard-Bildstein, Gabriel Schäfer, Laetitia Pouzol, Eleanor Lindenberg, François Lehembre, Hamed Aissaoui, Julien Pothier, Philippe Guerry, Carmela Gnerre
المصدر: Journal of Medicinal Chemistry. 63:15864-15882
مصطلحات موضوعية: Chemokine, Drug Evaluation, Preclinical, Molecular Conformation, Administration, Oral, Pharmacology, Crystallography, X-Ray, 01 natural sciences, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, 03 medical and health sciences, Chemokine receptor, Dogs, Piperidines, Oral administration, Drug Discovery, Extracellular, Animals, Humans, CXCL11, Amines, Receptor, 030304 developmental biology, G protein-coupled receptor, Receptors, CXCR, 0303 health sciences, biology, Chemistry, Antagonist, Amides, Chemokine CXCL12, Rats, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, biology.protein, Molecular Medicine, Half-Life, Protein Binding
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6
المؤلفون: Peter Seiler, L. Jacob, Swen Seeland, S. Diethelm, N. Tidten-Luksch, Jean-Philippe Surivet, M. Wicki, Georg Rueedi, Jean-Luc Specklin, Michel Enderlin-Paput, Christian Hubschwerlen, Azely Mirre, R. Lange, G. Mathieu, Christine Schmitt, C. Herrmann, Philippe Panchaud, A.-C. Blumstein, A. Mac Sweeney, F. Masse, Daniel Ritz, Jean-Christophe Gauvin, Carmela Gnerre
المصدر: Journal of Medicinal Chemistry. 63:66-87
مصطلحات موضوعية: Gram-negative bacteria, Microbial Sensitivity Tests, Hydroxamic Acids, medicine.disease_cause, Amidohydrolases, In vivo, Gram-Negative Bacteria, Drug Discovery, Hydrolase, Escherichia coli, medicine, Animals, Pyrroles, Enzyme Inhibitors, Escherichia coli Infections, Mice, Inbred ICR, biology, Chemistry, Pseudomonas aeruginosa, biology.organism_classification, Enterobacteriaceae, In vitro, Anti-Bacterial Agents, Multiple drug resistance, Klebsiella pneumoniae, Biochemistry, Molecular Medicine, Female, Bacteria
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7
المؤلفون: Christine, Huynh, Swen, Seeland, Jerome, Segrestaa, Carmela, Gnerre, Jens, Hogeback, Henriette E, Meyer Zu Schwabedissen, Jasper, Dingemanse, Patricia N, Sidharta
المصدر: Frontiers in pharmacology. 13
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::ccbd7b5b44b619c122e55eec640f8bac
https://pubmed.ncbi.nlm.nih.gov/35431953 -
8
المؤلفون: Michel Enderlin-Paput, Swen Seeland, A.-C. Blumstein, Daniel Ritz, Peter Seiler, R. Lange, Jean-Philippe Surivet, Christine Schmitt, F. Masse, Jean-Christophe Gauvin, S. Diethelm, L. Jacob, Charlyse Herrmann, Carmela Gnerre, Hans H. Locher, G. Mathieu, Azely Mirre, Georg Rueedi, Philippe Panchaud
المصدر: Journal of medicinal chemistry. 63(1)
مصطلحات موضوعية: Drug, media_common.quotation_subject, Microbial Sensitivity Tests, Pharmacology, Hydroxamic Acids, 01 natural sciences, Amidohydrolases, 03 medical and health sciences, Mice, In vivo, Drug Discovery, Gram-Negative Bacteria, Animals, Solubility, Enzyme Inhibitors, Lead (electronics), Escherichia coli Infections, 030304 developmental biology, media_common, 0303 health sciences, Molecular Structure, Chemistry, 0104 chemical sciences, Anti-Bacterial Agents, Rats, 010404 medicinal & biomolecular chemistry, Hepatocytes, Molecular Medicine, Administration, Intravenous
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9
المؤلفون: Keith Morrison, Daniel Wanner, Marc Iglarz, Martine Clozel, Katalin Menyhart, John Gatfield, Carmela Gnerre, Oliver Nayler, Lucile Monnier, Patrick Hess
المصدر: Journal of Pharmacology and Experimental Therapeutics. 362:186-199
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, Agonist, medicine.drug_class, Prostacyclin, Selexipag, Beraprost, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, chemistry, 030220 oncology & carcinogenesis, medicine, Molecular Medicine, Receptor, Active metabolite, Iloprost, medicine.drug, Treprostinil
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::938c47656b3da45652a07208bf6eeb23
https://doi.org/10.1124/jpet.116.239665 -
10
المؤلفون: Markus Rey, Alexander Treiber, Francis Hubler, Patrick Hess, Dorte Renneberg, Eva Caroff, Carmela Gnerre, Emmanuel Meyer, Kurt Hilpert, Markus A. Riederer, Beat Steiner
المصدر: Journal of Medicinal Chemistry. 58:9133-9153
مصطلحات موضوعية: chemistry.chemical_classification, Stereochemistry, Carboxylic acid, Pharmacology, Prodrug, Clopidogrel, Bioavailability, Piperazine, chemistry.chemical_compound, P2Y12, chemistry, In vivo, Drug Discovery, medicine, Molecular Medicine, Potency, medicine.drug