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1
المؤلفون: Pier D’Alessandro, Doug Minick, Sonia Delle-Fratte, Sharon Butler, Paul W. Smith, Adelheid Roth, Stephen P. Watson, Ezio Bettini, Vincenzo Garzya, Michela Andreoli, Caroline J. Goodacre, Palmina Cavallini, Roberto Benedetti, Catherine Ball, Parita Shah, Olivier Lorthioir, Fiona Brown, Ben Tehan, Maria Pilla, Michela Tessari
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:7521-7524
مصطلحات موضوعية: Mglur5 antagonist, Receptor, Metabotropic Glutamate 5, animal diseases, Clinical Biochemistry, Allosteric regulation, Administration, Oral, Pharmaceutical Science, Pharmacology, Receptors, Metabotropic Glutamate, Biochemistry, Mice, Structure-Activity Relationship, Allosteric Regulation, Oral administration, mental disorders, Drug Discovery, Animals, Molecular Biology, Chemistry, Organic Chemistry, Antagonist, Brain, Biological activity, Rats, stomatognathic diseases, Orally active, nervous system, Molecular Medicine, Heterocyclic Compounds, 3-Ring
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2
المؤلفون: Paul W. Smith, Caroline J. Goodacre, Wyman Paul Adrian, Sara A. Coggon, Vong Antonio Kuok Keong, Jeannette M. Watson, William J. Martin, Kirsten L. Searle, Daniel Marcus Bradley, Zining Wu, Peter J. Lovell, Lee A. Dawson, Harrington Frank Peter, David R. Thomas, Roderick A. Porter, Graham Murkitt, Halina T Serafinowska, Sean Thomas Flynn
المصدر: Bioorganicmedicinal chemistry letters. 19(3)
مصطلحات موضوعية: Central Nervous System, Male, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Gerbil, Biochemistry, Rats, Sprague-Dawley, chemistry.chemical_compound, In vivo, Drug Discovery, Talnetant, medicine, Animals, Amines, Molecular Biology, Cerebral Cortex, Chemistry, Organic Chemistry, Quinoline, Antagonist, Brain, Receptors, Neurokinin-3, Rats, Models, Chemical, Area Under Curve, Lipophilicity, Quinolines, Molecular Medicine, Gerbillinae, Ex vivo, medicine.drug
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3
المؤلفون: Claire M. Scott, Vong Antonio Kuok Keong, Paul W. Smith, Caroline J. Goodacre, Jeannette M. Watson, Frank E. Blaney, Simon E. Ward, Kathryn R. Starr, Peter J. Lovell, Kevin M. Thewlis
المصدر: Bioorganicmedicinal chemistry letters. 17(4)
مصطلحات موضوعية: Models, Molecular, Magnetic Resonance Spectroscopy, Stereochemistry, Pyridines, Clinical Biochemistry, Guinea Pigs, Pharmaceutical Science, CHO Cells, Inhibitory postsynaptic potential, Biochemistry, Chemical synthesis, Binding, Competitive, Mass Spectrometry, Piperazines, Cell Line, chemistry.chemical_compound, Radioligand Assay, Cricetulus, Cricetinae, Drug Discovery, Animals, Humans, Receptor, Molecular Biology, Cerebral Cortex, Bicyclic molecule, Chemistry, Benzoxazinones, Organic Chemistry, Antagonist, Callithrix, Benzoxazines, Rats, Receptor, Serotonin, 5-HT1D, Receptor, Serotonin, 5-HT1A, Receptor, Serotonin, 5-HT1B, Molecular Medicine, 5-HT1A receptor, Indicators and Reagents, Serotonin Antagonists, Lead compound, Selective Serotonin Reuptake Inhibitors, Synaptosomes
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4
المؤلفون: Caroline J. Goodacre, et al. et al.
المصدر: ChemInform. 37
مصطلحات موضوعية: 5-HT2C receptor, Orally active, Stereochemistry, Chemistry, General Medicine
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5
المؤلفون: Peter J. Lovell, Caroline J. Goodacre, Brenda K. Trail, Graham J. Riley, Kathryn R. Starr, Michael Allen, Steven Mark Bromidge, Vicky Holland, David E. Clapham, Lorraine Campbell, Frank D. King, Martyn D. Wood
المصدر: Bioorganicmedicinal chemistry letters. 15(22)
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Administration, Oral, Imidazolidines, Biochemistry, Chemical synthesis, Sensitivity and Specificity, Cell Line, Substrate Specificity, chemistry.chemical_compound, Structure-Activity Relationship, Oral administration, Drug Discovery, Receptor, Serotonin, 5-HT2B, Receptor, Serotonin, 5-HT2C, Inverse agonist, Animals, Humans, Receptor, Serotonin, 5-HT2A, Receptor, Molecular Biology, 5-HT receptor, Molecular Structure, Chemistry, Organic Chemistry, Antagonist, Rats, 5-HT2C receptor, SB-243213, Serotonin 5-HT2 Receptor Antagonists, Molecular Medicine