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المؤلفون: Raymond E. Meyn, Kathryn A. Mason, Jessica M. Molkentine, Thomas A. Buchholz, Huifeng Liu, Colin Brooks, Carolyn A. Buser, Hiroshi Hirai, Kathleen A. Bridges
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7cf08c363837d0ba0914c4a603485323
https://doi.org/10.1158/1078-0432.22442226 -
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المؤلفون: Raymond E. Meyn, Kathryn A. Mason, Jessica M. Molkentine, Thomas A. Buchholz, Huifeng Liu, Colin Brooks, Carolyn A. Buser, Hiroshi Hirai, Kathleen A. Bridges
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::01014d7c5f01e804857d8d6cf44ce2b2
https://doi.org/10.1158/1078-0432.22442214 -
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المؤلفون: Raymond E. Meyn, Kathryn A. Mason, Jessica M. Molkentine, Thomas A. Buchholz, Huifeng Liu, Colin Brooks, Carolyn A. Buser, Hiroshi Hirai, Kathleen A. Bridges
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::76e72f6c26681d3b99fe5bfb640f4a5b
https://doi.org/10.1158/1078-0432.22442229 -
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المؤلفون: Raymond E. Meyn, Kathryn A. Mason, Jessica M. Molkentine, Thomas A. Buchholz, Huifeng Liu, Colin Brooks, Carolyn A. Buser, Hiroshi Hirai, Kathleen A. Bridges
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7df91317be846fddd348f9a8c4c1422d
https://doi.org/10.1158/1078-0432.22442232 -
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المؤلفون: Raymond E. Meyn, Kathryn A. Mason, Jessica M. Molkentine, Thomas A. Buchholz, Huifeng Liu, Colin Brooks, Carolyn A. Buser, Hiroshi Hirai, Kathleen A. Bridges
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0653bea5bb08d55cc7fc4d848a89e41b
https://doi.org/10.1158/1078-0432.22442220.v1 -
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المؤلفون: Raymond E. Meyn, Kathryn A. Mason, Jessica M. Molkentine, Thomas A. Buchholz, Huifeng Liu, Colin Brooks, Carolyn A. Buser, Hiroshi Hirai, Kathleen A. Bridges
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0b2cb6b819876a63a999c52bc36156f9
https://doi.org/10.1158/1078-0432.22442217.v1 -
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المؤلفون: Raymond E. Meyn, Kathryn A. Mason, Jessica M. Molkentine, Thomas A. Buchholz, Huifeng Liu, Colin Brooks, Carolyn A. Buser, Hiroshi Hirai, Kathleen A. Bridges
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8fbfa6fcbea849181690711487a614a1
https://doi.org/10.1158/1078-0432.22442223.v1 -
8High-Throughput Screening and Triage Assays Identify Small Molecules Targeting c-MYC in Cancer Cells
المؤلفون: Jon-Paul Jaworski, Lisa A. Payne, Anna Waszkiewicz, Biju Mangatt, Anthony J. Jurewicz, Lorena A. Kallal, Jesus R. Medina, Pat Brady, Xin Zeng, Thomas J. Berrodin, Carolyn Doepner-Buser, Anthony Della Pietra
المصدر: SLAS discovery : advancing life sciences RD. 26(2)
مصطلحات موضوعية: 0301 basic medicine, High-throughput screening, Genes, myc, Biochemistry, Analytical Chemistry, Flow cytometry, Small Molecule Libraries, 03 medical and health sciences, 0302 clinical medicine, Drug Discovery, medicine, Fluorescence Resonance Energy Transfer, Humans, Transcription factor, Reporter gene, medicine.diagnostic_test, Cell growth, Chemistry, Reverse Transcriptase Polymerase Chain Reaction, Cell cycle, Gene signature, Flow Cytometry, Molecular biology, High-Throughput Screening Assays, Gene Expression Regulation, Neoplastic, 030104 developmental biology, 030220 oncology & carcinogenesis, Cancer cell, Molecular Medicine, Drug Screening Assays, Antitumor, Biotechnology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::0dbee602aec0943dd6af57df9d435d52
https://pubmed.ncbi.nlm.nih.gov/33482073 -
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المؤلفون: Carlo Toniatti, Carolyn A. Buser, Kathleen Bridges, Raymond E. Meyn, Huifeng Liu, Thomas A. Buchholz
المصدر: Oncotarget
مصطلحات موضوعية: Male, Radiation-Sensitizing Agents, Indazoles, Lung Neoplasms, DNA Repair, Cell Survival, DNA repair, DNA damage, Poly ADP ribose polymerase, RAD51, Breast Neoplasms, Poly(ADP-ribose) Polymerase Inhibitors, Biology, Poly (ADP-Ribose) Polymerase Inhibitor, Cell Line, PARP, MK-4827, Histones, Piperidines, Carcinoma, Non-Small-Cell Lung, Cell Line, Tumor, medicine, Humans, DNA Breaks, Double-Stranded, DNA Breaks, Single-Stranded, Tumor Stem Cell Assay, Radiation, Prostatic Neoplasms, Cancer, Hydrogen Peroxide, Base excision repair, Oxidants, medicine.disease, Molecular biology, Microscopy, Fluorescence, Oncology, Female, Rad51 Recombinase, Poly(ADP-ribose) Polymerases, Tumor Suppressor Protein p53, niraparib, Research Paper
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::6fbfd3a8f1b823267419e77bebb3b9c4
https://doi.org/10.18632/oncotarget.2083 -
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المؤلفون: Steven M. Stirdivant, Carolyn A. Buser, Weikang Tao, Laura Sepp-Lorenzino, Cheng Wang, Mark E. Fraley, Robert B. Lobell, Keith W. Rickert, Kenneth L. Arrington, Kelly Hamilton, Vadim Y. Dudkin, James Hardwick, Eileen S. Walsh, George D. Hartman, Xianzhi Mao, Robert A. Drakas, Stephen C. Beck
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:2613-2619
مصطلحات موضوعية: Cell Membrane Permeability, Halogenation, Pyridines, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, Biochemistry, Polar surface area, Structure-Activity Relationship, chemistry.chemical_compound, Aminothiazole, Cell Line, Tumor, Drug Discovery, Humans, Potency, Protein Kinase Inhibitors, Molecular Biology, Molecular Structure, Kinase, Organic Chemistry, Cell Cycle Checkpoints, Biochemical Activity, Cyclin-Dependent Kinases, Kinetics, Thiazoles, chemistry, Drug Design, Checkpoint Kinase 1, Lipophilicity, Molecular Medicine, Cyclin-dependent kinase 7, Selectivity, Protein Kinases, Cyclin-Dependent Kinase-Activating Kinase