-
1
المؤلفون: Alison M. Strack, Xinchun Tong, Christina B. Madsen-Duggan, Lauren P. Shearman, Cathy R.-R.C. Huang, Mark T. Goulet, Thomas F. Walsh, Yue Feng, Jing Chen Xiao, D. Sloan Stribling, Junying Wang, John S. Debenham, Tung M. Fong, Chun-Pyn Shen, Sanjeev Kumar, Julie Lao, Donald J. Marsh, Richard B. Toupence
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:1448-1452
مصطلحات موضوعية: Cannabinoid 1 receptor, Pyridines, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Receptor, Cannabinoid, CB1, Pharmacokinetics, Drug Discovery, Pyridine, medicine, Animals, Humans, Inverse agonist, Benzopyrans, Furans, Receptor, Molecular Biology, Biological evaluation, Mice, Knockout, Molecular Structure, Chemistry, Organic Chemistry, Haplorhini, Rats, Orally active, Drug Design, Molecular Medicine, Cannabinoid
-
2
المؤلفون: Mark T. Goulet, Christina B. Madsen-Duggan, Yue Feng, George A. Doss, Jing Chen Xiao, John S. Debenham, Cathy R.-R.C. Huang, Lex H.T. Van der Ploeg, Alison M. Strack, Chun-Pyn Shen, Marie-Therese Schaeffer, Donald J. Marsh, Junying Wang, D. Euan MacIntyre, Julie Lao, Tung M. Fong, D. Sloan Stribling, Lauren P. Shearman, Thomas F. Walsh, Xinchun Tong
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:681-685
مصطلحات موضوعية: Cannabinoid receptor, medicine.medical_treatment, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Biochemistry, Chemical synthesis, Eating, Mice, Receptor, Cannabinoid, CB1, Oral administration, In vivo, Drug Discovery, medicine, Animals, Inverse agonist, Naphthyridines, Molecular Biology, Mice, Knockout, Binding Sites, Chemistry, Organic Chemistry, In vitro, Models, Chemical, nervous system, Knockout mouse, Molecular Medicine, lipids (amino acids, peptides, and proteins), Cannabinoid
-
3
المؤلفون: Christopher P. Austin, Doreen E. Cashen, Sheng-Shung Pong, Brian D. Spar, Brett Connolly, Tung Ming Fong, D. Euan MacIntyre, Carina P. Tan, Michael R. Tota, Ravi P. Nargund, R. S. L. Chang, Oksana C. Palyha, Constantin Tamvakopoulos, Deborah L. Drazen, Anthony G. DiLella, Jennifer E. Drisko, David J. Figueroa, Tanya MacNeil, Andreas W. Sailer, David H. Weinberg, Randy J. Nelson, Charles Rosenblum, Cathy R.-R.C. Huang, Rui Tang, Arthur A. Patchett, Xiao-Ming Guan, Hong Yu, George J. Christ, Andrew D. Howard, Lex H.T. Van der Ploeg, William J. Martin, Aurawan Vongs, Iyassu K. Sebhat, Ralph A. Stearns
المصدر: Proceedings of the National Academy of Sciences. 99:11381-11386
مصطلحات موضوعية: Male, Agonist, medicine.medical_specialty, DNA, Complementary, Intracranial Pressure, medicine.drug_class, Blood Pressure, In Vitro Techniques, Biology, Somatosensory system, Mice, Sexual Behavior, Animal, Nerve Fibers, Internal medicine, Copulation, medicine, Animals, Glans, In Situ Hybridization, DNA Primers, Multidisciplinary, Reverse Transcriptase Polymerase Chain Reaction, Human penis, Feeding Behavior, Ribonuclease, Pancreatic, Biological Sciences, Spinal cord, Electric Stimulation, Mice, Inbred C57BL, Melanocortin 4 receptor, medicine.anatomical_structure, Endocrinology, Receptors, Corticotropin, Models, Animal, Receptor, Melanocortin, Type 4, Brainstem, Energy Metabolism, Penis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::341db11f0e12a0307d07e04176cd4aad
https://doi.org/10.1073/pnas.172378699 -
4
المؤلفون: Pei Huo, Lauren P. Shearman, Thomas F. Walsh, Christina B. Madsen-Duggan, Jing Chen Xiao, Xinchun Tong, Alison M. Strack, Cathy R.-R.C. Huang, Tung M. Fong, Mark T. Goulet, Chun-Pyn Shen, Junying Wang, D. Sloan Stribling, Lin Yan, John S. Debenham, Julie Lao, Jeffrey J. Hale
المصدر: Bioorganicmedicinal chemistry letters. 20(12)
مصطلحات موضوعية: Food intake, Cannabinoid receptor, Stereochemistry, Pyridines, Clinical Biochemistry, Pharmaceutical Science, Administration, Oral, Biochemistry, Receptor, Cannabinoid, CB2, chemistry.chemical_compound, Eating, Structure-Activity Relationship, Pharmacokinetics, Receptor, Cannabinoid, CB1, Drug Discovery, Pyridine, Weight Loss, Inverse agonist, Animals, Humans, Naphthyridines, Receptor, Molecular Biology, Biological evaluation, Organic Chemistry, Rats, Orally active, chemistry, Molecular Medicine