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المؤلفون: Shaoxian Sun, Phuong Le, Shubha Bagrodia, Sadayappan V. Rahavendran, Eric Zhang, Cheng Hengmiao, Cathy Xiang, Robert Steven Kania, Jing Yuan, William Farrell, Jacqui Elizabeth Hoffman, Pairish Mason Alan, Deepak Dalvie
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:2787-2792
مصطلحات موضوعية: Pyridones, Carboxylic acid, Metabolite, Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, Pyrimidinones, Pharmacology, Crystallography, X-Ray, Biochemistry, Mice, Phosphatidylinositol 3-Kinases, Structure-Activity Relationship, chemistry.chemical_compound, Cell Line, Tumor, Amide, Drug Discovery, Animals, Humans, Structure–activity relationship, Protein Kinase Inhibitors, Molecular Biology, Protein kinase B, PI3K/AKT/mTOR pathway, Phosphoinositide-3 Kinase Inhibitors, chemistry.chemical_classification, Binding Sites, Kinase, Chemistry, TOR Serine-Threonine Kinases, Organic Chemistry, Xenograft Model Antitumor Assays, Protein Structure, Tertiary, Molecular Docking Simulation, Pyrimidines, Drug Design, Molecular Medicine, Signal transduction, Proto-Oncogene Proteins c-akt, Signal Transduction