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1
المؤلفون: Andreas Kuglstatter, Shirley Li, Robert Crowther, Christine Lukacs, Cheryl Janson, Srinivasan Swaminathan, Stacy Remiszewski, Manish Kumar Thakur, Andrew Schutt, Rajat Pandey, Waleed Danho, Barry Goggin, Rajiv Tyagi, Saroj K. Singh, Charles Belunis, Ramachandraiah Gosu, Lin Gao, Ajith V. Kamath
المصدر: Acta Crystallographica Section D: Biological Crystallography
مصطلحات موضوعية: Molecular Sequence Data, AVPI, Regulator, Apoptosis, X-Linked Inhibitor of Apoptosis Protein, Caspase 3, Crystallography, X-Ray, Inhibitor of apoptosis, Inhibitor of Apoptosis Proteins, Viral Proteins, XIAP, Structural Biology, Protein Interaction Mapping, Humans, Amino Acid Sequence, Peptide sequence, Caspase, Oligopeptide, biology, BIR domains, General Medicine, Research Papers, Caspase Inhibitors, Nucleopolyhedroviruses, Protein Structure, Tertiary, caspases, peptide complex, Biochemistry, inhibitor of apoptosis, Multigene Family, biology.protein, Biophysics, extrinsic pathway, Apoproteins, SMAC, Oligopeptides
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2
المؤلفون: Cheryl Janson, David C. Fry, Ursula Kammlott, Stefan Palme, Binh Thanh Vu, Bradford Graves, Christine Lukacs, Christian Klein, Charles Belunis, Charles Wartchow
المصدر: ACS Medicinal Chemistry Letters. 4:660-665
مصطلحات موضوعية: Drug discovery, Organic Chemistry, Nutlin, Computational biology, Biology, Biochemistry, Combinatorial chemistry, Protein–protein interaction, chemistry.chemical_compound, chemistry, Drug Discovery, biology.protein, Molecule, Mdm2, Surface plasmon resonance, Binding Determinants, Heteronuclear single quantum coherence spectroscopy
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3
المؤلفون: Rebecca Taub, David Robert Bolin, Shawn David Erickson, Charles Belunis, Stanley Wertheimer, Cristina M. Rondinone, Anish Konkar, Karin Conde-Knape
المصدر: Drug Discovery Today: Therapeutic Strategies. 4:129-135
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, medicine.medical_specialty, Calorie, Fatty acid, Adipose tissue, Type 2 diabetes, Biology, medicine.disease, Obesity, Insulin resistance, Endocrinology, chemistry, Internal medicine, Drug Discovery, medicine, Molecular Medicine, Lipolysis, Metabolic syndrome
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4
المؤلفون: Kurt Hollfelder, Charles Belunis, Robert Crowther, Pete William Dunten, David J. Weber, Ursula Kammlott, Wayne Levin, Hanspeter Michel, Gwendolyn Ramsey, Amy Swain, Stanley Wertheimer
المصدر: Journal of Molecular Biology. 316:257-264
مصطلحات موضوعية: Models, Molecular, endocrine system, endocrine system diseases, GTP', Protein Conformation, Phenylalanine, Biology, Crystallography, X-Ray, digestive system, Substrate Specificity, Phosphoenolpyruvate, Cytosol, Structural Biology, Humans, Binding site, Molecular Biology, chemistry.chemical_classification, Binding Sites, nutritional and metabolic diseases, Hydrogen Bonding, Lyase, Citric acid cycle, Metabolic pathway, Enzyme, Biochemistry, chemistry, Gluconeogenesis, Phosphoenolpyruvate Carboxykinase (GTP), Guanosine Triphosphate, Phosphoenolpyruvate carboxykinase, Phosphoenolpyruvate Carboxykinase (ATP), hormones, hormone substitutes, and hormone antagonists
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المؤلفون: Gary L. Olson, Damir Vidovic, Ramakanth Sarabu, J. Hammer, Francesco Sinigaglia, Zoltan A. Nagy, Michael Steinmetz, Nicholas John Silvester Huby, Jeanmarie Guenot, Charles Belunis, Kouichi Ito, Robert K. Campbell, Paul Gillespie, David Robert Bolin, Steven Joseph Berthel, Vincent S. Madison, Fiorenza Falcioni
المصدر: Nature Biotechnology. 17:562-567
مصطلحات موضوعية: Peptidomimetic, T-Lymphocytes, Antigen presentation, Biomedical Engineering, Arthritis, Bioengineering, Plasma protein binding, Biology, medicine.disease_cause, Applied Microbiology and Biotechnology, Cell Line, Arthritis, Rheumatoid, medicine, Humans, Amino Acid Sequence, Peptide sequence, Autoimmune disease, Antigen Presentation, Molecular Mimicry, Hydrogen Bonding, HLA-DR Antigens, medicine.disease, Cathepsins, Molecular mimicry, Amino Acid Substitution, Cell culture, Immunology, Molecular Medicine, Oligopeptides, Protein Binding, Biotechnology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::70409305cc5fff290c510e7758273981
https://doi.org/10.1038/9865 -
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المؤلفون: J Han, R Arceo, Damir Vidovic, Jeanne Magram, M Molina, David Robert Bolin, Fiorenza Falcioni, J. Hammer, E Saar, Zoltan A. Nagy, Charles Belunis, Kouichi Ito, Robert M. Campbell, H J Bian
المصدر: The Journal of Experimental Medicine
مصطلحات موضوعية: CD4-Positive T-Lymphocytes, Encephalomyelitis, Autoimmune, Experimental, Recombinant Fusion Proteins, T-Lymphocytes, Genes, MHC Class II, Molecular Sequence Data, Immunology, HLA-DR alpha-Chains, Mice, Transgenic, Human leukocyte antigen, Lymphocyte Activation, Polymerase Chain Reaction, Autoimmune Diseases, MHC Class II Gene, Mice, Antigen, HLA-DRA, MHC class I, HLA-DR4 Antigen, medicine, Animals, Humans, Immunology and Allergy, Amino Acid Sequence, Antigens, HLA-DR Antigen, DNA Primers, Inflammation, MHC class II, Binding Sites, Base Sequence, biology, Experimental autoimmune encephalomyelitis, Brain, Myelin Basic Protein, HLA-DR Antigens, Articles, Flow Cytometry, medicine.disease, Molecular biology, Mice, Inbred C57BL, Spinal Cord, biology.protein, Disease Susceptibility, Lymph Nodes, Myelin Proteins, HLA-DRB1 Chains
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::e21dc758902c6baaba4db2d63b877c01
https://doi.org/10.1084/jem.183.6.2635 -
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المؤلفون: Fiorenza Falcioni, David Robert Bolin, Botond Siklodi, Charles Belunis, Kouichi Ito, Damir Vidovic, Zoltan A. Nagy
المصدر: European Journal of Immunology. 25:3349-3355
مصطلحات موضوعية: T cell, Molecular Sequence Data, Immunology, Antigen presentation, Antigen-Presenting Cells, Down-Regulation, Major histocompatibility complex, Epitopes, Immunoglobulin Fab Fragments, Antigen, MHC class I, medicine, Humans, Immunology and Allergy, Cytotoxic T cell, Amino Acid Sequence, Antigen-presenting cell, biology, Histocompatibility Antigens Class II, Antibodies, Monoclonal, HLA-DR Antigens, T-Lymphocytes, Helper-Inducer, Molecular biology, medicine.anatomical_structure, biology.protein, CD8
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8
المؤلفون: Ryoichi Saitoh, Takaaki Miura, Takeshi Murata, Yasuaki Matsubara, Christine Lukacs, Eisaku Mizuguchi, Nobuo Shimma, Yasunori Chugai Seiyaku Kabushiki Kaisha Kohchi, Charles Belunis, Hisafumi Okabe, Yoshiaki Isshiki, Masanori Miwa, Verena Schück, Kohsuke Asoh, Kazuo Hattori, Hitoshi Iikura, Shinji Chugai Seiyaku Kabushiki Kaisha Tsujii, Naoaki Murao, Masami Kohchi, Cheryl Janson, Yasushi Yoshimura, Satoshi Aida
المصدر: Bioorganicmedicinal chemistry letters. 21(6)
مصطلحات موضوعية: MAPK/ERK pathway, Models, Molecular, Clinical Biochemistry, Allosteric regulation, Pharmaceutical Science, Administration, Oral, Antineoplastic Agents, Mitogen-activated protein kinase kinase, Pharmacology, Biochemistry, chemistry.chemical_compound, Allosteric Regulation, In vivo, Drug Discovery, Oxazines, Humans, Benzamide, Molecular Biology, Protein Kinase Inhibitors, chemistry.chemical_classification, biology, MEK inhibitor, Organic Chemistry, MAP Kinase Kinase Kinases, Enzyme, chemistry, Enzyme inhibitor, Benzamides, biology.protein, Molecular Medicine
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المؤلفون: Steven I. Reed, Kuo-Sen Huang, Wei Chu, David J. Weber, Lyubomir T. Vassilev, Kui Xu, Charles Belunis, Frank John Podlaski
المصدر: The Biochemical journal. 371(Pt 3)
مصطلحات موضوعية: Multiprotein complex, Ubiquitin-Protein Ligases, Allosteric regulation, Molecular Sequence Data, Cell Cycle Proteins, Biochemistry, Protein–protein interaction, Substrate Specificity, Ligases, DDB1, Ubiquitin, Allosteric Regulation, Skp1, Humans, Amino Acid Sequence, Molecular Biology, S-Phase Kinase-Associated Proteins, chemistry.chemical_classification, DNA ligase, biology, Sequence Homology, Amino Acid, Tumor Suppressor Proteins, Cell Biology, Cyclin-Dependent Kinases, Recombinant Proteins, Ubiquitin ligase, chemistry, biology.protein, Cyclin-Dependent Kinase Inhibitor p27, Protein Binding, Research Article
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::de3bd480825e4a7d90baf5beaaa232c4
https://pubmed.ncbi.nlm.nih.gov/12529174 -
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المؤلفون: Ramakanth Sarabu, Fiorenza Falcioni, Amy Swain, Lucja Orzechowski, Raymond Makofske, Ursula Kammlott, Xiaolei Zhang, Jeanmarie Guenot, Donald C. Cox, Damir Vidovic, Gary L. Olson, Nan Jiang, David Robert Bolin, Robert Crowther, Joel P. Cooper, Paul Gillespie, Diana Gaizband, Robert M. Campbell, Charles Belunis, David J. Weber, Kouichi Ito, Steven Joseph Berthel, Agostino Perrotta, Robert Palermo, Nicholas John Silvester Huby, Zoltan A. Nagy, Katherine Toth
المصدر: Journal of medicinal chemistry. 43(11)
مصطلحات موضوعية: Models, Molecular, Peptide Biosynthesis, Phage display, Stereochemistry, Protein Conformation, T-Lymphocytes, Antigen presentation, Carbohydrates, Peptide, Major histocompatibility complex, Crystallography, X-Ray, Binding, Competitive, Methylation, Cathepsin B, chemistry.chemical_compound, Structure-Activity Relationship, Antigen, Drug Discovery, HLA-DR, Humans, chemistry.chemical_classification, MHC class II, Antigen Presentation, Dipeptide, biology, Molecular Mimicry, Dipeptides, HLA-DR Antigens, chemistry, Biochemistry, biology.protein, Molecular Medicine, Cell Division