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1دورية أكاديمية
المؤلفون: Rudolf Mueller, Virsinha Reddy, Aloysius T. Nchinda, Fanuel Mebrahtu, Dale Taylor, Nina Lawrence, Lloyd Tanner, Marine Barnabe, Charles J. Eyermann, Bin Zou, Ravinder R. Kondreddi, Suresh B. Lakshminarayana, Matthias Rottmann, Leslie J. Street, Kelly Chibale
المصدر: ACS Omega, Vol 5, Iss 12, Pp 6967-6982 (2020)
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2470-1343
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المؤلفون: Preshendren Govender, Rudolf Müller, Kawaljit Singh, Virsinha Reddy, Charles J. Eyermann, Stephen Fienberg, Sandeep R. Ghorpade, Lizbé Koekemoer, Alissa Myrick, Dirk Schnappinger, Curtis Engelhart, Jaclynn Meshanni, Jo Ann W. Byl, Neil Osheroff, Vinayak Singh, Kelly Chibale, Gregory S. Basarab
المصدر: J Med Chem
مصطلحات موضوعية: DNA Gyrase, Gram-Negative Bacteria, Drug Discovery, Antitubercular Agents, Topoisomerase II Inhibitors, Molecular Medicine, Microbial Sensitivity Tests, Mycobacterium tuberculosis, Gram-Positive Bacteria, Article, Anti-Bacterial Agents
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3
المؤلفون: Lauren B. Arendse, Gyles E. Cozier, Charles J. Eyermann, Gregory S. Basarab, Sylva L. Schwager, Kelly Chibale, K. Ravi Acharya, Edward D. Sturrock
المصدر: Arendse, L B, Cozier, G, Eyermann, C, Basarab, G, Schwager, S L U, Chibale, K, Acharya, R & Sturrock, E D 2022, ' Probing the requirements for dual angiotensin-converting enzyme C-domain selective/neprilysin inhibition ', Journal of Medicinal Chemistry, vol. 65, no. 4, pp. 3371-3387 . https://doi.org/10.1021/acs.jmedchem.1c01924
مصطلحات موضوعية: Binding Sites, Pyridines, Thiazepines, Angiotensin-Converting Enzyme Inhibitors, Peptidyl-Dipeptidase A, Bradykinin, Crystallography, X-Ray, Kinetics, Lisinopril, Drug Discovery, Humans, Molecular Medicine, Computer Simulation, Neprilysin
وصف الملف: application/pdf
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المؤلفون: Stephen Fienberg, Gregory S. Basarab, Anne J. Lenaerts, Virsinha Reddy, Sandeep R. Ghorpade, Mathew Njoroge, Grant A. Boyle, Charles J. Eyermann, Clifton E. Barry, Timothy G. Myers, Efrem Abay, Nina Lawrence, Alissa Myrick, Helena I. Boshoff, Vinayak Singh, Lutete Peguy Khonde, Lisa M. Massoudi, Paul D. van Helden, Frederick A. Sirgel, Gregory T. Robertson, Rudolf Müller, Kelly Chibale, Aloysius T. Nchinda, Qin Su
المصدر: Journal of Medicinal Chemistry. 64:12790-12807
مصطلحات موضوعية: biology, Chemistry, INHA, biology.organism_classification, In vitro, Cell wall, Mycobacterium tuberculosis, Biochemistry, In vivo, Drug Discovery, Molecular Medicine, Potency, Pharmacophore, Drug metabolism
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المؤلفون: Shilpi Arora, Anna Kohlmann, Christopher D. Hupp, Julie Liu, Christelle Huguet, Allison Olszewski, Moritz von Rechenberg, John W. Cuozzo, Ying Zhang, Katy E Georgiadis, Matthew A. Clark, Esther C.Y. Lee, Charles J. Eyermann, Andrew J. McRiner, Paolo A. Centrella, Michael I Monteiro, Anthony D. Keefe, Benjamin Levin, Andrew D. Ferguson, Zooey Wang, Yanbin Liu
المصدر: Journal of Medicinal Chemistry. 64:6730-6744
مصطلحات موضوعية: Male, Indoles, Crystallography, X-Ray, 01 natural sciences, Chemical library, Small Molecule Libraries, Mice, Structure-Activity Relationship, 03 medical and health sciences, chemistry.chemical_compound, Pharmacokinetics, Drug Discovery, Animals, Humans, Structure–activity relationship, Potency, Transaminases, 030304 developmental biology, ADME, 0303 health sciences, Oxidase test, Binding Sites, Chemistry, DNA, Metabolism, 0104 chemical sciences, Molecular Docking Simulation, Alcohol Oxidoreductases, Thiazoles, 010404 medicinal & biomolecular chemistry, Biochemistry, Drug Design, Hyperoxaluria, Primary, Molecular Medicine, Glucuronide, Half-Life
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المؤلفون: John E. Burke, Jacob A. McPhail, Charles J. Eyermann, Kelly Chibale, Stephen Fienberg, Gregory S. Basarab, Lauren B. Arendse
المصدر: ACS Infectious Diseases. 6:3048-3063
مصطلحات موضوعية: 0301 basic medicine, Drug, biology, Chemistry, Kinase, media_common.quotation_subject, 030106 microbiology, Plasmodium falciparum, Computational biology, biology.organism_classification, 3. Good health, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, Infectious Diseases, Docking (molecular), Potency, Phosphatidylinositol, Homology modeling, Kinase activity, media_common
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7
المؤلفون: Gregory S. Basarab, Marshall Morningstar, Sheila Irene Hauck, Gunther Kern, Amy Kimzey, Vincent Galullo, Peter Doig, Charles J. Eyermann, Karthick Vishwanathan, Amy Kutschke, Virna J A Schuck, Fei Zhou, Madhusudhan Reddy Gowravaram
المصدر: Journal of Medicinal Chemistry. 63:11882-11901
مصطلحات موضوعية: Azoles, Staphylococcus aureus, Scaffold, Microbial Sensitivity Tests, Pyrimidinones, DNA gyrase, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Animals, Topoisomerase II Inhibitors, Spiro Compounds, Rats, Wistar, chemistry.chemical_classification, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Benzisoxazole, Isoxazoles, Staphylococcal Infections, Combinatorial chemistry, Anti-Bacterial Agents, Rats, Disease Models, Animal, DNA Gyrase, Molecular Medicine, Azole, Antibacterial activity
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المؤلفون: Lutete Peguy, Khonde, Rudolf, Müller, Grant A, Boyle, Virsinha, Reddy, Aloysius T, Nchinda, Charles J, Eyermann, Stephen, Fienberg, Vinayak, Singh, Alissa, Myrick, Efrem, Abay, Mathew, Njoroge, Nina, Lawrence, Qin, Su, Timothy G, Myers, Helena I M, Boshoff, Clifton E, Barry, Frederick A, Sirgel, Paul D, van Helden, Lisa M, Massoudi, Gregory T, Robertson, Anne J, Lenaerts, Gregory S, Basarab, Sandeep R, Ghorpade, Kelly, Chibale
المصدر: Journal of medicinal chemistry. 64(17)
مصطلحات موضوعية: Models, Molecular, Structure-Activity Relationship, Sulfonamides, Molecular Structure, Cell Wall, Drug Discovery, Antitubercular Agents, Humans, Hep G2 Cells, Microbial Sensitivity Tests, Mycobacterium tuberculosis
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9
المؤلفون: Dom Bellini, Neil G. Paterson, Grant A. Boyle, Hector Newman, Frank von Delft, Alen Krajnc, Kelly Chibale, Robert Lesniak, Katherine McAuley, Jürgen Brem, Christopher J. Schofield, Charles J. Eyermann, Christopher G. Dowson, Mukesh Gangar
المصدر: Journal of medicinal chemistry. 64(15)
مصطلحات موضوعية: inorganic chemicals, Boron Compounds, Models, Molecular, RM, Penicillin binding proteins, medicine.drug_class, Antibiotics, chemistry.chemical_element, Crystal structure, Microbial Sensitivity Tests, medicine.disease_cause, Crystallography, X-Ray, beta-Lactamases, RS, 03 medical and health sciences, Structure-Activity Relationship, Nucleophile, Drug Discovery, medicine, Penicillin-Binding Proteins, QD, Boron, 030304 developmental biology, 0303 health sciences, Vaborbactam, Binding Sites, Dose-Response Relationship, Drug, Molecular Structure, 030306 microbiology, Chemistry, Pseudomonas aeruginosa, QP, 3. Good health, Anti-Bacterial Agents, High-Throughput Screening Assays, Crystallography, Molecular Medicine, Antibacterial activity, beta-Lactamase Inhibitors
وصف الملف: application/pdf
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المؤلفون: Wei-Sheng Huang, Sara Nadworny, Narayana Narasimhan, Charles J. Eyermann, David C. Dalgarno, Victor M. Rivera, William C. Shakespeare
المصدر: Cancer Research. 82:3342-3342
مصطلحات موضوعية: Cancer Research, Oncology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::3b478b2d980afa91a4eec642fa30c3f7
https://doi.org/10.1158/1538-7445.am2022-3342