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1
المؤلفون: Mark J. O'Connor, Alan Lau, Keith W. Caldecott, Niall M.B. Martin, David Rudge, Jos Jonkers, Sven Rottenberg, Marina Pajic, Robert H. Bradbury, Attilla Ting, Bastiaan Evers, Charlotte Knights, Louise Jones, Janneke E. Jaspers, Henry Brown, Rajesh Odedra, Aaron N. Cranston, Stuart L. Rulten, Lenka Oplustil O'Connor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2109b65c80b64c5dc8e0c07cc7793822
https://doi.org/10.1158/0008-5472.c.6508109 -
2
المؤلفون: Mark J. O'Connor, Alan Lau, Keith W. Caldecott, Niall M.B. Martin, David Rudge, Jos Jonkers, Sven Rottenberg, Marina Pajic, Robert H. Bradbury, Attilla Ting, Bastiaan Evers, Charlotte Knights, Louise Jones, Janneke E. Jaspers, Henry Brown, Rajesh Odedra, Aaron N. Cranston, Stuart L. Rulten, Lenka Oplustil O'Connor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::730097b7c140c8178ff65dd44a170b76
https://doi.org/10.1158/0008-5472.22410926.v1 -
3
المؤلفون: Niall M. B. Martin, Bastiaan Evers, Charlotte Knights, Janneke E. Jaspers, Jos Jonkers, Attilla Ting, Henry Brown, Keith W. Caldecott, Sven Rottenberg, Rajesh Odedra, Lenka Oplustil O'Connor, Robert Hugh Bradbury, Aaron Cranston, David Alan Rudge, Mark J. O'Connor, Marina Pajic, Louise J. Jones, Alan Lau, Stuart L. Rulten
المصدر: Cancer Research. 76:6084-6094
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, DNA Repair, medicine.medical_treatment, Genes, BRCA1, Synthetic lethality, Poly(ADP-ribose) Polymerase Inhibitors, Pharmacology, Biology, Q1, Piperazines, Olaparib, Mice, 03 medical and health sciences, chemistry.chemical_compound, Piperidines, Bone Marrow, Cell Line, Tumor, Drug Discovery, Temozolomide, medicine, Animals, Humans, ATP Binding Cassette Transporter, Subfamily B, Member 1, PARP Inhibitor AZD2461, Chemotherapy, Cancer, Neoplasms, Experimental, medicine.disease, Xenograft Model Antitumor Assays, Rats, 3. Good health, Dacarbazine, 030104 developmental biology, medicine.anatomical_structure, Oncology, Tolerability, chemistry, PARP inhibitor, Phthalazines, Bone marrow, Poly(ADP-ribose) Polymerases, DNA Damage
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::318c6f6c6cc972443af48c50dbf1283f
https://doi.org/10.1158/0008-5472.can-15-3240 -
4
المؤلفون: Xavier Jacq, Martin Stockley, Karl Richard Gibson, Charlotte Knights, Jennifer Ward, Lauren McLellan, Jeanine A. Harrigan, Gavin A. Whitlock, Edward W. Tate
مصطلحات موضوعية: Proteomics, 0301 basic medicine, EXPRESSION, Ubiquitin-Specific Proteases, Biochemistry & Molecular Biology, INHIBITION, Molecular Probe Techniques, HIF-1-ALPHA, Biochemistry, Deubiquitinating enzyme, Small Molecule Libraries, 03 medical and health sciences, Cell Line, Tumor, Neoplasms, Humans, Pyrroles, PROBE, DEUBIQUITINATION, Science & Technology, biology, Proteomic Profiling, ACTIVE-SITE, Organic Chemistry, PATHWAYS, General Medicine, 06 Biological Sciences, REACTIVITY, Cell biology, 030104 developmental biology, Cell culture, Alkynes, Molecular Probes, DEUBIQUITYLATING ENZYMES, ATM, Cancer cell, biology.protein, Molecular Medicine, Molecular probe, 03 Chemical Sciences, Life Sciences & Biomedicine, Deubiquitination
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8d98c10d4d8599a2af2f3c449a4c023f
http://hdl.handle.net/10044/1/43848 -
5دورية أكاديمية
المؤلفون: Hannah Farmer, Nuala McCabe, Christopher J. Lord, Andrew N. J. Tutt, Damian A. Johnson, Tobias B. Richardson, Manuela Santarosa, Krystyna J. Dillon, Ian Hickson, Charlotte Knights, Niall M.
المصدر: Nature, Nature. 434(7035):917-921
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6
المؤلفون: Xiao-Ling Fan Cockcroft, Graeme C. M. Smith, Marc Geoffrey Hummersone, David R. Newell, Mark Frigerio, Heather Mary Ellen Duggan, Olivier Barbeau, Christine Bailey, Nicola J. Curtin, Bernard T. Golding, Ian R. Hardcastle, Caroline Richardson, Charlotte Knights, Roger J. Griffin, Ben Spittle, Celine Cano, Keith Allan Menear
المصدر: Journal of medicinal chemistry. 53(24)
مصطلحات موضوعية: Cell Membrane Permeability, Stereochemistry, Pyridines, DNA-Dependent Protein Kinase, DNA-Activated Protein Kinase, Pyrimidinones, Thiophenes, Quinolones, Small Molecule Libraries, chemistry.chemical_compound, Structure-Activity Relationship, Morpholine, Drug Discovery, Moiety, Humans, Benzopyrans, Protein kinase A, Furans, IC50, Chemotype, Biological activity, chemistry, Chemical engineering, Molecular Medicine, DNA, DNA Damage, HeLa Cells
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7
المؤلفون: Xavier Jacq, Niall M. B. Martin, Stephen P. Jackson, Helen Robinson, Lisa Smith, Aaron Cranston, Yaara Ofir-Rosenfeld, Charlotte Knights, Jeanine A. Harrigan, Kemp Mark Ian
المصدر: Cancer Research. 75:1728-1728
مصطلحات موضوعية: Genetics, Cancer Research, Oncogene, DNA damage, Drug discovery, Cancer, Synthetic lethality, Biology, medicine.disease, Oncology, In vivo, Cell culture, Cancer research, medicine, Homologous recombination
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::20e2465ebcfedccbd255f4be29a3595c
https://doi.org/10.1158/1538-7445.am2015-1728 -
8
المؤلفون: Krystyna J. Dillon, Niall M. B. Martin, Ian Hickson, Andrew Tutt, Manuela Santarosa, Tobias B. Richardson, Damian A. Johnson, Charlotte Knights, Christopher J. Lord, Stephen P. Jackson, Hannah Farmer, Graeme C. M. Smith, Alan Ashworth, Nuala McCabe
المصدر: Nature. 434(7035)
مصطلحات موضوعية: DNA Repair, DNA repair, Cell Survival, Genes, BRCA2, Genes, BRCA1, Mice, Nude, Antineoplastic Agents, Apoptosis, Biology, Poly(ADP-ribose) Polymerase Inhibitors, Models, Biological, Substrate Specificity, Mice, PARP1, Neoplasms, Animals, Multidisciplinary, Base excision repair, DNA repair protein XRCC4, Xenograft Model Antitumor Assays, Homologous Recombination Pathway, PARP inhibitor, Mutation, Cancer research, DNA mismatch repair, Poly(ADP-ribose) Polymerases, Nucleotide excision repair, DNA Damage
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المؤلفون: James Carmichael, Richard S. Finn, Dennis J. Slamon, Aisling O'Shaughnessy, Mark J. O'Connor, Dylan Conklin, Charlotte Knights, Ondrej Kalous, Lucy Riches, A. Lau
المصدر: European Journal of Cancer Supplements. 6:175-176
مصطلحات موضوعية: Genetics, Cancer Research, Oncology, business.industry, PARP Inhibitor AZD2281, Cancer research, Medicine, DNA repair protein XRCC4, Homologous recombination, business, Triple-negative breast cancer
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المؤلفون: Helen Wombwell, Seock-Ah Im, Hyung-Seok Hur, Tae-You Kim, Young-Kwang Yoon, Do-Youn Oh, Sang Hyun Song, Mark J. O'Connor, Sae-Won Han, Lucy Riches, Ahrum Min, Yung-Jue Bang, Yi Gu, Charlotte Knights, Alan Lau
المصدر: Cancer Research. 70:1775-1775
مصطلحات موضوعية: Cisplatin, Cancer Research, business.industry, Cancer, Pharmacology, medicine.disease, Oxaliplatin, Olaparib, chemistry.chemical_compound, Oncology, chemistry, Apoptosis, Cancer cell, PARP inhibitor, medicine, Cytotoxic T cell, business, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::e7c8bd7710086a4b787d4dff96159eac
https://doi.org/10.1158/1538-7445.am10-1775