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1
المؤلفون: Liang Liu, Yasheen Zhou, Kurt Jarnagin, Charlotte Virtucio, Xiaoqing Fan, Yong-Kang Zhang, Fernando Rock, Wei Bu, Tsutomu Akama, David C. Sullivan, Yvonne Freund, Chen Dong, Anne Wu
المصدر: Journal of Pharmacology and Experimental Therapeutics. 347:615-625
مصطلحات موضوعية: Boron Compounds, Models, Molecular, Muscle Relaxation, Myocytes, Smooth Muscle, Aorta, Thoracic, Blood Pressure, Biology, Muscle, Smooth, Vascular, Rats, Sprague-Dawley, Jurkat Cells, Structure-Activity Relationship, Protein Phosphatase 1, Rats, Inbred SHR, Animals, Humans, Structure–activity relationship, Kinome, Phosphorylation, Protein kinase A, Protein Kinase Inhibitors, Rho-associated protein kinase, Pharmacology, rho-Associated Kinases, Kinase, Muscle, Smooth, Smooth muscle contraction, Rats, Trachea, Biochemistry, Cytokines, Molecular Medicine, Cytokine secretion, Muscle Contraction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9a61c7ae48bc6b47d1f668dbb71e4d37
https://doi.org/10.1124/jpet.113.207662 -
2Inhibition of Toll-Like Receptor-Mediated Inflammation In Vitro and In Vivo by a Novel Benzoxaborole
المؤلفون: Charlotte Virtucio, Kurt Jarnagin, Yvonne Freund, Chen Dong, Xiaoqin Fan, Wei Bu, Ana Gertrudes, Lisa Feng, Liang Liu, Tsutomu Akama, Holly Sexton, Shamra Martin, Chiao-Wen Chen, Anne Wu
المصدر: Journal of Pharmacology and Experimental Therapeutics. 344:436-446
مصطلحات موضوعية: Boron Compounds, Lipopolysaccharides, Male, Cell Survival, medicine.medical_treatment, Administration, Oral, Arthritis, Inflammation, Pharmacology, Drug Hypersensitivity, Mice, Oral administration, In vivo, medicine, Animals, Humans, Hypersensitivity, Delayed, Cells, Cultured, Mice, Inbred BALB C, Toll-like receptor, Dose-Response Relationship, Drug, business.industry, Anti-Inflammatory Agents, Non-Steroidal, Toll-Like Receptors, Bridged Bicyclo Compounds, Heterocyclic, medicine.disease, TLR2, Cytokine, Dermatitis, Allergic Contact, Immunology, Leukocytes, Mononuclear, TLR4, Cytokines, Molecular Medicine, Female, medicine.symptom, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::35733c4804935c88f905e51531f98e16
https://doi.org/10.1124/jpet.112.200030 -
3
المؤلفون: Yasheen Zhou, Charlotte Virtucio, Yvonne Mak, Diogo Baia, Maliwan Meewan, Shamra Martin, Shannon Jones-Iatauro, Holly Sexton, Joshua Dee, Chen Dong, Kurt Jarnagin, Grober Baltazar, Tsutomu Akama, Olga Zemska, Fernando Rock
المصدر: The Journal of pharmacology and experimental therapeutics. 358(3)
مصطلحات موضوعية: 0301 basic medicine, Boron Compounds, Models, Molecular, medicine.medical_specialty, Thymic stromal lymphopoietin, medicine.medical_treatment, Administration, Topical, Pharmacology, Biology, Dermatitis, Atopic, 03 medical and health sciences, Mice, Thymic Stromal Lymphopoietin, Internal medicine, Psoriasis, Catalytic Domain, medicine, Leukocytes, Animals, Phosphorylation, Cyclic AMP Response Element-Binding Protein, Skin, Mitogen-Activated Protein Kinase 1, Mitogen-Activated Protein Kinase 3, Kinase, Phosphodiesterase, Crisaborole, Atopic dermatitis, medicine.disease, Bridged Bicyclo Compounds, Heterocyclic, Cyclic Nucleotide Phosphodiesterases, Type 4, 030104 developmental biology, Cytokine, Endocrinology, Gene Expression Regulation, Molecular Medicine, Cytokines, Tumor necrosis factor alpha, Female, Phosphodiesterase 4 Inhibitors
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d29584d7d00d52630836ced5f18a7821
https://pubmed.ncbi.nlm.nih.gov/27353073 -
4
المؤلفون: Wei Bu, Daitao Chen, Charlotte Virtucio, Yong-Kang Zhang, Tsutomu Akama, Vincent Hernandez, Robert T. Jacobs, Yvonne Freund, Jacob J. Plattner, Anne Wu, Yang Liu, Liang Liu, Chen Dong, Matthew Orr, Kurt Jarnagin
المصدر: Bioorganicmedicinal chemistry letters. 23(21)
مصطلحات موضوعية: Boron Compounds, Lipopolysaccharides, Lipopolysaccharide, medicine.drug_class, medicine.medical_treatment, Clinical Biochemistry, Interleukin-1beta, Anti-Inflammatory Agents, Pharmaceutical Science, Arthritis, Pharmacology, Biochemistry, Peripheral blood mononuclear cell, Anti-inflammatory, chemistry.chemical_compound, Mice, Structure-Activity Relationship, Pharmacokinetics, Drug Discovery, medicine, Benzene Derivatives, Animals, Interleukin 6, Molecular Biology, biology, Interleukin-6, Tumor Necrosis Factor-alpha, Organic Chemistry, medicine.disease, Arthritis, Experimental, Cytokine, chemistry, biology.protein, Leukocytes, Mononuclear, Molecular Medicine, Tumor necrosis factor alpha
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المؤلفون: Yong-Kang Zhang, Chen Dong, Marcelo Sales, Yvonne Freund, Anne Wu, James A. Nieman, Liang Liu, Jacob J. Plattner, Rajeshwar Singh, Charlotte Virtucio, Xiaoqing Fan, Richard Kimura, Kurt Jarnagin, Rashmi Sharma, Xiaosong Lu, Tsutomu Akama
المصدر: Bioorganicmedicinal chemistry letters. 23(6)
مصطلحات موضوعية: Boron Compounds, Lipopolysaccharides, Lipopolysaccharide, medicine.drug_class, Stereochemistry, medicine.medical_treatment, Clinical Biochemistry, Interleukin-1beta, Anti-Inflammatory Agents, Pharmaceutical Science, Pharmacology, Biochemistry, Peripheral blood mononuclear cell, Anti-inflammatory, chemistry.chemical_compound, Mice, Structure-Activity Relationship, Pharmacokinetics, Drug Discovery, medicine, Animals, Humans, Molecular Biology, Benzoxazoles, Interleukin-6, Tumor Necrosis Factor-alpha, Organic Chemistry, Bridged Bicyclo Compounds, Heterocyclic, Kinetics, Cytokine, chemistry, Leukocytes, Mononuclear, Molecular Medicine, Tumor necrosis factor alpha, Half-Life, Protein Binding
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6
المؤلفون: Yvonne Freund, Chen Dong, Charlotte Virtucio-Frates, Fernando Rock, Yvonne Mak, Yasheen Zhou, Lee Zane, Kurt Jarnagin
المصدر: The Journal of Immunology. 194:57.28-57.28
مصطلحات موضوعية: Immunology, Immunology and Allergy
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::6c7df6b648fdabcf1b0983edab9de650
https://doi.org/10.4049/jimmunol.194.supp.57.28