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المؤلفون: Matthew D. Hill, Haiquan Fang, Derek Norris, George V. Delucca, Hong Huang, Mikkel DeBenedetto, Claude Quesnelle, William D. Schmitz, John S. Tokarski, Steven Sheriff, Chunhong Yan, Caroline Fanslau, Zuzana Haarhoff, Christine Huang, Melissa Kramer, Shilpa Madari, Krista Menard, Laura Monereau, John Morrison, Nirmala Raghavan, Eric E. Shields, Jean Simmermacher-Mayer, Michael Sinz, Ching Kim Tye, Richard Westhouse, Chunshan Xie, Haiying Zhang, Lisa Zhang, Tatyana Zvyaga, Francis Lee, Ashvinikumar V. Gavai, Andrew P. Degnan
المصدر: ACS Medicinal Chemistry Letters. 13:1165-1171
مصطلحات موضوعية: Organic Chemistry, Drug Discovery, Biochemistry
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المؤلفون: Ching Kim Tye, Chunhong Yan, Sarah C. Traeger, Wayne Vaccaro, Yingru Zhang, Gerry Everlof, Jianqing Li, Henry Yip, Peng Li, John T. Hunt, Michael A. Poss, Gregory D. Vite, Mussari Christopher P, Steven Sheriff, Asoka Ranasinghe, Haiying Zhang, Richard A. Westhouse, Dharmpal S. Dodd, Richard Rampulla, Zheng Yang, Frank Marsilio, Derek J. Norris, Wen-Ching Han, Tram N. Huynh, Yufen Zhao, Patrice Gill, Nirmala Raghavan, Lalgudi S. Harikrishnan, Ashvinikumar V. Gavai, Susan Wee, John S. Tokarski, Dauh-Rurng Wu, Arvind Mathur, Mei-Li Wen, Huiping Zhang, David R. Tortolani, George V. Delucca, Krista Menard, Francis Y. Lee, Claude A. Quesnelle, Dawn Sun, Vijay T. Ahuja, Daniel O'malley, Christine Huang, Muthoni G. Kamau
المصدر: Journal of Medicinal Chemistry. 64:14247-14265
مصطلحات موضوعية: Drug, Proline, Phenylalanine, media_common.quotation_subject, Carbazoles, Administration, Oral, Antineoplastic Agents, Cell Cycle Proteins, Computational biology, BET inhibitor, Structure-Activity Relationship, Pharmacokinetics, In vivo, Drug Discovery, Transcriptional regulation, Humans, Potency, media_common, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Tryptophan, Signal transducing adaptor protein, Bromodomain, Molecular Medicine, Transcription Factors
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المؤلفون: Chunhong Yan, Francis Y. Lee, Ashvinikumar V. Gavai, Melissa Kramer, Frank Marsilio, Eric Shields, Laura Monereau, Zuzana Haarhoff, Richard A. Westhouse, Lisa Zhang, Gerry Everlof, John S. Tokarski, Matthew D. Hill, Tatyana Zvyaga, Asoka Ranasinghe, Carolynn Fanslau, Ching Kim Tye, Steven Sheriff, Christine Huang, Andrew P. Degnan, Krista Menard, John Morrison, Haiquan Fang
المصدر: Bioorganic & Medicinal Chemistry Letters. 44:128108
مصطلحات موضوعية: Clinical Biochemistry, Pharmaceutical Science, Structural diversity, Antineoplastic Agents, Biochemistry, BET inhibitor, Mice, Structure-Activity Relationship, Drug Development, Drug Discovery, medicine, Animals, Humans, Moiety, Potency, Mouse tumor, Molecular Biology, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Organic Chemistry, Proteins, Cancer, Triazoles, medicine.disease, Combinatorial chemistry, Bromodomain, Molecular Medicine, Multiple Myeloma, Carbolines
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المؤلفون: Zhanbin Wang, Randy C. Dockens, Ching Chiang Su, Yingru Zhang, Michael J. Hageman, Blisse Vakkalagadda, Chunlei Wang, Ching Kim Tye
المصدر: International journal of pharmaceutics. 514(2)
مصطلحات موضوعية: Drug, Drug Liberation, Digoxin, Chemical Phenomena, media_common.quotation_subject, Drug Compounding, Flurbiprofen, Pharmaceutical Science, Pharmacology, 030226 pharmacology & pharmacy, 03 medical and health sciences, 0302 clinical medicine, medicine, Dissolution testing, Drug Interactions, Omeprazole, media_common, Chromatography, Chemistry, Hydrogen-Ion Concentration, Drug Combinations, 030220 oncology & carcinogenesis, Compatibility (mechanics), Pravastatin, medicine.drug
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المؤلفون: Michael M. Morgen, Roy Haskell, Ching Kim Tye, Kimberly A. Foster
المصدر: Discovering and Developing Molecules with Optimal Drug-Like Properties ISBN: 9781493913985
مصطلحات موضوعية: Risk analysis (engineering), Process (engineering), Computer science, Scalability, Stability (learning theory), Key (cryptography), Timeline, Adaptation (computer science), Chemical space
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::278a4c20d8daf8e80b1ce8ea68f73ecf
https://doi.org/10.1007/978-1-4939-1399-2_3 -
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المؤلفون: Valerie E. Doyle, Richard Weaver, Ching-Kim Tye, Alan H. Fairlamb, Michael P. Barrett, Ganasan Kasinathan, Ian H. Gilbert, Reto Brun
المصدر: Bioorganic & Medicinal Chemistry Letters. 8:811-816
مصطلحات موضوعية: Adenosine, Trypanosoma brucei brucei, Clinical Biochemistry, Protozoan Proteins, Pharmaceutical Science, Trypanosoma brucei, Biochemistry, Chemical synthesis, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Polyamines, medicine, Animals, Molecular Biology, biology, Chemistry, Organic Chemistry, Kinetoplastida, Biological Transport, Biological activity, biology.organism_classification, Trypanocidal Agents, In vitro, Adenosine transporter, Kinetics, Molecular Medicine, Indicators and Reagents, Carrier Proteins, Polyamine, medicine.drug
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المؤلفون: Alan H. Fairlamb, Reto Brun, Richard Weaver, Valerie E. Doyle, Ian H. Gilbert, Ganasan Kasinathan, Ching-Kim Tye, Michael P. Barrett
المصدر: ChemInform. 29
مصطلحات موضوعية: chemistry.chemical_compound, Biochemistry, Chemistry, Substrate (chemistry), General Medicine, Polyamine, Adenosine transporter
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المؤلفون: Patrice Gill, Daniel O'malley, Mary Ellen Cvijic, George L. Trainor, Gregory D. Vite, Yingru Zhang, Richard Rampulla, Richard A. Westhouse, Celia D’Arienzo, Derek J. Norris, Wen-Ching Han, Ching Su, Mei-Li Wen, Libing Chen, Arvind Mathur, Andrew J. Tebben, Brian E. Fink, Bruce S. Fischer, Robin Moore, Francis Y. Lee, David Rodrigues, Qian Ruan, Gerry Everlof, Weifang Shan, John T. Hunt, Claude A. Quesnelle, Soong-Hoon Kim, Krista Menard, Dauh-Rurng Wu, Asoka Ranasinghe, Zheng Yang, Yufen Zhao, Ashvinikumar V. Gavai, Aaron Balog, Haiqing Wang, Ching Kim Tye, Melissa Yarde
المصدر: Cancer Research. 74:1643-1643
مصطلحات موضوعية: Gerontology, Cancer Research, Angiogenesis, Colorectal cancer, business.industry, Notch signaling pathway, medicine.disease, Metastasis, Breast cancer, Oncology, Cancer stem cell, Apoptosis, Cancer research, medicine, business, Transcription factor
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::761271a037a354d0d93f3b39b4fca9c3
https://doi.org/10.1158/1538-7445.am2014-1643 -
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المؤلفون: Gregory E. Amidon, Changquan Calvin Sun, Ching Kim Tye
المصدر: Journal of pharmaceutical sciences. 94(3)
مصطلحات موضوعية: Materials science, Time Factors, Compressive Strength, Compaction, Pharmaceutical Science, Compression (physics), Dosage form, Tableting, Compressive strength, Tensile Strength, Ultimate tensile strength, Compressibility, Composite material, Porosity, Tablets