-
1
المؤلفون: Steven C. R. Williams, Ndaba Mazibuko, Owen O’Daly, Christian Zurth, Fiona Patrick, Christian Kappeler, Iris Kuss, Patricia E. Cole
المصدر: Targeted Oncology. 18:403-413
مصطلحات موضوعية: Cancer Research, Oncology, Pharmacology (medical)
-
2
المؤلفون: Päivi Taavitsainen, Hille Gieschen, Christian Zurth, Mikko Koskinen, Clemens-Jeremias von Bühler, Karsten Denner, Annamari Vuorela, Michael Niehues, Timo Korjamo, Natalia A. Jungmann, Marja Kähkönen, Pirjo Nykänen, Olaf Prien
المصدر: Drug Metabolism and Disposition. 49:420-433
مصطلحات موضوعية: Adult, Male, Glucuronidation, Pharmaceutical Science, Drug Elimination Routes, Reductase, 030226 pharmacology & pharmacy, Mass Spectrometry, Excretion, 03 medical and health sciences, Glucuronides, 0302 clinical medicine, Androgen Receptor Antagonists, Cytochrome P-450 CYP3A, Humans, Biotransformation, Active metabolite, Pharmacology, Chromatography, CYP3A4, Chemistry, Metabolism, Healthy Volunteers, Pharmaceutical Solutions, 030220 oncology & carcinogenesis, UDP-Glucuronosyltransferase 1A9, Pyrazoles, Scintillation Counting, Stereoselectivity, Oxidation-Reduction, Drug metabolism
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::3b42599ea99983d8c72a5a26ff4bf32e
https://doi.org/10.1124/dmd.120.000309 -
3
المؤلفون: Gary Wilkinson, Robert Fricke, Timo Korjamo, Mikko Koskinen, Olaf Prien, Hille Gieschen, Kristina Graudenz, Karsten Denner, Michaela Bairlein, Clemens-Jeremias Von Bühler, Christian Zurth
المصدر: European Journal of Drug Metabolism and Pharmacokinetics
مصطلحات موضوعية: Male, Clinical chemistry, Midazolam, MEDLINE, Pharmacy, Pharmacology, 030226 pharmacology & pharmacy, 03 medical and health sciences, Prostate cancer, 0302 clinical medicine, Cytochrome P-450 Enzyme System, Humans, Medicine, Drug Interactions, Pharmacology (medical), Original Research Article, Rosuvastatin Calcium, Cells, Cultured, Aged, business.industry, Antagonist, Cytochrome P-450 CYP3A Inducers, Membrane Transport Proteins, Middle Aged, medicine.disease, Dabigatran, Androgen receptor, Clinical trial, Darolutamide, Enzyme Induction, 030220 oncology & carcinogenesis, Microsomes, Liver, Cytochrome P-450 CYP3A Inhibitors, Pyrazoles, Female, Itraconazole, Rifampin, business
-
4
المؤلفون: Christian Zurth, Pirjo Nykänen, Gary Wilkinson, Päivi Taavitsainen, Annamari Vuorela, Funan Huang, Susanne Reschke, Mikko Koskinen
المصدر: Clinical pharmacokinetics. 61(4)
مصطلحات موضوعية: Pharmacology, Male, Clinical Trials as Topic, Receptors, Androgen, Androgen Receptor Antagonists, Humans, Pyrazoles, Pharmacology (medical), Healthy Volunteers
-
5
المؤلفون: Hille Gieschen, Mikko Koskinen, Pirjo Nykänen, Christian Zurth, Timo Korjamo
المصدر: Drug metabolism letters. 14(1)
مصطلحات موضوعية: Male, Mice, Inbred BALB C, Chemistry, Biochemistry (medical), Clinical Biochemistry, Cmax, Diastereomer, Pharmaceutical Science, Plasma protein binding, Metabolism, Pharmacology, 030226 pharmacology & pharmacy, In vitro, 03 medical and health sciences, Mice, 0302 clinical medicine, Pharmacokinetics, In vivo, 030220 oncology & carcinogenesis, Androgen Receptor Antagonists, Animals, Pyrazoles, Pharmacology (medical), Active metabolite, Chromatography, Liquid
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ea44c126bf405b634aca1db4e12a1874
https://pubmed.ncbi.nlm.nih.gov/32436836 -
6
المؤلفون: Olaf Prien, Iris Kuss, Kristina Graudenz, Karim Fizazi, Bart Ploeger, Gustavo Borghesi, Teuvo L.J. Tammela, Neal D. Shore, Robert Fricke, Jonathan Moss, Hille Gieschen, Oana Petrenciuc, Frank Verholen, Christian Zurth, Mikko Koskinen, Matthew R. Smith
المصدر: Targeted Oncology
مصطلحات موضوعية: 0301 basic medicine, Male, Cancer Research, medicine.medical_specialty, Drug-Related Side Effects and Adverse Reactions, Population, Antineoplastic Agents, Comorbidity, Placebo, law.invention, Placebos, 03 medical and health sciences, Prostate cancer, 0302 clinical medicine, Randomized controlled trial, Double-Blind Method, law, Internal medicine, medicine, Androgen Receptor Antagonists, Humans, Pharmacology (medical), Drug Interactions, Castration, Original Research Article, Neoplasm Metastasis, Rosuvastatin Calcium, education, Adverse effect, Aged, Polypharmacy, Aged, 80 and over, education.field_of_study, business.industry, Anticholesteremic Agents, Incidence, Prostatic Neoplasms, Middle Aged, medicine.disease, Clinical trial, 030104 developmental biology, Darolutamide, Oncology, 030220 oncology & carcinogenesis, Pyrazoles, Neoplasm Recurrence, Local, business
-
7
المؤلفون: Nobuaki Matsubara, Hirofumi Mukai, Ako Hosono, Mai Onomura, Masaoki Sasaki, Yoko Yajima, Kensei Hashizume, Masanobu Yasuda, Miho Uemura, Christian Zurth
المصدر: Cancer Chemotherapy and Pharmacology. 80:1073-1077
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, 03 medical and health sciences, Cancer Research, 030104 developmental biology, 0302 clinical medicine, Oncology, 030220 oncology & carcinogenesis, Pharmacology (medical), Toxicology
-
8
المؤلفون: Ako Hosono, Kensei Hashizume, Masanobu Yasuda, Christian Zurth, Masaoki Sasaki, Yoko Yajima, Miho Uemura, Hirofumi Mukai, Nobuaki Matsubara, Mai Onomura
المصدر: Cancer Chemotherapy and Pharmacology
مصطلحات موضوعية: Male, Oncology, Cancer Research, medicine.medical_specialty, Nausea, 030232 urology & nephrology, Darolutamide, Pharmacokinetic, Phase 1, Toxicology, Gastroenterology, 03 medical and health sciences, Prostate cancer, 0302 clinical medicine, Androgen receptor antagonist, Asian People, Pharmacokinetics, Internal medicine, Androgen Receptor Antagonists, medicine, Humans, Pharmacology (medical), Neoplasm Metastasis, Adverse effect, Aged, Pharmacology, business.industry, Incidence (epidemiology), medicine.disease, ODM-201, Prostatic Neoplasms, Castration-Resistant, Fasting Status, 030220 oncology & carcinogenesis, Cohort, Pyrazoles, Original Article, Erratum, medicine.symptom, business
-
9
المؤلفون: Matthew R. Smith, Christian Zurth, Karim Fizazi, M-A. Le Berre, T Tammela, Iris Kuss, Oana Petrenciuc, N.D. Shore
المصدر: Annals of Oncology. 31:S1327-S1328
مصطلحات موضوعية: Oncology, medicine.medical_specialty, Treatment response, business.industry, Hematology, Castration resistant, medicine.disease, Prostate cancer, Darolutamide, Tolerability, Internal medicine, medicine, Non metastatic, In patient, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::b370f67ab203c1d963482d90b0e4c9fa
https://doi.org/10.1016/j.annonc.2020.10.442 -
10
المؤلفون: Shankar Srinivasan, Marie-Aude Le Berre, Teuvo L.J. Tammela, Karim Fizazi, Matthew R. Smith, Christopher Michael Pieczonka, Christian Zurth, Oana Petrenciuc, David L. Morris, Iris Kuss, Jeanny B. Aragon-Ching, Neal D. Shore
المصدر: Journal of Clinical Oncology. 39:5079-5079
مصطلحات موضوعية: Oncology, Cancer Research, medicine.medical_specialty, Treatment response, business.industry, medicine.disease, Prostate cancer, Darolutamide, Tolerability, Quality of life, Internal medicine, Toxicity, medicine, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::248864529c7b125bf5c2d7939fca5eb2
https://doi.org/10.1200/jco.2021.39.15_suppl.5079