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1
المؤلفون: Benoit Pasquier, Youssef El-Ahmad, Bruno Filoche-Rommé, Christine Dureuil, Florence Fassy, Pierre-Yves Abecassis, Magali Mathieu, Thomas Bertrand, Tsiala Benard, Cédric Barrière, Samira El Batti, Jean-Philippe Letallec, Véronique Sonnefraud, Maurice Brollo, Laurence Delbarre, Véronique Loyau, Fabienne Pilorge, Luc Bertin, Patrick Richepin, Jérôme Arigon, Jean-Robert Labrosse, Jacques Clément, Florence Durand, Romain Combet, Pierre Perraut, Vincent Leroy, Frédéric Gay, Dominique Lefrançois, François Bretin, Jean-Pierre Marquette, Nadine Michot, Anne Caron, Christelle Castell, Laurent Schio, Gary McCort, Hélène Goulaouic, Carlos Garcia-Echeverria, Baptiste Ronan
المصدر: Journal of Medicinal Chemistry. 58:376-400
مصطلحات موضوعية: Male, Models, Molecular, Stereochemistry, Molecular Sequence Data, Antineoplastic Agents, Mice, SCID, Pyrimidinones, Plasma protein binding, Crystallography, X-Ray, Rats, Sprague-Dawley, chemistry.chemical_compound, In vivo, Cell Line, Tumor, Neoplasms, Morpholine, Drug Discovery, Animals, Humans, Transferase, Amino Acid Sequence, Enzyme Inhibitors, Trifluoromethyl, Molecular Structure, Sequence Homology, Amino Acid, Drug discovery, Kinase, fungi, Synthon, Bridged Bicyclo Compounds, Heterocyclic, Class III Phosphatidylinositol 3-Kinases, Xenograft Model Antitumor Assays, Protein Structure, Tertiary, Models, Chemical, chemistry, Area Under Curve, Thermodynamics, Molecular Medicine, Caco-2 Cells, HeLa Cells, Protein Binding
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2
المؤلفون: Laurent Vidard, Christine Dureuil-Sizaire, Jérémy Baudhuin, Lionel Vescovi, Laurence Durand, Véronique Sierra, Eric Parmantier
المصدر: Cancer Research. 79:1524-1524
مصطلحات موضوعية: Cancer Research, Oncology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::4914ade70f90f7d1742458a2cef2fd30
https://doi.org/10.1158/1538-7445.am2019-1524 -
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المؤلفون: Christine Dureuil, Jean-Pierre Marquette, Marie-France Bachelot, Baptiste Ronan, Carlos Garcia-Echeverria, Magali Mathieu, Annabelle Lamberton, Benoit Pasquier, Florence Fassy, Youssef El-Ahmad, Thomas Bertrand, Laurence Durand, Bruno Filoche-Romme, Hélène Goulaouic, Laurent Schio, O. Flamand, Lionel Vescovi
المصدر: Nature chemical biology. 10(12)
مصطلحات موضوعية: Gene isoform, Pyridines, Gene Expression, Antineoplastic Agents, Endosomes, Pyrimidinones, Biology, Kidney, Adenosine Triphosphate, Catalytic Domain, Cell Line, Tumor, Autophagy, Humans, Everolimus, Kinase activity, Molecular Biology, Protein Kinase Inhibitors, PI3K/AKT/mTOR pathway, Cell Proliferation, Sirolimus, Kinase, TOR Serine-Threonine Kinases, fungi, Drug Synergism, Cell Biology, Small molecule, Class III Phosphatidylinositol 3-Kinases, Recombinant Proteins, Cell biology, Molecular Docking Simulation, Kinetics, Cell culture, Signal transduction, Lysosomes, Signal Transduction
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المؤلفون: Manuela Argentini, Isabelle Delumeau, Bohdan Wasylyk, Roberto Salvi, Laurent Debussche, Christine Dureuil, Joseph Abecassis, Christine Wasylyk
المصدر: Oncogene. 18:1921-1934
مصطلحات موضوعية: Cancer Research, Programmed cell death, Cell cycle checkpoint, Tumor suppressor gene, Cell Survival, Molecular Sequence Data, Biology, Proto-Oncogene Proteins, Tumor Cells, Cultured, Genetics, Humans, E2F1, Amino Acid Sequence, E2F, neoplasms, Molecular Biology, Cell Death, Effector, Cell Cycle, Nuclear Proteins, Proto-Oncogene Proteins c-mdm2, Apoptosis, Cell culture, Cancer research, Tumor Suppressor Protein p53, HeLa Cells
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::542fc87e1c123a26ae64055fbb23e6c4
https://doi.org/10.1038/sj.onc.1202528 -
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المؤلفون: Corinne Venot, Laurent Debussche, Emmanuel Conseiller, Nadège Gruel, Laurent Bracco, Bruno Tocque, Christine Dureuil, Jean-Luc Teillaud, Claude Caron de Fromentel
المصدر: Oncogene. 18(2)
مصطلحات موضوعية: Cancer Research, Transcription, Genetic, medicine.drug_class, Mutant, Genetic Vectors, Molecular Sequence Data, Biology, medicine.disease_cause, Monoclonal antibody, Transfection, Genetics, medicine, Tumor Cells, Cultured, Humans, Amino Acid Sequence, Molecular Biology, Immunoglobulin Fragments, DNA Primers, Expression vector, Base Sequence, Sequence Homology, Amino Acid, In vitro, Cell biology, Cytoplasm, Cell culture, Cancer research, Tumor Suppressor Protein p53, Carcinogenesis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::bfb4e3889bf8b069f3db1e13e9f7a4e1
https://pubmed.ncbi.nlm.nih.gov/9927212 -
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المؤلفون: Christine Dureuil, Laurent Bracco, Michel Maratrat, Laurent Debussche, Emmanuel Conseiller, Corinne Venot
المصدر: The EMBO journal. 17(16)
مصطلحات موضوعية: Cyclin-Dependent Kinase Inhibitor p21, Transcriptional Activation, Tumor suppressor gene, Proline, Repressor, Apoptosis, General Biochemistry, Genetics and Molecular Biology, Cell Line, Transactivation, Bcl-2-associated X protein, Transcription (biology), Cyclins, Proto-Oncogene Proteins, Humans, Promoter Regions, Genetic, Molecular Biology, Psychological repression, DNA Primers, Sequence Deletion, bcl-2-Associated X Protein, General Immunology and Microbiology, biology, Base Sequence, General Neuroscience, Cell Cycle, Antibodies, Monoclonal, Nuclear Proteins, Promoter, Proto-Oncogene Proteins c-mdm2, Molecular biology, TATA Box, Cell biology, DNA-Binding Proteins, Repressor Proteins, Proto-Oncogene Proteins c-bcl-2, biology.protein, Mdm2, Tumor Suppressor Protein p53, Reactive Oxygen Species, Research Article
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المصدر: Biochemistry. 32(43)
مصطلحات موضوعية: Leucine zipper, Proto-Oncogene Proteins c-jun, Molecular Sequence Data, Basic helix-loop-helix leucine zipper transcription factors, Biotin, Peptide, Biology, In Vitro Techniques, Biochemistry, DNA-binding protein, Iodine Radioisotopes, Xenopus laevis, Animals, Amino Acid Sequence, chemistry.chemical_classification, Leucine Zippers, bZIP domain, Peptide Fragments, Dissociation constant, Scintillation proximity assay, chemistry, Biotinylation, Luminescent Measurements, Oocytes, Female, Proto-Oncogene Proteins c-fos, Protein Binding, Signal Transduction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::95536208e5e443bcd1d93756a44eca1e
https://pubmed.ncbi.nlm.nih.gov/8218236