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1دورية أكاديمية
المؤلفون: Deborah J. Harvey, József Vuts, Antony Hooper, John C. Caulfield, Paul Finch, Christine M. Woodcock, Alan C. Gange, Jason W. Chapman, Michael A. Birkett, John A. Pickett
المصدر: Scientific Reports, Vol 14, Iss 1, Pp 1-11 (2024)
وصف الملف: electronic resource
Relation: https://doaj.org/toc/2045-2322
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2
المؤلفون: Philip J. Jewsbury, Rajesh Odedra, Alan Lau, Sylvie Guichard, James W.T. Yates, Kevin Blades, Gary Wilkinson, Kevin Michael Foote, Dan Heathcote, Turner Paul, Christine M. Wood, J. Willem M. Nissink, Zena Wilson, Thomas M. McGuire
المصدر: Journal of Medicinal Chemistry. 61:9889-9907
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Indoles, Chemical Phenomena, Morpholines, Molecular Conformation, Regulator, Antineoplastic Agents, Context (language use), Ataxia Telangiectasia Mutated Proteins, Mice, 03 medical and health sciences, chemistry.chemical_compound, 0302 clinical medicine, Pharmacokinetics, Cell Line, Tumor, Drug Discovery, Animals, Humans, Tissue Distribution, Protein Kinase Inhibitors, Clinical Trials as Topic, Sulfonamides, CYP3A4, Kinase, Drug discovery, Pyrimidines, 030104 developmental biology, chemistry, Cell culture, Sulfoxides, 030220 oncology & carcinogenesis, Cancer research, Molecular Medicine, Female, DNA
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3
المؤلفون: Rajesh Odedra, Sylvie S. Guichard, Philip J. Jewsbury, Abid Suleman, Christine M. Wood, Lorraine A. Hassall, Kevin Blades, Thomas M. McGuire, Pia Thommes, Xavier Jacq, Paula Perkins, Ian Hickson, Ken Page, J. Willem M. Nissink, Kevin Michael Foote, Kin Yip Tam, Shaun M. Fillery, Rebecca Broadhurst, Anna Cronin
المصدر: Journal of Medicinal Chemistry. 56:2125-2138
مصطلحات موضوعية: Models, Molecular, Radiosensitizer, Morpholines, Antineoplastic Agents, Cell Cycle Proteins, Ataxia Telangiectasia Mutated Proteins, Protein Serine-Threonine Kinases, Pharmacology, Crystallography, X-Ray, HeLa, Mice, Structure-Activity Relationship, chemistry.chemical_compound, In vivo, Drug Discovery, Animals, Humans, Structure–activity relationship, Protein Kinase Inhibitors, IC50, biology, Chemistry, Drug discovery, biology.organism_classification, Xenograft Model Antitumor Assays, In vitro, Pyrimidines, Molecular Medicine, Female, Growth inhibition, HeLa Cells
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4
المؤلفون: Michael James, Gordon A. Hamlin, Stefan Gerhardt, David Ryan, Nash Ian Alun, Attilla Ting, Stephen J. Norris, Galith Karoutchi, Chris De Savi, Neil Rankine, David J. Hargreaves, Christine M. Wood, Sarah V. Baker, Philip A. MacFaul, Andrew David Morley, Kostas Karabelas
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:4215-4219
مصطلحات موضوعية: Molecular model, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Stereoisomerism, Carboxamide, Matrix Metalloproteinase Inhibitors, Crystallography, X-Ray, Biochemistry, Structure-Activity Relationship, Catalytic Domain, Matrix Metalloproteinase 13, Drug Discovery, Hydrolase, medicine, Structure–activity relationship, Protease Inhibitors, Binding site, Molecular Biology, Binding Sites, biology, Chemistry, Organic Chemistry, Zinc, Enzyme inhibitor, biology.protein, Molecular Medicine, Selectivity
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5
المؤلفون: Peter Newham, Eleanor Henshaw, Philip A. MacFaul, Keith Oldham, Andrew David Morley, Neil Rankine, Christine M. Wood, David Elliot, Ken Page, Attilla Ting, Paul T. Sharpe
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:4832-4835
مصطلحات موضوعية: biology, Cell adhesion molecule, medicine.drug_class, Chemistry, Organic Chemistry, Clinical Biochemistry, Integrin, Pharmaceutical Science, Carboxamide, Biochemistry, In vitro, embryonic structures, Drug Discovery, cardiovascular system, medicine, biology.protein, Molecular Medicine, Structure–activity relationship, Potency, Binding site, Arginine binding, Molecular Biology
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6
المؤلفون: David Waterson, Julian A. Hudson, Michael James, Andrew D. Campbell, Turner Paul, Justin Bower, Benjamin P. McDermott, Christine M. Wood, Jon Winter, Philip J. Poyser, Alan Wellington Faull, John G. Cumming
المصدر: Bioorganicmedicinal chemistry letters. 22(12)
مصطلحات موضوعية: CCR2, medicine.drug_class, Stereochemistry, Receptors, CCR2, Clinical Biochemistry, hERG, Anti-Inflammatory Agents, Pharmaceutical Science, Carboxamide, CCR5 receptor antagonist, Pharmacology, Biochemistry, Piperazines, chemistry.chemical_compound, Chemokine receptor, Dogs, Drug Discovery, medicine, Animals, Humans, Molecular Biology, Inflammation, biology, Organic Chemistry, Ether-A-Go-Go Potassium Channels, Rats, Piperazine, chemistry, Drug Design, Lipophilicity, biology.protein, Molecular Medicine, Calcium, Lead compound, Hydrophobic and Hydrophilic Interactions, Protein Binding
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7
المؤلفون: David, Elliot, Eleanor, Henshaw, Philip A, MacFaul, Andrew D, Morley, Peter, Newham, Keith, Oldham, Ken, Page, Neil, Rankine, Paul, Sharpe, Attilla, Ting, Christine M, Wood
المصدر: Bioorganicmedicinal chemistry letters. 19(16)
مصطلحات موضوعية: Small Molecule Libraries, Structure-Activity Relationship, Binding Sites, Drug Design, Animals, Humans, Computer Simulation, Integrin alphaVbeta3, Oligopeptides, Rats
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8دورية أكاديمية
المؤلفون: Diego M. Magalhães, Miguel Borges, Raúl A. Laumann, Christine M. Woodcock, David M. Withall, John A. Pickett, Michael A. Birkett, Maria C. Blassioli-Moraes
المصدر: Frontiers in Ecology and Evolution, Vol 6 (2018)
مصطلحات موضوعية: cotton, kairomone, herbivore-induced plant volatiles, insect-plant interaction, semiochemicals, Evolution, QH359-425, Ecology, QH540-549.5
وصف الملف: electronic resource