-
1
المؤلفون: Jianxia Shi, Xiaoning Zhao, Samer Chmait, Mary Dovlatyan, Silke Miller, Kristin L. Andrews, Geraldine Hill Della Puppa, James J. S. Treanor, Dianna Lester-Zeiner, Carl Davis, Essa Hu, Christopher Biorn, Jessica Able, Hang Chen, Jennifer R. Allen, Ji Ma
المصدر: ACS Medicinal Chemistry Letters. 5:700-705
مصطلحات موضوعية: Stereochemistry, Organic Chemistry, Phosphodiesterase, Biochemistry, Cocrystal, Bioavailability, chemistry.chemical_compound, chemistry, Morpholine, Drug Discovery, Pyridine, Potency, PDE10A, Receptor
-
2
المؤلفون: Dianna Lester-Zeiner, Christopher Biorn, Essa Hu, Jianxia Shi, James J. S. Treanor, Sharon Zhao, Jennifer R. Allen, Amy Porter, Kristin L. Andrews, Samer Chmait, Shannon Rumfelt, Aaron C. Siegmund, Roxanne Kunz, Ning Chen, Hang Chen, Carl Davis, Ji Ma
المصدر: Journal of Medicinal Chemistry. 56:8781-8792
مصطلحات موضوعية: Male, Models, Molecular, Phosphodiesterase Inhibitors, Swine, Pharmacology, Rats, Sprague-Dawley, Structure-Activity Relationship, In vivo, Drug Discovery, Animals, Humans, Potency, Receptor, Cells, Cultured, chemistry.chemical_classification, Dose-Response Relationship, Drug, Molecular Structure, Phosphoric Diester Hydrolases, Phosphodiesterase, Ketones, Rats, Bioavailability, Enzyme, chemistry, Biochemistry, Drug Design, Molecular Medicine, Benzimidazoles, Efflux, PDE10A
-
3
المؤلفون: Dah-Ren Hwang, Geraldine Hill Della Puppa, Jamie Wong, Essa Hu, Thomas Nixey, Silke Miller, Hang Chen, Jessica Able, Dianna Lester-Zeiner, James J. S. Treanor, Robert Cho, Santosh Talreja, Roxanne Kunz, Jianxia Shi, Ji Ma, David C. Immke, Jennifer R. Allen, Christopher Biorn, Amy Porter, Klaus Michelsen, Shannon Rumfelt, Stephen Hitchcock
المصدر: Journal of Medicinal Chemistry. 55:4776-4787
مصطلحات موضوعية: Male, Phosphodiesterase Inhibitors, Aminopyridines, Striatum, In Vitro Techniques, Tritium, Permeability, Cell Line, Rats, Sprague-Dawley, Dogs, Tandem Mass Spectrometry, In vivo, TRACER, Drug Discovery, Animals, Humans, Tissue Distribution, ATP Binding Cassette Transporter, Subfamily B, Member 1, Radionuclide Imaging, Phosphoric Diester Hydrolases, Drug discovery, Chemistry, Brain, Phosphodiesterase, Stereoisomerism, Surface Plasmon Resonance, Molecular biology, Small molecule, Rats, Pyridazines, Rapid identification, Quinolines, Pyrazoles, Molecular Medicine, PDE10A, Radiopharmaceuticals, Chromatography, Liquid, Protein Binding
-
4
المؤلفون: Hu Ye, Tim Kazules, Ji Ma, Dianna Lester-Zeiner, Essa Hu, Santosh Talreja, Carl Davis, Charlie Glaus, Oliver R. Thiel, Ning Chen, Geraldine Hill Della Puppa, James J. S. Treanor, Shannon Rumfelt, Hui Hannah Dou, Roxanne Kunz, David C. Immke, Jessica Able, Jennifer R. Allen, Silke Miller, Xiaoning Zhao, Hang Chen, Jianxia Shi, Jamie Wong, Toni Williamson, Christopher Biorn, Amy Porter, Klaus Michelsen, Ada Chen
المصدر: The Journal of pharmacology and experimental therapeutics. 352(2)
مصطلحات موضوعية: Male, Fluorine Radioisotopes, Phosphodiesterase Inhibitors, Pharmacology, Mass Spectrometry, Rats, Sprague-Dawley, Radioligand Assay, Species Specificity, medicine, Distribution (pharmacology), Animals, Humans, Tissue Distribution, medicine.diagnostic_test, Molecular Structure, Chemistry, Drug discovery, Phosphoric Diester Hydrolases, Antagonist, Phosphodiesterase, Brain, Stereoisomerism, Surface Plasmon Resonance, Small molecule, Drug development, Positron emission tomography, Positron-Emission Tomography, Pyrazines, Molecular Medicine, Benzimidazoles, Female, PDE10A, Chromatography, Liquid, Papio, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d2114c0263395e74897b10174822cf2a
https://pubmed.ncbi.nlm.nih.gov/25502803