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1
المؤلفون: Ian B. Campbell, George E. Tranter, Ashley Paul Hancock, Christopher R Molloy, Karl Huffman, Gary I. Mills, Philip Charles Box, Ann Louise Walker, Gerard Martin Paul Giblin, Susan R. Doctrow, Susan Roomans, Bernard Malfroy
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:1367-1370
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, chemistry.chemical_element, Manganese, Electrophilic aromatic substitution, Biochemistry, Chemical synthesis, Antioxidants, 2,2'-Bipyridine, Superoxide dismutase, Structure-Activity Relationship, chemistry.chemical_compound, Bipyridine, Superoxides, Drug Discovery, Organometallic Compounds, Molecular Biology, chemistry.chemical_classification, biology, Superoxide Dismutase, Organic Chemistry, Hydrogen Peroxide, Catalase, Salicylates, Enzyme, Manganese Compounds, chemistry, biology.protein, Molecular Medicine
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2
المؤلفون: Lee Andrew Harrison, Michael Dennis Dowle, Harry Finch, Robin Andrew Smith, Pritom Shah, K.Abhhilash Kumar, Gill Fleetwood, Simon Teanby Hodgson, George W. Hardy, Graham Murkitt, Simon J. F. Macdonald, Graham G. A. Inglis, Christopher R Molloy, Geoffrey D. Clarke, Augustin Amour, Rosalind E Godward, Tony Padfield, Davina Humphreys, M. R. Johnson, Mary Dixon, Tadeusz Skarzynski, Onkar M. P. Singh
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:895-898
مصطلحات موضوعية: Lactams, Human neutrophil, Metabolic Clearance Rate, Clinical Biochemistry, Administration, Oral, Biological Availability, Pharmaceutical Science, Pharmacology, Biochemistry, Dogs, Drug Stability, Piperidines, Pharmacokinetics, Cricetinae, Drug Discovery, Animals, Molecular Biology, Short duration, Serpins, Bacteria, Pancreatic Elastase, Chemistry, Serine Endopeptidases, Organic Chemistry, Elastase, Bacterial Infections, Rats, Bioavailability, Orally active, Pharmacodynamics, Molecular Medicine, Crystallization, Leukocyte Elastase, Intracellular
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3
المؤلفون: Michael S. Anson, Keith Mills, Simon J. F. Macdonald, Doreen M. Buckley, Richard J. Upton, Lee Andrew Harrison, Catherine Risley, David J. Belton, Michael Dennis Dowle, Christopher R Molloy, Julie E. Spooner, Robin A.J. Smith
المصدر: Journal of Medicinal Chemistry. 41:3919-3922
مصطلحات موضوعية: chemistry.chemical_classification, Serine Proteinase Inhibitors, Lactams, biology, Bicyclic molecule, Neutrophils, Stereochemistry, Chemical synthesis, Piperazines, Pyrrolidine, Lactones, Structure-Activity Relationship, chemistry.chemical_compound, chemistry, Enzyme inhibitor, Drug Discovery, biology.protein, Lactam, Azetidines, Humans, Molecular Medicine, Structure–activity relationship, Enantiomer, Leukocyte Elastase, Lactone
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4
المؤلفون: Bernard Malfroy, Charlotte Atkin, Gary I. Mills, I. Anderson, J.C. Barnes, Tony Wong, Susan R. Doctrow, Ken A. Joy, Gill Brown, Christopher R Molloy, Peter Soden, H. Thomas R. Rupniak
المصدر: Neurotoxicity research. 2(2-3)
مصطلحات موضوعية: biology, Superoxide, General Neuroscience, Nitrotyrosine, Neurotoxicity, Toxicology, medicine.disease_cause, medicine.disease, Neuroprotection, Superoxide dismutase, chemistry.chemical_compound, Biochemistry, chemistry, medicine, biology.protein, Oxidative stress, Peroxynitrite, Free-radical theory of aging
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5
المؤلفون: Alan J. Wonacott, Rosalind E Godward, Gill Fleetwood, Robin Andrew Smith, Pritom Shah, Simon J. F. Macdonald, Martin R. Johnson, Christopher R Molloy, George Hardy, Simon Teanby Hodgson, Lee Andrew Harrison, Augustin Amour, Michael Dennis Dowle, Onkar M. P. Singh, Graham G. A. Inglis, Mary Dixon, Davina Humphreys, Geoffrey D. Clarke
المصدر: Journal of medicinal chemistry. 45(18)
مصطلحات موضوعية: Male, Models, Molecular, Pyrrolidines, Lactams, Swine, Crystallography, X-Ray, Chemical synthesis, Pyrrolidine, chemistry.chemical_compound, Structure-Activity Relationship, Dogs, In vivo, Drug Discovery, Structure–activity relationship, Animals, Combinatorial Chemistry Techniques, Humans, Pyrroles, Enzyme Inhibitors, Pancreatic elastase, Sulfonamides, biology, Molecular Structure, Chemistry, Elastase, Stereoisomerism, In vitro, Rats, Biochemistry, Enzyme inhibitor, biology.protein, Molecular Medicine, Leukocyte Elastase
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6
المؤلفون: Christopher R Molloy, Simon Teanby Hodgson, Robin A.J. Smith, Tadeusz Skarzynski, Onkar M. P. Singh, Rosalind E Godward, Julie E. Spooner, Harry Finch, Mary Dixon, K.Abhhilash Kumar, David J. Belton, Graham G. A. Inglis, Pritom Shah, Simon J. F. Macdonald, Graham Murkitt, Martin R. Johnson, Edward McDonald, Lee Andrew Harrison, Davina Humphreys, Gill Fleetwood, Geoffrey D. Clarke, George W. Hardy, Michael Dennis Dowle
المصدر: Bioorganic & Medicinal Chemistry Letters. 11:1249
مصطلحات موضوعية: Human neutrophil, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Elastase, Pharmaceutical Science, Biochemistry, Pyrrolidine, chemistry.chemical_compound, Orally active, chemistry, Drug Discovery, Molecular Medicine, Theology, Molecular Biology