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1
المؤلفون: Thao Ung, Ronald Robinson, Chrysanthe Spais, Justin Schreiber, Hussein Hallak, Jean Husten, Thelma S. Angeles, Jacquelyn Lyons, Yun Liu
المصدر: Bioanalysis. 13:575-585
مصطلحات موضوعية: Drug, media_common.quotation_subject, Clinical Biochemistry, Ligands, 030226 pharmacology & pharmacy, 01 natural sciences, Analytical Chemistry, Meso scale, 03 medical and health sciences, 0302 clinical medicine, Drug Development, Drug interference, Animals, Free drug, General Pharmacology, Toxicology and Pharmaceutics, media_common, Chromatography, Chemistry, Ligand binding assay, 010401 analytical chemistry, General Medicine, Nonhuman primate, 0104 chemical sciences, Medical Laboratory Technology, Pharmaceutical Preparations, Biomarker (medicine), Free form, Biomarkers
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2
المؤلفون: Sheryl L. Meyer, Jean Husten, Thelma S. Angeles, Chrysanthe Spais, Mark A. Ator, Seetha Murthy, Jennifer L. Mason, Mark S. Albom, Lisa Saville
المصدر: ASSAY and Drug Development Technologies. 10:551-557
مصطلحات موضوعية: DNA, Complementary, Drug Evaluation, Preclinical, Protein tag, Polymerase Chain Reaction, Antibodies, Receptor tyrosine kinase, Cell Line, Focal adhesion, Proto-Oncogene Proteins, Drug Discovery, Fluorescence Resonance Energy Transfer, Humans, Enzyme Inhibitors, Coloring Agents, c-Mer Tyrosine Kinase, biology, Kinase, Cellular Assay, Phosphotransferases, Receptor Protein-Tyrosine Kinases, Fusion protein, Antibodies, Anti-Idiotypic, Förster resonance energy transfer, Biochemistry, Data Interpretation, Statistical, Focal Adhesion Protein-Tyrosine Kinases, biology.protein, Molecular Medicine, Fluorescein, Tyrosine kinase
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::b5912b44be55c0e7bad9f066e4b6cbfc
https://doi.org/10.1089/adt.2011.439 -
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المؤلفون: Thomas J. Connors, Jie Qian, Zeck Huang, Joanne R. Mathiasen, Edward R. Bacon, Thelma S. Angeles, Mark J. Huffman, Emir Duzic, Joseph M. Salvino, Beth Ann McKenna, Hervé Schaffhauser, Robert J. McHugh, Lily D. Lu, George C. Morton, Beverly P. Holskin, Karla Kopec, Amy DiCamillo, Gerard C. Rosse, Chrysanthe Spais, Rabindranath Tripathy, Lisa D. Aimone
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:1421-1426
مصطلحات موضوعية: Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Antagonist, Pharmaceutical Science, Stereoisomerism, Biochemistry, Sulfone, chemistry.chemical_compound, In vivo, Drug Discovery, 5-HT6 receptor, Molecular Medicine, Pharmacophore, Receptor, Molecular Biology, 5-HT receptor
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المؤلفون: Beverly P. Holskin, Karla Kopec, Joanne R. Mathiasen, Amy DiCamillo, Babu G. Sundar, Thomas J. Connors, Emir Duzic, Edward R. Bacon, Gerard C. Rosse, Chrysanthe Spais, Thomas R. Bailey, Beth Ann McKenna, Rebecca A. Brown, Jie Qian, Derek Dunn, Mark J. Huffman, Joseph M. Salvino, Huang Zeqi, Lisa D. Aimone, Hervé Schaffhauser, Deborah Galinis, Thelma S. Angeles, Lily D. Lu, George C. Morton
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:120-123
مصطلحات موضوعية: biology, Organic Chemistry, Clinical Biochemistry, hERG, Pharmaceutical Science, Pharmacology, Biochemistry, Social recognition, chemistry.chemical_compound, chemistry, Drug Discovery, biology.protein, 5-HT6 receptor, Molecular Medicine, Structure–activity relationship, Serotonin Antagonists, Penetrant (biochemical), Receptor, Molecular Biology, 5-HT receptor
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5
المؤلفون: Ken Morii, Roberto A. Macina, Chrysanthe Spais, Harold Riethman, Dimitri G. Negorev, X.-L. Hu, Lisa A. Ruthig
المصدر: Genome Research. 5:225-232
مصطلحات موضوعية: Yeast artificial chromosome, Molecular Sequence Data, Restriction Mapping, Human artificial chromosome, Molecular cloning, Biology, Polymerase Chain Reaction, Restriction map, Genetics, Chromosomes, Human, Humans, Cloning, Molecular, Chromosomes, Artificial, Yeast, In Situ Hybridization, Fluorescence, Genetics (clinical), Cloning, Chromosomes, Human, Pair 12, Base Sequence, Telomere, Molecular biology, genomic DNA, Restriction enzyme, Chromosomes, Human, Pair 2, Chromosomes, Human, Pair 6, Human genome, Chromosomes, Human, Pair 18, Chromosomes, Human, Pair 8
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::dd76bae58c4b933d056800ab7d0b8a96
https://doi.org/10.1101/gr.5.3.225 -
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المؤلفون: Thelma S. Angeles, Chrysanthe Spais, Jean Husten, Jennifer L. Mason, Mark A. Ator, Mark S. Albom, Sheryl L. Meyer, Eric Prouty
المصدر: Assay and drug development technologies. 10(5)
مصطلحات موضوعية: Drug discovery, Kinase, Chemistry, Surface Plasmon Resonance, Staurosporine, Small molecule, Receptor–ligand kinetics, Focal adhesion, Biochemistry, Focal Adhesion Kinase 1, Drug Discovery, Molecular Medicine, Humans, Kinase binding, Surface plasmon resonance, Protein Kinase Inhibitors, Alexa Fluor, Protein Binding
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::fe8aa4196266a6e01a1fc657448f18aa
https://pubmed.ncbi.nlm.nih.gov/22690705 -
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المؤلفون: Dmitri Negorev, Roberto A. Macina, Lisa A. Ruthig, X.-L. Hu, Harold Riethman, Chrysanthe Spais
المصدر: Genomics. 22:569-578
مصطلحات موضوعية: Yeast artificial chromosome, Genetic Linkage, Molecular Sequence Data, P1-derived artificial chromosome, Molecular cloning, Biology, Polymerase Chain Reaction, DNA sequencing, Mice, Restriction map, Species Specificity, Gene mapping, Sequence Homology, Nucleic Acid, Genetics, Animals, Humans, Cloning, Molecular, Chromosomes, Artificial, Yeast, In Situ Hybridization, Fluorescence, DNA Primers, Repetitive Sequences, Nucleic Acid, Base Sequence, Nucleic acid sequence, Chromosome Mapping, DNA, Telomere, Molecular biology, Restriction enzyme, Oligodeoxyribonucleotides, Chromosomes, Human, Pair 1
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المؤلفون: X.-L. Hu, Lisa A. Ruthig, Dmitri Negorev, Chrysanthe Spais, Harold Riethman, Roberto A. Macina
المصدر: Human Molecular Genetics. 3:1847-1853
مصطلحات موضوعية: Molecular Sequence Data, Restriction Mapping, Biology, Polymerase Chain Reaction, chemistry.chemical_compound, Restriction map, Gene duplication, Genetics, Humans, Chromosomes, Artificial, Yeast, Molecular Biology, In Situ Hybridization, Fluorescence, Genetics (clinical), DNA Primers, Repetitive Sequences, Nucleic Acid, Base Sequence, Chromosome Mapping, Chromosome, General Medicine, Telomere, Subtelomere, Molecular biology, Chromosome Banding, Restriction enzyme, genomic DNA, chemistry, Chromosomes, Human, Pair 2, DNA
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::966c05a337cecd08e3090face460b78a
https://doi.org/10.1093/hmg/3.10.1847 -
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المؤلفون: Rabindranath, Tripathy, Robert J, McHugh, Edward R, Bacon, Joseph M, Salvino, George C, Morton, Lisa D, Aimone, Zeck, Huang, Joanne R, Mathiasen, Amy, DiCamillo, Mark J, Huffman, Beth A, McKenna, Karla, Kopec, Lily D, Lu, Jie, Qian, Thelma S, Angeles, Thomas, Connors, Chrysanthe, Spais, Beverly, Holskin, Emir, Duzic, Hervé, Schaffhauser, Gerard C, Rossé
المصدر: Bioorganicmedicinal chemistry letters. 22(3)
مصطلحات موضوعية: Molecular Structure, Brain, Stereoisomerism, Rats, Inhibitory Concentration 50, Mice, Dogs, Receptors, Serotonin, Microsomes, Liver, Animals, Humans, Serotonin Antagonists, Sulfones, Heterocyclic Compounds, 3-Ring
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10
المؤلفون: Babu G, Sundar, Thomas R, Bailey, Derek D, Dunn, Edward R, Bacon, Joseph M, Salvino, George C, Morton, Lisa D, Aimone, Huang, Zeqi, Joanne R, Mathiasen, Amy, Dicamillo, Mark J, Huffman, Beth A, McKenna, Karla, Kopec, Lily D, Lu, Rebecca, Brown, Jie, Qian, Thelma, Angeles, Thomas, Connors, Chrysanthe, Spais, Beverly, Holskin, Deborah, Galinis, Emir, Duzic, Herve, Schaffhauser, Gerard C, Rosse
المصدر: Bioorganicmedicinal chemistry letters. 22(1)
مصطلحات موضوعية: ERG1 Potassium Channel, Brain, Ether-A-Go-Go Potassium Channels, Rats, Inhibitory Concentration 50, Kinetics, Structure-Activity Relationship, Memory, Short-Term, Models, Chemical, Piperidines, Receptors, Serotonin, Schizophrenia, Animals, Humans, Serotonin Antagonists, Benzofurans