-
1
المؤلفون: Kephart Susan Elizabeth, Annette John-Baptiste, Deal Judith G, Danlin Gu, Shubha Bagrodia, Cui Jingrong Jean, Shinji Yamazaki, Djamal Bouzida, Pairish Mason Alan, Evan Smith, Chuangxing Guo, Robert Steven Kania, Dong Liming, Angelica Linton, Indrawan James Mcalpine, Cynthia Louise Palmer
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:7605-7609
مصطلحات موضوعية: Time Factors, Stereochemistry, Metabolite, Clinical Biochemistry, Aminopyridines, Pharmaceutical Science, Electrons, Biochemistry, Dependent drug, chemistry.chemical_compound, Drug Discovery, Humans, Molecular Biology, ADME, Ligand efficiency, Molecular Structure, Mutagenicity Tests, Kinase, Organic Chemistry, Drug interaction, chemistry, Reactive metabolite, Toxicity, Microsomes, Liver, Molecular Medicine, Oxidation-Reduction
-
2
المؤلفون: Jon Engebretsen, Martha A. Ornelas, Kephart Susan Elizabeth, Natilie Hosea, Angelica Linton, Asako Nagata, Javier Gonzalez, Samantha Elizabeth Greasley, Chuangxing Guo, Andrea Fanjul, Pairish Mason Alan, Jeff Elleraas
المصدر: Bioorganic & Medicinal Chemistry Letters. 22:1230-1236
مصطلحات موضوعية: Male, Models, Molecular, Lactams, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, Prostate cancer, chemistry.chemical_compound, Drug Discovery, medicine, Humans, Receptor, Molecular Biology, ADME, Ligand efficiency, Dose-Response Relationship, Drug, Molecular Structure, Drug discovery, Chemistry, Organic Chemistry, Antagonist, Prostatic Neoplasms, Stereoisomerism, medicine.disease, High-Throughput Screening Assays, Androgen receptor, Receptors, Androgen, Lactam, Molecular Medicine
-
3
المؤلفون: Qiyue Hu, Kephart Susan Elizabeth, Angelica Linton, Pairish Mason Alan, Ying Jiang, Chuangxing Guo, Ping Kang, Martha A. Ornelas
المصدر: Journal of Medicinal Chemistry. 54:7705-7712
مصطلحات موضوعية: Models, Molecular, Pyrimidine, Stereochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Protein structure, In vivo, Catalytic Domain, Drug Discovery, Humans, Moiety, Aldehyde oxidase, Drug discovery, Imidazoles, Stereoisomerism, Metabolism, Bridged Bicyclo Compounds, Heterocyclic, Aldehyde Oxidase, Androgen receptor, Pyrimidines, Biochemistry, chemistry, Molecular Medicine, Oxidation-Reduction, Cyclobutanes, Protein Binding
-
4
المؤلفون: Kephart Susan Elizabeth, Angelica Linton, Javier Gonzalez, Kevin D. Bunker, Paul F. Richardson, Chuangxing Guo, Pairish Mason Alan, Martha A. Ornelas, Neal W. Sach
المصدر: Tetrahedron Letters. 52:4760-4763
مصطلحات موضوعية: chemistry.chemical_compound, Chemistry, Organic Chemistry, Drug Discovery, polycyclic compounds, Lactam, Organic chemistry, biochemical phenomena, metabolism, and nutrition, Biochemistry, Reductive amination
-
5
المصدر: Tetrahedron Letters. 52:1692-1696
مصطلحات موضوعية: Reaction conditions, Nucleophilic aromatic substitution, Chemistry, Organic Chemistry, Drug Discovery, Organic chemistry, macromolecular substances, Weakly-reactive, Biochemistry, Combinatorial chemistry
-
6
المؤلفون: Xinjun Hou, Kephart Susan Elizabeth, Dong Liming, Chuangxing Guo
المصدر: Tetrahedron Letters. 51:2909-2913
مصطلحات موضوعية: Solvent, chemistry.chemical_compound, chemistry, Organic Chemistry, Drug Discovery, Organic chemistry, Biochemistry, Linker, Sulfamide, Catalysis
-
7
المؤلفون: Todd VanArsdale, RoseAnn Ferre, David A. Matthews, Ian Popoff, Marakovits Joseph T, Brion W. Murray, Joseph Piraino, Barbara Mroczkowski, Dong Liming, Stephen Margosiak, Xinjun Hou, M. Catherine Johnson, James Arthur Thomson, Gerrit Los, Eleanor Dagostino, Chuangxing Guo, Samantha Elizabeth Greasley, Hans E. Parge
المصدر: Bioorganic & Medicinal Chemistry Letters. 19:5613-5616
مصطلحات موضوعية: Molecular model, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Computational biology, Crystallography, X-Ray, Biochemistry, Structure-Activity Relationship, Drug Discovery, Combinatorial Chemistry Techniques, Humans, Structure–activity relationship, Computer Simulation, Amino Acid Sequence, Enzyme Inhibitors, NIMA-Interacting Peptidylprolyl Isomerase, Molecular Biology, Peptidylprolyl isomerase, Binding Sites, Ligand efficiency, Chemistry, Organic Chemistry, Peptidylprolyl Isomerase, Drug Design, Cis-trans-Isomerases, PIN1, Molecular Medicine
-
8
المؤلفون: Dong Liming, Xinjun Hou, Elizabeth A. Lunney, Corinne E. Augelli-Szafran, Deal Judith G, Christopher F. Bigge, Darin Vanderpool, Raymond Andrew Hudack, Nancy Sue Barta, Bradley William Caprathe, Chuangxing Guo, Steve Bender, Richard E. Showalter, Lorraine Kathleen Fay, Arindam Chatterjee
المصدر: Journal of Medicinal Chemistry. 49:1202-1206
مصطلحات موضوعية: Peptidylprolyl isomerase, Aza Compounds, Binding Sites, Neurite, Chemistry, Hydrogen Bonding, Biological activity, Tacrolimus Binding Protein 1A, Isoquinolines, Ligands, Amides, Heterocyclic Compounds, 4 or More Rings, Tacrolimus, Structure-Activity Relationship, Neuroprotective Agents, FKBP, Biochemistry, Cis-trans-Isomerases, Drug Discovery, Molecular Medicine, Structure–activity relationship, Binding site, Cognitive decline
-
9
المؤلفون: Bo Yang, Ye Sun, Guolan Wei, Youzhi Tong, Chuangliang Xu, Shancheng Ren, Jianguo Hou, Chunyun Chen, Xu Gao, Weidong Xu, Karl Zhou, Ying-Hao Sun, Chuangxing Guo, Tie Zhou
المصدر: Journal of Clinical Oncology. 35:e16511-e16511
مصطلحات موضوعية: Androgen receptor, Cancer Research, Oncology, business.industry, Antagonist, Cancer research, Medicine, In patient, Proxalutamide, First in human, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::a267146e7479c07e0169308f8a48b99a
https://doi.org/10.1200/jco.2017.35.15_suppl.e16511 -
10
المؤلفون: Li Haitao, Paderes Genevieve Deguzman, Brion W. Murray, Xinjun Hou, RoseAnn Ferre, Marakovits Joseph T, M. Catherine Johnson, Paul S. Humphries, Samantha Elizabeth Greasley, Eugenia Kraynov, Joseph Piraino, Dong Liming, Eleanor Dagostino, Chuangxing Guo
المصدر: Bioorganicmedicinal chemistry letters. 24(17)
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Carboxylic Acids, Pharmaceutical Science, Proline binding, Biochemistry, Epitope, Phosphates, chemistry.chemical_compound, Structure-Activity Relationship, Catalytic Domain, Drug Discovery, Humans, Carboxylate, Enzyme Inhibitors, Molecular Biology, Cell permeability, biology, Dose-Response Relationship, Drug, Molecular Structure, Organic Chemistry, Active site, Peptidylprolyl Isomerase, Phosphate, NIMA-Interacting Peptidylprolyl Isomerase, chemistry, biology.protein, PIN1, Molecular Medicine, Structure based, Benzimidazoles