-
1
المؤلفون: Amy E. M. Newman, Neil J. MacLusky, Hayley A. Wilson, Elena Choleris, Colin Howes, Cameron S. Wasson, Emily Martin
المصدر: Brain research. 1729
مصطلحات موضوعية: 0301 basic medicine, Litter (animal), Testosterone propionate, Male, Hypothalamo-Hypophyseal System, Gonad, Offspring, Physiology, Pituitary-Adrenal System, 03 medical and health sciences, chemistry.chemical_compound, Basal (phylogenetics), Mice, 0302 clinical medicine, Corticosterone, Pregnancy, Medicine, Juvenile, Animals, Testosterone, Molecular Biology, Sex Characteristics, business.industry, General Neuroscience, Testosterone (patch), 030104 developmental biology, medicine.anatomical_structure, chemistry, Prenatal Exposure Delayed Effects, Female, Neurology (clinical), business, 030217 neurology & neurosurgery, Stress, Psychological, Developmental Biology
-
2
المؤلفون: Nathalie Cassoux, Rania El Botty, Joanne Wilson, Emma J. Davies, Béré Diallo, Gérald Massonnet, Colin Howes, Adnan Naguez, Chloé Raymondie, Aaron Smith, Sophie Piperno-Neumann, Sergio Roman-Roman, Paul D. Smith, Fariba Nemati, Justine Fleury, Didier Decaudin
المصدر: Oncotarget
مصطلحات موضوعية: 0301 basic medicine, MAPK/ERK pathway, medicine.medical_treatment, 03 medical and health sciences, 0302 clinical medicine, pharmacodynamics, medicine, selumetinib, Chemotherapy, GNA11, business.industry, MEK inhibitor, Melanoma, medicine.disease, targeted therapies, 030104 developmental biology, Oncology, Docetaxel, 030220 oncology & carcinogenesis, Selumetinib, Cancer research, uveal melanoma, patient-derived xenografts, business, GNAQ, Research Paper, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::88f4a0d59115d955bb836fcd38a72b86
https://doi.org/10.18632/oncotarget.24670 -
3
المؤلفون: Karen So, Christine Pattison, Stuart Mair, Mark Savage, Gabriella Mariani, Angela W. Dymond, Gill Ford, Colin Howes, Paul D. Martin
المصدر: Clinical therapeutics. 38(11)
مصطلحات موضوعية: Male, Metabolite, Glucuronidation, Phases of clinical research, Administration, Oral, Urine, Pharmacology, 030226 pharmacology & pharmacy, Excretion, 03 medical and health sciences, chemistry.chemical_compound, Feces, 0302 clinical medicine, Pharmacokinetics, Medicine, Humans, Pharmacology (medical), Carbon Radioisotopes, selumetinib, business.industry, Middle Aged, Tolerability, chemistry, 030220 oncology & carcinogenesis, Selumetinib, excretion, Benzimidazoles, business, metabolism, pharmacokinetics
-
4
المؤلفون: Marine Dubois, Béré Diallo, Didier Decaudin, Aaron Smith, Emma J. Davies, Rania El Botty, Pascale Mariani, Sophie Piperno-Neumann, Colin Howes, Justine Fleury, Fariba Nemati, Paul D. Smith, Adnan Naguez, Nathalie Cassoux, Sergio Roman Roman, Gérald Massonnet, Joanne Wilson
المصدر: Cancer Research. 78:5782-5782
مصطلحات موضوعية: Oncology, Cancer Research, medicine.medical_specialty, Melanoma patient, business.industry, Internal medicine, medicine, Selumetinib, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::e193cc1c2e9904e74ef279bb521a9b81
https://doi.org/10.1158/1538-7445.am2018-5782 -
5
المؤلفون: Robin Alec Fairhurst, Joseph D. Fullerton, David Andrew Sandham, Heinz E. Moser, Mauro Zurini, Sandra Haberthuer, Darryl Brynley Jones, Mark Dodds, Julia Hatto, Gurdip Bhalay, Colin Howes, Paul Nicklin, Simon J. Watson, David Farr, Reto Naef, Irene Muller, Andrew Dunstan, Nichola J. Arnold, Nicholas James Devereux, Morris Tweed, Angela Glen, Katharine L. Turner, Beate Leuenberger, David Beer, Sylvie Gomez, Ruth Arnold, Thomas H. Keller, Stephen Paul Collingwood, Sarah Craig
المصدر: Bioorganic & Medicinal Chemistry Letters. 17:2376-2379
مصطلحات موضوعية: Male, Clinical Biochemistry, Biological Availability, Pharmaceutical Science, Biochemistry, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Erectile Dysfunction, 3',5'-Cyclic-GMP Phosphodiesterases, In vivo, Drug Discovery, Animals, Humans, Protein Isoforms, Structure–activity relationship, Pharmacokinetics, Enzyme Inhibitors, Molecular Biology, Cyclic Nucleotide Phosphodiesterases, Type 5, chemistry.chemical_classification, Organic Chemistry, Biological activity, Xanthine, In vitro, Bioavailability, Enzyme, chemistry, Xanthines, cGMP-specific phosphodiesterase type 5, Molecular Medicine, Cattle, sense organs
-
6
المؤلفون: I Williams, Lazzaro Mazzoni, John R. Fozard, Colin Howes, Jason P. Hannon, Cedric Wolber, Bruno Tigani
المصدر: British Journal of Pharmacology. 135:685-696
مصطلحات موضوعية: Pharmacology, medicine.medical_specialty, medicine.drug_class, business.industry, respiratory system, Adenosine A3 receptor, Receptor antagonist, Adenosine receptor, Adenosine, Adenosine A1 receptor, chemistry.chemical_compound, Endocrinology, chemistry, Internal medicine, CGS-15943, medicine, Receptor, business, medicine.drug, CGS-21680
-
7
المؤلفون: Matthew Ling, Paula Taylor, Keith Parry, Doug Ferguson, Alexander MacDonald, Sean Redmond, Howard A. Burris, Simon T. Barry, Colin Howes, Simon Smith, Young-Ho Song, Elizabeth Janet Pease, A. Hughes, Wolfram Brugger, Maureen Hattersley, Nicholas Floch, Kim Maratea, James Martin Nolan, Susan Ashton, Shenghua Wen
المصدر: Cancer Research. 77:311-311
مصطلحات موضوعية: 0301 basic medicine, Oncology, Drug, Cancer Research, medicine.medical_specialty, business.industry, media_common.quotation_subject, Phases of clinical research, Cancer, Neutropenia, Prodrug, medicine.disease, 03 medical and health sciences, 030104 developmental biology, Therapeutic index, Internal medicine, Drug delivery, Immunology, Medicine, Aurora Kinase B, business, media_common
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::a1edd7c1c41f6f37bee81bb4978e5ef2
https://doi.org/10.1158/1538-7445.am2017-311 -
8
المؤلفون: Sergio Roman-Roman, R. El-Botty, Didier Decaudin, Fariba Nemati, Chloé Raymondie, Aaron Smith, Paul D. Smith, Béré Diallo, Emma J. Davies, Colin Howes, Joanne Wilson, Gérald Massonnet
المصدر: European Journal of Cancer. 69:S132
مصطلحات موضوعية: Oncology, Cancer Research, medicine.medical_specialty, business.industry, medicine.medical_treatment, Melanoma, medicine.disease, Targeted therapy, Internal medicine, medicine, Selumetinib, In patient, business, Adjuvant
-
9
المؤلفون: Simon T. Barry, Richard J. A. Goodwin, John G. Swales, Philip J. Jewsbury, Zoltan Takats, Nicola Strittmatter, Anna Nilsson, Colin Howes, Per E. Andrén, Susan Ashton, Paula Taylor
المصدر: Cancer Research. 75:3678-3678
مصطلحات موضوعية: Cancer Research, Oncology, Chemistry, Cancer research, Nanoparticle
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::6f8cdf22e38038cb10a296460a54c08e
https://doi.org/10.1158/1538-7445.am2015-3678 -
10
المؤلفون: John R. Fozard, Thomas H. Keller, Robin Alec Fairhurst, Alan Steward, Bernard Faller, David Bentley, Ian N. Bruce, David A. Sykes, David Beattie, John Reilly, Zhengjin Jiang, Joe Fullerton, David Beer, Christine Lewis, Frederique Loeuillet-Ritzler, Claire Hayden, Heinz E. Moser, Alexandre Trifilieff, Bernard Cuenoud, Steven J. Charlton, Lauren M. Tedaldi, Colin Howes, Elke Wissler, François Baur, Simon J. Watson, Morris Tweed, Julia Hatto, Sheila Garman, Roland Ernst, Handan He, Diana Janus, Daniel Wyss, Michelle Bradley, David Farr
المصدر: Journal of medicinal chemistry. 53(9)
مصطلحات موضوعية: Intrinsic activity, Chemistry, Guinea Pigs, Pharmacology, Quinolones, Bronchodilator Agents, Structure-Activity Relationship, Therapeutic index, In vivo, Drug Discovery, Lipophilicity, Administration, Inhalation, Indans, medicine, Molecular Medicine, Potency, Indacaterol, Structure–activity relationship, Animals, Humans, Receptor, Adrenergic beta-2 Receptor Agonists, Hydrophobic and Hydrophilic Interactions, medicine.drug