-
1
المؤلفون: Allyn T. Londregan, John M. Curto, Emma Hastry, Colin R. Rose, Simon Berritt
المصدر: The Journal of Organic Chemistry. 88:5671-5675
مصطلحات موضوعية: Organic Chemistry
-
2
المؤلفون: John C. Murray, Colin R. Rose, John M. Curto
المصدر: The Journal of Organic Chemistry. 88:3340-3345
مصطلحات موضوعية: Organic Chemistry
-
3
المؤلفون: Daniel W. Widlicka, Nathan E. Genung, Jana Polivkova, Daniel W. Kung, Wiglesworth Kristin, Thomas Andrew Brandt, Jun Xiao, Matthew S. Dowling, Yingxin Zhang, Paul M. Herrinton, David J. Edmonds, Todd Zahn, Ka Ning Yip, Colin R. Rose, Qifang Li, Jane Panteleev, Shawn Cabral, Andre Shavnya, Nandell F. Keene, John D. Weaver, Benjamin A. Thuma, Michael Herr, Ian Edmonds, Gary Erik Aspnes, Guoqiang Wang, Philip D. Dent, Dilinie P. Fernando, Aaron C. Smith, Michael G. Vetelino, Sophie Y. Lavergne, Edward L. Conn
المصدر: Organic Process Research & Development. 22:681-696
مصطلحات موضوعية: Indole test, 010405 organic chemistry, Chemistry, Organic Chemistry, AMPK, Investigational New Drug, Pharmacology, 010402 general chemistry, medicine.disease, 01 natural sciences, 0104 chemical sciences, Diabetic nephropathy, medicine, Physical and Theoretical Chemistry, Protein kinase A
-
4
المؤلفون: Jianmin Sun, Thomas Ryckmans, David Fengas, Colin R. Rose, M. Scott Johnson, Matthew Corbett, David James Rawson, Nigel Alan Swain, Joseph S. Warmus, Lyn H. Jones, Brian E. Marron, Aristos J. Alexandrou, David Printzenhoff, C. Elizabeth Payne, Bruce M. Bechle, Rubben Torella, Neil A. Castle, Jonathan W. Theile, Elaine Tseng, David C. Blakemore, Andrew Pike, R. Ian Storer, Neil J. Flanagan, Alan Daniel Brown
المصدر: Bioorganic & Medicinal Chemistry Letters. 27:4805-4811
مصطلحات موضوعية: 0301 basic medicine, Voltage-gated ion channel, Chemistry, Sodium channel, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, In vivo, Drug Discovery, NAV1, Molecular Medicine, Potency, Molecular Biology, 030217 neurology & neurosurgery, Ion channel, Conjugate, ADME
-
5
المؤلفون: Bruce M. Bechle, Joseph S. Warmus, Jianmin Sun, David C. Blakemore, Chunhui Dai, Chan Woo Huh, Julien Genovino, Colin R. Rose, Matthew Corbett
المصدر: Organic Letters. 19:1064-1067
مصطلحات موضوعية: Carbamate, Olefin fiber, Nitrile, 010405 organic chemistry, Chemistry, medicine.medical_treatment, Organic Chemistry, One-pot synthesis, 010402 general chemistry, 01 natural sciences, Biochemistry, Chemical synthesis, 0104 chemical sciences, chemistry.chemical_compound, Furan, Reagent, medicine, Organic chemistry, Amine gas treating, Physical and Theoretical Chemistry
-
6
المؤلفون: Colin R. Rose, Elisabeth Mortimer-Cassen, Juha Kammonen, Rebecca L. Fish, David C. Pryde, Lishuang Cao, Sarah A. Nickolls, Neil J. Flanagan, Karl Richard Gibson, Joseph S. Warmus, Christine Anne Louise Watson, Chan Woo Huh, David J. Reynolds, Rachel Gurrell, Kiyoyuki Omoto, Andrew Pike, Clara Stead, David C. Blakemore, Rosemarie Roeloffs, Dafydd R. Owen, Mifune Takeuchi, Robert M. Owen
المصدر: Journal of Medicinal Chemistry.
مصطلحات موضوعية: 0303 health sciences, Allosteric modulator, Safety studies, Chemistry, GABAA receptor, Allosteric regulation, Computational biology, Subtype selective, 01 natural sciences, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, Identification (information), Drug Discovery, Functional selectivity, Molecular Medicine, Functional activity, 030304 developmental biology
-
7
المؤلفون: Jane M. Withka, Daniel W. Kung, Russell A. Miller, Matthew S. Dowling, Aaron C. Smith, Angela Wolford, Heather Eng, Janice A. Brown, Jun Xiao, Kris A. Borzilleri, Ravi G. Kurumbail, David J. Edmonds, Jessica Ward, Amit S. Kalgutkar, Colin R. Rose, Tim F. Ryder, Meihua Tu, Dilinie P. Fernando, Emily Cokorinos, David Hepworth, James A. Landro, Kimberly O. Cameron, Matthew F. Calabrese, Christopher T. Salatto, Francis Rajamohan, Andre Shavnya, Markus Boehm, Yuxia Mao, Allan R. Reyes, Richard K. Frisbie, Nicole Caspers, Edward L. Conn, Samit Kumar Bhattacharya
المصدر: Journal of Medicinal Chemistry. 59:8068-8081
مصطلحات موضوعية: Male, Models, Molecular, 0301 basic medicine, Adenosine monophosphate, Indazoles, Indoles, Protein Conformation, Administration, Oral, Enzyme Activators, AMP-Activated Protein Kinases, Crystallography, X-Ray, 03 medical and health sciences, chemistry.chemical_compound, Dogs, 0302 clinical medicine, AMP-activated protein kinase, Drug Discovery, medicine, Animals, Humans, Diabetic Nephropathies, Protein kinase A, Indole test, Indazole, biology, Activator (genetics), Chemistry, AMPK, Adenosine, High-Throughput Screening Assays, Rats, Macaca fascicularis, 030104 developmental biology, Biochemistry, 030220 oncology & carcinogenesis, Injections, Intravenous, biology.protein, Molecular Medicine, Adsorption, medicine.drug
-
8
المؤلفون: Daniel W. Kung, James A. Southers, Shawn Cabral, Carmen N. Garcia-Irizarry, Aaron C. Smith, Colin R. Rose, Scott W. Bagley, David A. Griffith, David B. Damon
المصدر: The Journal of Organic Chemistry. 81:3509-3519
مصطلحات موضوعية: Nitrile, 010405 organic chemistry, Organic Chemistry, Azetidine, Alkylation, 010402 general chemistry, Ring (chemistry), 01 natural sciences, Reductive amination, Pyrrolidine, 0104 chemical sciences, chemistry.chemical_compound, chemistry, Organic chemistry, Piperidine, Enantiomer
-
9
المؤلفون: R. Ian Storer, James A. Clulow, Joseph S. Warmus, Jianmin Sun, Victoria E. Albrow, Colin R. Rose, Rachel L. Grimley, Lyn H. Jones, Edward W. Tate
المصدر: Mol. BioSyst.. 12:1781-1789
مصطلحات موضوعية: Proteomics, 0301 basic medicine, Cell Membrane Permeability, Proteome, Histone Deacetylases, Mass Spectrometry, 03 medical and health sciences, Drug Discovery, Humans, Molecular Biology, Regulation of gene expression, Molecular Structure, Staining and Labeling, biology, Acetylation, Recombinant Proteins, Chromatin, Enzyme Activation, Histone Deacetylase Inhibitors, 030104 developmental biology, Histone, Tubulin, Biochemistry, Molecular Probes, biology.protein, Histone deacetylase, Bioorthogonal chemistry, Biotechnology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1a3c2c61f48d910356fe2d6f9c9d2a69
https://doi.org/10.1039/c6mb00109b -
10
المؤلفون: Colin R. Rose, Dilinie P. Fernando, James Saenz, Kimberly Lapham, Suvi T. M. Orr, Paula M. Loria, Maria von Volkenburg, Beveridge Ramsay, Samit Kumar Bhattacharya, Kimberly O. Cameron, Margaret V. Jackson, Steven B. Coffey, Jun Xiao, Gregory Storer, Vishal Khot, Jigna D. Patel, Ingrid A. Stock, Yingxin Zhang, Kim F. McClure, Derek Vrieze, David Hepworth, Guoqiang Wang, Rachel E. Kosa
المصدر: ACS Medicinal Chemistry Letters. 6:156-161
مصطلحات موضوعية: Chemistry, medicine.drug_class, Aryl, Organic Chemistry, Growth hormone secretagogue receptor, Carboxamide, Biochemistry, Combinatorial chemistry, Safety profile, chemistry.chemical_compound, Drug Discovery, medicine, Inverse agonist, Ghrelin, Chemical stability, Piperidine