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1
المؤلفون: R A, Daines, P A, Chambers, D S, Eggleston, J J, Foley, D E, Griswold, R C, Haltiwanger, D R, Jakas, W D, Kingsbury, L D, Martin, I, Pendrak
المصدر: Journal of Medicinal Chemistry. 37:3327-3336
مصطلحات موضوعية: Neutrophils, Pyridines, medicine.drug_class, Stereochemistry, Carboxylic acid, Receptors, Leukotriene B4, Thio, Crystallography, X-Ray, Cytoplasmic Granules, Benzoates, Binding, Competitive, Leukotriene B4, Sulfone, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Humans, Benzoic acid, chemistry.chemical_classification, Molecular Structure, Chemistry, Sulfoxide, Biological activity, respiratory system, Receptor antagonist, Molecular Medicine, Calcium, lipids (amino acids, peptides, and proteins), Receptor antagonist activity
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2
المؤلفون: S. M. Hech, Francis L. McCabe, Jeffrey C. Boehm, M. J. Caranfa, K. G. Holden, Randall K. Johnson, William D. Kingsbury, G. Gallagher, Leo F. Faucette, D. R. Jakas, R. P. Hertzberg
المصدر: ChemInform. 22
مصطلحات موضوعية: Antitumor activity, Water soluble, Biochemistry, biology, Chemistry, Topoisomerase, medicine, biology.protein, General Medicine, Camptothecin, medicine.drug
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3
المؤلفون: K W, Ward, L M, Azzarano, W E, Bondinell, R D, Cousins, W F, Huffman, D R, Jakas, R M, Keenan, T W, Ku, D, Lundberg, W H, Miller, J A, Mumaw, K A, Newlander, J L, Pirhalla, T J, Roethke, K L, Salyers, P R, Souder, G J, Stelman, B R, Smith
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 27(11)
مصطلحات موضوعية: Male, Rats, Sprague-Dawley, Macaca fascicularis, Mice, Dogs, Species Specificity, Aminopyridines, Animals, Receptors, Vitronectin, Acetates, Chromatography, High Pressure Liquid, Mass Spectrometry, Rats
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::e030481b63061d6287d5df04c74a5102
https://pubmed.ncbi.nlm.nih.gov/10534306 -
4
المؤلفون: N. M. Hall, D. R. Jakas, A. W. Chow, B. P. Trotter, J. R. E. Hoover
المصدر: Journal of Heterocyclic Chemistry. 10:71-75
مصطلحات موضوعية: chemistry.chemical_classification, chemistry, 2-aminobenzimidazole, Carboxylic acid, Organic Chemistry, Organic chemistry
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5
المؤلفون: J. R. E. Hoover, G. L. Dunn, D. R. Jakas, L. L. Lam, J. J. Taggart, J. R. Guarini, L. Phillips
المصدر: Journal of medicinal chemistry. 17(1)
مصطلحات موضوعية: Magnetic Resonance Spectroscopy, Bacteria, Stereoisomerism, Microbial Sensitivity Tests, Staphylococcal Infections, Amides, Cephalosporins, Klebsiella Infections, Mice, Structure-Activity Relationship, Dogs, Drug Discovery, Molecular Medicine, Animals, Mandelic Acids, Rabbits, Escherichia coli Infections
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6
المؤلفون: D. R. Jakas, L. Phillips, J. R. Guarini, L. L. Lam, G. L. Dunn, John J. Taggart, John R. E. Hoover
المصدر: Chemischer Informationsdienst. 5
مصطلحات موضوعية: Cephem, medicine.drug_class, Chemistry, Stereochemistry, Cephalosporin, medicine, General Medicine
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7
المؤلفون: D. R. Jakas, Donald Pitkin, Lillian Phillips, Paul Actor, Sarah F. Grappel, George L. Dunn
المصدر: Antimicrobial agents and chemotherapy. 25(6)
مصطلحات موضوعية: Male, Cefotaxime, medicine.drug_class, Cephalosporin, Biology, medicine.disease_cause, Microbiology, Cefmenoxime, Minimum inhibitory concentration, Mice, Ceftizoxime, medicine, Animals, Pharmacology (medical), Saimiri, Antibacterial agent, Pharmacology, Bacteria, Rats, Inbred Strains, Bacterial Infections, Blood Proteins, Cephalosporins, Rats, Kinetics, Infectious Diseases, Staphylococcus aureus, Moxalactam, medicine.drug, Protein Binding, Research Article
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1ac9c88e1f5d80c945a84df2238020ef
https://pubmed.ncbi.nlm.nih.gov/6742815 -
8
المؤلفون: D. R. Jakas, Jerry A. Weisbach, L.D. Davis, George L. Dunn, Joseph V. Uri, John R. E. Hoover, Paul Actor, E.M. Dietz, David A. Berges, John J. Taggart, N. Yim
المصدر: The Journal of antibiotics. 29(1)
مصطلحات موضوعية: Male, Time Factors, Chemical Phenomena, medicine.drug_class, Cephalosporin, Pharmacology, Hydroxylation, chemistry.chemical_compound, Mice, Structure-Activity Relationship, In vivo, Oral administration, Drug Discovery, medicine, Animals, Escherichia coli Infections, Cephaloglycin, Bacteria, Chemistry, Cefatrizine, In vitro, Cephalosporins, Antibacterial activity, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d1a57b79096b705dab3872ba4d73b293
https://pubmed.ncbi.nlm.nih.gov/776915 -
9ChemInform Abstract: HERST. EINIGER TRIMETHYLPENTACYCLO(5,4,0,0(2,6)0(3,10)0(5,9))UNDECAN-8,11-DIONE
المؤلفون: D. R. Jakas, A. W. Chow, J. R. Hoover
المصدر: Chemischer Informationsdienst. 3
مصطلحات موضوعية: Chemistry, General Medicine, Medicinal chemistry
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10
المؤلفون: B. P. Trotter, N. M. Hall, J. R. E. Hoover, D. R. Jakas, A. W. Chow
المصدر: Chemischer Informationsdienst. 4
مصطلحات موضوعية: Chemistry, Stereochemistry, General Medicine