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1
المؤلفون: Gary E. Zurenko, Betty H. Yagi, Douglas K Hutchinson, D E Emmert, David R. Graber, Jackson B. Hester, Stuart A. Garmon, Judith C. Hamel, Michael R Barbachyn, Ronda D. Schaadt, Michael J. Genin, Douglas Stapert, Joel Morris, David J. Anderson, Debra A. Allwine, R J Reischer, Charles W. Ford, Kevin C. Grega
المصدر: Journal of Medicinal Chemistry. 43:953-970
مصطلحات موضوعية: Azoles, Stereochemistry, Triazole, Administration, Oral, Microbial Sensitivity Tests, Pyrazole, medicine.disease_cause, Haemophilus influenzae, Mice, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, medicine, Eperezolid, Animals, Humans, Organic chemistry, Oxazoles, Moraxella, Antibacterial agent, chemistry.chemical_classification, biology, biology.organism_classification, Anti-Bacterial Agents, chemistry, Molecular Medicine, Azole, Methicillin Resistance, Antibacterial activity, Moraxella catarrhalis
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2
المؤلفون: Charles W. Ford, Gary E. Zurenko, Hutchinson Douglas K, Betty H. Yagi, Janice M. Friis, D E Emmert, Michael J. Genin, Shobe Em, Jackson B. Hester, Stuart A. Garmon, Debra A. Allwine, Wade J. Adams, Ronda D. Schaadt, Judith C. Hamel, Douglas Stapert
المصدر: Journal of Medicinal Chemistry. 41:5144-5147
مصطلحات موضوعية: Male, Fastidious organism, Gram-negative bacteria, Colony Count, Microbial, Administration, Oral, medicine.disease_cause, Haemophilus influenzae, Microbiology, Rats, Sprague-Dawley, Moraxella catarrhalis, Inhibitory Concentration 50, Mice, Structure-Activity Relationship, Drug Discovery, medicine, Animals, Pyrroles, Oxazoles, Moraxella, Antibacterial agent, biology, Chemistry, Staphylococcal Infections, biology.organism_classification, Anti-Bacterial Agents, Rats, Injections, Intravenous, Pyrazoles, Molecular Medicine, Antibacterial activity, Bacteria
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3
المؤلفون: W. J. Howe, W. T. Lowther, J. O. Hui, W. G. Tarpley, D. E. Emmert, Chetana Rao, A G Tomasselli, John H. Kinner, V. S. Bradford, D. L. Alexander, Tomi K. Sawyer, B.M. Dunna, Robert A. Conradi, D. L. Decamp, Clark W. Smith, Allen W. Harrison, Charles S. Craik, James Michael Tustin, T. J. Mcquade, Robert L. Heinrikson, Y. Z. Zhang, Philip S. Burton, Jed F. Fisher, Roger A. Poorman, Joseph B. Moon, Jackson B. Hester, D J Staples, L. Liu, P. E. Scarborough, Maggiora Linda Louise
المصدر: Bioorganic & Medicinal Chemistry Letters. 3:819-824
مصطلحات موضوعية: Cathepsin, Protease, Dipeptide, biology, Isostere, Peptidomimetic, Chemistry, medicine.medical_treatment, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Pharmacology, Biochemistry, Enzyme binding, chemistry.chemical_compound, Pepsin, Drug Discovery, medicine, biology.protein, Molecular Medicine, Pharmacophore, Molecular Biology
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المؤلفون: W. J. Howe, W. T. Lowther, A G Tomasselli, D. E. Emmert, D J Staples, Jackson B. Hester, W. G. Tarpley, J. O. Hui, Ben M. Dunn, John H. Kinner, Robert L. Heinrikson, Y. Z. Zhang, Tomi K. Sawyer, Charles S. Craik, D. L. Decamp, James Michael Tustin, T. J. Mcquade, D. L. Alexander, Allen W. Harrison, P. E. Scarborough, Robert A. Conradi, Jed F. Fisher, Roger A. Poorman, Philip S. Burton, Maggiora Linda Louise, V. S. Bradford, Joseph B. Moon, L. Liu, Clark W. Smith, Chetana Rao
المصدر: ChemInform. 26
مصطلحات موضوعية: Enzyme binding, Protease, Chemistry, Peptidomimetic, medicine.medical_treatment, Human immunodeficiency virus (HIV), medicine, General Medicine, Selectivity, medicine.disease_cause, Cell permeability, Virology
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المؤلفون: J. K. Gibson, Jackson B. Hester, M. G. Cimini, B. E. West, Louis L. Skaletzky, P. K. Locker, J. K. Sykes, D. E. Emmert, S. C. Perricone
المصدر: Journal of medicinal chemistry. 34(1)
مصطلحات موضوعية: Male, Magnetic Resonance Spectroscopy, Tertiary amine, Refractory period, Heart Ventricles, Myocardial Infarction, Pharmacology, In Vitro Techniques, Structure-Activity Relationship, Dogs, Drug Discovery, medicine, Animals, Ventricular Function, Papillary muscle, Sulfonamides, Molecular Structure, Cardiac electrophysiology, Chemistry, Ibutilide Fumarate, Sotalol, Effective refractory period, Biological activity, Arrhythmias, Cardiac, Heart, Myocardial Contraction, medicine.anatomical_structure, Biochemistry, cardiovascular system, Molecular Medicine, Female, Indicators and Reagents, Rabbits, Anti-Arrhythmia Agents, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::a9f50c9f1fc13dcdb9c3d033633809b4
https://pubmed.ncbi.nlm.nih.gov/1992131 -
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المؤلفون: M. I. Dietrick, D. E. Emmert
المصدر: Rubber Chemistry and Technology. 50:217-223
مصطلحات موضوعية: Standard sample, Materials science, Polymers and Plastics, Test procedures, law, Sample (material), Materials Chemistry, Vulcanization, Forensic engineering, Adhesion, Composite material, law.invention, Tensile testing
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::988afaac8e5ad2736eaf5cf7b40d11e6
https://doi.org/10.5254/1.3535128 -
7
المؤلفون: M. I. Dietrick, D. E. Emmert, D. A. Lederer
المصدر: Journal of Elastomers & Plastics. 9:77-93
مصطلحات موضوعية: Cure rate, Materials science, Polymers and Plastics, Materials Chemistry, Adhesion, Composite material
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::e5cab922a9d75a818195a0f39fc459de
https://doi.org/10.1177/009524437700900105 -
8
المؤلفون: J. H. Ludens, D. E. Emmert, B. E. West, Jackson B. Hester
المصدر: Journal of Medicinal Chemistry. 32:1157-1163
مصطلحات موضوعية: Male, Chemical Phenomena, Stereochemistry, medicine.medical_treatment, Substituent, Natriuresis, Kidney, Benzodiazepines, Structure-Activity Relationship, chemistry.chemical_compound, Dogs, Chlorides, Oral administration, Drug Discovery, Side chain, medicine, Animals, heterocyclic compounds, Dose-Response Relationship, Drug, Molecular Structure, Chemistry, Aryl, Rats, Inbred Strains, Triazoles, Diuretic Activity, Diuresis, Rats, Potassium, Molecular Medicine, Diuretic
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ea89a3f96d5ac7c15abf85414f7b781a
https://doi.org/10.1021/jm00126a003 -
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المؤلفون: Daniel Lednicer, D. E. Emmert, C. G. Chidester, D. J. Duchamp
المصدر: The Journal of Organic Chemistry. 36:3260-3266
مصطلحات موضوعية: Structure-Activity Relationship, Crystallography, Estradiol, X-Ray Diffraction, Chemistry, Organic Chemistry, X-ray crystallography, Structure–activity relationship, Total synthesis, Testosterone, Methylation, Norsteroids
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ffa1b8e872a94b2b17538d41e854a68b
https://doi.org/10.1021/jo00821a002 -
10
المؤلفون: D E Emmert, D Lednicer
المصدر: Journal of Medicinal Chemistry. 11:1258-1262
مصطلحات موضوعية: Fertility, Chemistry, Drug Discovery, Methods, Animals, Molecular Medicine, Organic chemistry, Oxazoles, Omega, Sulfur, Oxyphenbutazone, Rats
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4f9a01ca05a1c89899add2c57e6b9ed8
https://doi.org/10.1021/jm00312a608