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1دورية أكاديميةOral Absorption of Middle-to-Large Molecules and Its Improvement, with a Focus on New Modality Drugs
المؤلفون: Daigo Asano, Hideo Takakusa, Daisuke Nakai
المصدر: Pharmaceutics, Vol 16, Iss 1, p 47 (2023)
مصطلحات موضوعية: middle-to-large molecule, absorption enhancer, new modality, Lipinski’s rule of five, cyclic peptide, antisense oligonucleotide, Pharmacy and materia medica, RS1-441
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Kentaro Ito, Hideo Takakusa, Masayo Kakuta, Akira Kanda, Nana Takagi, Hiroyuki Nagase, Nobuaki Watanabe, Daigo Asano, Ryoya Goda, Takeshi Masuda, Akifumi Nakamura, Yoshiyuki Onishi, Toshio Onoda, Makoto Koizumi, Yasuhiro Takeshima, Masafumi Matsuo, Kiyosumi Takaishi
المصدر: Current Issues in Molecular Biology, Vol 43, Iss 3, Pp 1267-1281 (2021)
مصطلحات موضوعية: Duchenne muscular dystrophy, exon skipping, antisense oligonucleotide, dystrophin, 2′-O,4′-C-ethylene-bridged nucleic acid (ENA), renadirsen sodium, Biology (General), QH301-705.5
وصف الملف: electronic resource
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المؤلفون: Daigo Asano, Koichi Nakamura, Yumi Nishiya, Hideyuki Shiozawa, Hideo Takakusa, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Takakazu Hamada, Chizuko Yahara, Nobuaki Watanabe, Kouichi Yoshinari
المصدر: Drug Metabolism and Disposition. 51:67-80
مصطلحات موضوعية: Pharmacology, Pharmaceutical Science
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::b60456efe4bbedd2b0c9bab443faf822
https://doi.org/10.1124/dmd.122.001000 -
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المؤلفون: Narayan Karanjule, Noriyuki Hayashi, Sayaka Suzuki, Toshifumi Tsuda, Eri Tokumaru, Kyosuke Tanaka, Hiroko Kimoto, Yuki Domon, Sakiko Takahashi, Kazufumi Kubota, Yutaka Kitano, Tomihisa Yokoyama, Ryuta Koishi, Chie Fujiwara, Shinichi Inaba, Daigo Asano, Tomoko Sakakura, Kiyoshi Takasuna, Tsuyoshi Shinozuka
المصدر: ACS Medicinal Chemistry Letters.
مصطلحات موضوعية: Organic Chemistry, Drug Discovery, Biochemistry
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5
المؤلفون: Daigo Asano, Syoya Hamaue, Hamim Zahir, Hideyuki Shiozawa, Yumi Nishiya, Takako Kimura, Miho Kazui, Naotoshi Yamamura, Marie Ikeguchi, Takahiro Shibayama, Shin-ichi Inoue, Tsuyoshi Shinozuka, Toshiyuki Watanabe, Chizuko Yahara, Nobuaki Watanabe, Kouichi Yoshinari
المصدر: Drug Metabolism and Disposition. 50:235-242
مصطلحات موضوعية: Pharmacology, Pharmaceutical Science
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::70186cea69d28e89cf0b2a4873bd0d31
https://doi.org/10.1124/dmd.121.000665 -
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المؤلفون: Tsuyoshi Nakamura, Mika Yokoyama, Mayuko Akiu, Takashi Tsuji, Kouki Iida, Ken Sakurai, Yoshitaka Sogawa, Koji Terayama, Tomohiro Honda, Jun Tanaka, Daigo Asano, Anthony B. Pinkerton
المصدر: Chemical and Pharmaceutical Bulletin. 69:1110-1122
مصطلحات موضوعية: Male, Nicotinamide phosphoribosyltransferase, Mice, Obese, Type 2 diabetes, Pharmacology, Nicotinamide adenine dinucleotide, Small Molecule Libraries, Structure-Activity Relationship, chemistry.chemical_compound, Pharmacokinetics, Oral administration, Drug Discovery, medicine, Animals, Humans, Urea, Obesity, Nicotinamide Phosphoribosyltransferase, Nucleotide salvage, Chemistry, Activator (genetics), Body Weight, General Chemistry, General Medicine, NAD, medicine.disease, Diabetes Mellitus, Type 2, Anti-Obesity Agents, NAD+ kinase
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1559d4d089014d0c71e8a23a236697a9
https://doi.org/10.1248/cpb.c21-00700 -
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المؤلفون: Akifumi Nakamura, Akira Kanda, Kiyosumi Takaishi, Nobuaki Watanabe, Hideo Takakusa, Toshio Onoda, Masayo Kakuta, Yasuhiro Takeshima, Hiroyuki Nagase, Daigo Asano, Ito Kentaro, Takeshi Masuda, Yoshiyuki Onishi, Makoto Koizumi, Masafumi Matsuo, Nana Takagi, Ryoya Goda
المصدر: Current Issues in Molecular Biology, Vol 43, Iss 90, Pp 1267-1281 (2021)
Current Issues in Molecular Biology
Volume 43
Issue 3
Pages 90-1281مصطلحات موضوعية: Duchenne muscular dystrophy, antisense oligonucleotide, musculoskeletal diseases, Microbiology (medical), congenital, hereditary, and neonatal diseases and abnormalities, cardiac muscle, QH301-705.5, Nonsense mutation, Microbiology, dystrophin, Exon, medicine, renadirsen sodium, Biology (General), Muscular dystrophy, Molecular Biology, 2′-O,4′-C-ethylene-bridged nucleic acid (ENA), biology, business.industry, Cardiac muscle, Skeletal muscle, General Medicine, medicine.disease, Exon skipping, medicine.anatomical_structure, biology.protein, Cancer research, business, Dystrophin, exon skipping
وصف الملف: application/pdf
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::39145bf396bf8da7e422b375dd43fe94
https://doi.org/10.3390/cimb43030090 -
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المؤلفون: Kouichi Yoshinari, Nobuaki Watanabe, Daigo Asano, Tsuyoshi Shinozuka, Hideyuki Shiozawa, Shinji Murata, Takahiro Shibayama, Shin-ichi Inoue
المصدر: Xenobiotica. 51:1060-1070
مصطلحات موضوعية: Pharmacology, chemistry.chemical_classification, Cytochrome, biology, Health, Toxicology and Mutagenesis, Metabolite, Cytochrome P450, General Medicine, Toxicology, Biochemistry, chemistry.chemical_compound, Enzyme, chemistry, S9 fraction, In vivo, biology.protein, Microsome, Aldehyde oxidase
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9Drug‐Like Properties in Macrocycles above MW 1000: Backbone Rigidity versus Side‐Chain Lipophilicity
المؤلفون: R. Scott Lokey, Victoria G. Klein, Daigo Asano, Quinn Edmondson, Cameron R. Pye, Akihiro Furukawa, Joshua Schwochert, Satoshi Ono, Okimasa Okada, Alexandra C Turmon
المصدر: Angew Chem Int Ed Engl
مصطلحات موضوعية: chemistry.chemical_classification, Macrocyclic Compounds, Molecular Structure, Membrane permeability, 010405 organic chemistry, Peptoid, General Medicine, General Chemistry, 010402 general chemistry, 01 natural sciences, Combinatorial chemistry, Article, Catalysis, Cyclic peptide, Chemical space, 0104 chemical sciences, Molecular Weight, chemistry.chemical_compound, Rigidity (electromagnetism), chemistry, Lipophilicity, Side chain, Peptides, Hydrophobic and Hydrophilic Interactions, ADME
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المؤلفون: Yutaka Kitano, Chie Fujiwara, Sayaka Suzuki, Ryuta Koishi, Tomihisa Yokoyama, Satoshi Shibuya, Daigo Asano, Yuki Domon, Kyosuke Tanaka, Hiroko Kimoto, Akiko Shimizugawa, Tsuyoshi Shinozuka, Kazufumi Kubota, Hiroyuki Kobayashi
المصدر: Chemical and Pharmaceutical Bulletin. 68:653-663
مصطلحات موضوعية: biology, Chemistry, medicine.drug_class, Sodium channel, hERG, Analgesic, Central nervous system, General Chemistry, General Medicine, Pharmacology, Quinolone, medicine.anatomical_structure, Drug Discovery, Neuropathic pain, NAV1, biology.protein, medicine, ED50
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::89845e45af2cb38ea79da89f3f6a10c8
https://doi.org/10.1248/cpb.c20-00126