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المؤلفون: Mari Manuia, Wenshuo Lu, Laura J. Kingsley, Zhiwei Ma, Vicki Zhou, Darbi Witmer, Glen Spraggon, Mu-Yun Gao, Pierre-Yves Michellys, Min Lu, Yong Jia, Matthew McNeill, Sarah Greenblatt, Bender Steven Lee, Andreas Kreusch, Gerald Lelais, Xiaohui He, Victor Nikulin, Mei-Ting Vaillancourt, Christian C. Lee, Jacob R. Haling, John Nelson, Ajay A. Vashisht
المصدر: Journal of Medicinal Chemistry. 64:4857-4869
مصطلحات موضوعية: Drug, 0303 health sciences, Protease, Cancer cell proliferation, media_common.quotation_subject, medicine.medical_treatment, 01 natural sciences, 20s proteasome, In vitro, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, chemistry.chemical_compound, chemistry, Biochemistry, Drug Discovery, medicine, Molecular Medicine, Structure based, Protein folding, Boronic acid, 030304 developmental biology, media_common
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المؤلفون: Laura J, Kingsley, Xiaohui, He, Matthew, McNeill, John, Nelson, Victor, Nikulin, Zhiwei, Ma, Wenshuo, Lu, Vicki W, Zhou, Mari, Manuia, Andreas, Kreusch, Mu-Yun, Gao, Darbi, Witmer, Mei-Ting, Vaillancourt, Min, Lu, Sarah, Greenblatt, Christian, Lee, Ajay, Vashisht, Steven, Bender, Glen, Spraggon, Pierre-Yves, Michellys, Yong, Jia, Jacob R, Haling, Gérald, Lelais
المصدر: Journal of medicinal chemistry. 64(8)
مصطلحات موضوعية: Proteasome Endopeptidase Complex, Binding Sites, Cell Survival, Boronic Acids, Cell Line, Bortezomib, Mitochondrial Proteins, Molecular Docking Simulation, Protein Subunits, Structure-Activity Relationship, ATP-Dependent Proteases, Drug Design, Humans, Protease Inhibitors
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المؤلفون: Ryokichi Koyama, Geza Ambrus-Aikelin, Darbi Witmer, Bi-Ching Sang, Yasunori Fukuda, Hidehisa Iwata, Hideyuki Nakagawa, Masaharu Nakayama, Yusuke Kamada
المصدر: ASSAY and Drug Development Technologies. 16:194-204
مصطلحات موضوعية: Orphan receptor, Sulfonamides, Reporter gene, Hydrocarbons, Fluorinated, Molecular Structure, Chemistry, Cholesterol binding, Drug Evaluation, Preclinical, Nuclear Receptor Subfamily 1, Group F, Member 3, Spodoptera, Pharmacology, Cholesterol, RAR-related orphan receptor gamma, Drug Discovery, Coactivator, Sf9 Cells, Animals, Humans, Th17 Cells, Molecular Medicine, Inverse agonist, lipids (amino acids, peptides, and proteins), Receptor, IC50
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::59d9bc10dbf1390655dbeac60d89a052
https://doi.org/10.1089/adt.2018.852 -
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المؤلفون: Jennifer J. Lentz, Judy Cunnigham, Mark Winland, Darbi Witmer, Vanik Sarkissian, Steven L. Rose
المصدر: The American Journal of Gastroenterology. 95:2586-2586
مصطلحات موضوعية: Hepatology, Gastroenterology