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1دورية أكاديمية
المؤلفون: JP Johnson, Thilo Focken, Kuldip Khakh, Parisa Karimi Tari, Celine Dube, Samuel J Goodchild, Jean-Christophe Andrez, Girish Bankar, David Bogucki, Kristen Burford, Elaine Chang, Sultan Chowdhury, Richard Dean, Gina de Boer, Shannon Decker, Christoph Dehnhardt, Mandy Feng, Wei Gong, Michael Grimwood, Abid Hasan, Angela Hussainkhel, Qi Jia, Stephanie Lee, Jenny Li, Sophia Lin, Andrea Lindgren, Verner Lofstrand, Janette Mezeyova, Rostam Namdari, Karen Nelkenbrecher, Noah Gregory Shuart, Luis Sojo, Shaoyi Sun, Matthew Taron, Matthew Waldbrook, Diana Weeratunge, Steven Wesolowski, Aaron Williams, Michael Wilson, Zhiwei Xie, Rhena Yoo, Clint Young, Alla Zenova, Wei Zhang, Alison J Cutts, Robin P Sherrington, Simon N Pimstone, Raymond Winquist, Charles J Cohen, James R Empfield
المصدر: eLife, Vol 11 (2022)
مصطلحات موضوعية: epilepsy, SCN8A, NBI-921352, anti-seizure medicine, Medicine, Science, Biology (General), QH301-705.5
وصف الملف: electronic resource
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المؤلفون: Sultan Chowdhury, David Bogucki, Rostam Namdari, Girish Bankar, Wei Zhang, James Roy Empfield, Matthew Waldbrook, Stephanie M Lee, Lofstrand Verner Alexander, Karen Nelkenbrecher, Samuel J. Goodchild, Rhena Yoo, Noah G. Shuart, Wesolowski Steven Sigmund, Elaine Chang, Mandy Feng, Clint Young, Christoph Martin Dehnhardt, Jenny Li, Zhiwei Xie, Michael Edward Grimwood, Abid Hasan, Sophia Lin, Kristen Burford, Raymond J. Winquist, Charles J. Cohen, Alla Yurevna Zenova, Simon N. Pimstone, Michael R. Wilson, Parisa Karimi Tari, Kuldip Khakh, Celine Dube, Aaron M. Williams, Robin Sherrington, Luis Sojo, Andrea Lindgren, J. P. Johnson, Thilo Focken, Qi Jia, Jean-Christophe Andrez, Shannon Decker, Matthew Taron, Diana Weeratunge, Richard T. Dean, Janette Mezeyova, Shaoyi Sun, Wei Gong, Angela Hussainkhel, Gina de Boer, Alison Jane Cutts
مصطلحات موضوعية: Phenytoin, Glutamatergic, Lacosamide, Chemistry, Sodium channel, Excitatory postsynaptic potential, medicine, Carbamazepine, Pharmacology, Inhibitory postsynaptic potential, IC50, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::32e2e6674136369f3abcd5070b52e762
https://doi.org/10.1101/2021.08.29.458125 -
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المؤلفون: J P, Johnson, Thilo, Focken, Kuldip, Khakh, Parisa Karimi, Tari, Celine, Dube, Samuel J, Goodchild, Jean-Christophe, Andrez, Girish, Bankar, David, Bogucki, Kristen, Burford, Elaine, Chang, Sultan, Chowdhury, Richard, Dean, Gina, de Boer, Shannon, Decker, Christoph, Dehnhardt, Mandy, Feng, Wei, Gong, Michael, Grimwood, Abid, Hasan, Angela, Hussainkhel, Qi, Jia, Stephanie, Lee, Jenny, Li, Sophia, Lin, Andrea, Lindgren, Verner, Lofstrand, Janette, Mezeyova, Rostam, Namdari, Karen, Nelkenbrecher, Noah Gregory, Shuart, Luis, Sojo, Shaoyi, Sun, Matthew, Taron, Matthew, Waldbrook, Diana, Weeratunge, Steven, Wesolowski, Aaron, Williams, Michael, Wilson, Zhiwei, Xie, Rhena, Yoo, Clint, Young, Alla, Zenova, Wei, Zhang, Alison J, Cutts, Robin P, Sherrington, Simon N, Pimstone, Raymond, Winquist, Charles J, Cohen, James R, Empfield
المصدر: eLife. 11
مصطلحات موضوعية: Neurons, Mice, Epilepsy, NAV1.6 Voltage-Gated Sodium Channel, Gain of Function Mutation, Mutation, Sodium, Animals, Rats, Sodium Channel Blockers
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المؤلفون: Charles J. Cohen, Brian Safina, Daniel P. Sutherlin, Michael Edward Grimwood, Thilo Focken, J. P. Johnson, Shifeng Liu, Maxim Dauphinais, Matthew Waldbrook, C. Lee Robinette, Girish Bankar, Ivan William Hemeon, Noah G. Shuart, Jae H. Chang, Sultan Chowdhury, David Bogucki, Luis Sojo, Clint Young, Rainbow Kwan, Paul Robert Bichler, Renata Oballa, Tarek S. Mansour, Sophia Lin, Christoph Martin Dehnhardt, Jodie Pang, Navjot Chahal
المصدر: ACS Medicinal Chemistry Letters. 7:277-282
مصطلحات موضوعية: 0301 basic medicine, Drug, Gene isoform, biology, Aryl, Sodium channel, media_common.quotation_subject, Organic Chemistry, Analgesic, Pharmacology, Nav1.5, Biochemistry, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, chemistry, In vivo, Drug Discovery, biology.protein, Potency, 030217 neurology & neurosurgery, media_common
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المؤلفون: Tong-Shuang Li, Simon P. Fricker, Gang Chen, Renato Skerlj, David Bogucki, Markus Metz, Gary Bridger, Susan Nan, Rebecca S.Y. Wong, Dominique Schols, Jean Labrecque, Gloria Lau, Marilyn C. Darkes, Bryon Carpenter
المصدر: Virology. 413(2):231-243
مصطلحات موضوعية: Models, Molecular, Receptors, CCR5, Protein Conformation, Vicriviroc, viruses, Aplaviroc, Drug design, CCR5 receptor antagonist, Computational biology, Biology, Maraviroc, chemistry.chemical_compound, HIV Fusion Inhibitors, Virology, High-Throughput Screening Assays, medicine, Homology modeling, Binding site characterization, virus diseases, Reproducibility of Results, Stereoisomerism, Virus Internalization, Molecular biology, Small molecule, Small molecule antagonists, Antifusogenic assay, chemistry, Mutagenesis, CCR5 Receptor Antagonists, Mutation, HIV-1, Mutagenesis, Site-Directed, CCR5, medicine.drug
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المؤلفون: Renato Skerlj, Gary Bridger, Yuanxi Zhou, Elyse Bourque, Jonathan Langille, Maria Di Fluri, David Bogucki, Wen Yang, Tongshuang Li, Letian Wang, Susan Nan, Ian Baird, Markus Metz, Marilyn Darkes, Jean Labrecque, Gloria Lau, Simon Fricker, Dana Huskens, Dominique Schols
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:2450-2455
مصطلحات موضوعية: Receptors, CCR5, Pyridines, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Virus Replication, Amides, Biochemistry, Rats, Cyclic N-Oxides, Structure-Activity Relationship, Dogs, Piperidines, Drug Design, CCR5 Receptor Antagonists, Oximes, Drug Discovery, HIV-1, Animals, Humans, Molecular Medicine, Molecular Biology
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المؤلفون: Curtis Harwig, Rossana Wauthy, Renato Skerlj, Fluri Maria Di, Yongbao Zhu, Duane Veale, Dominique Schols, Gary Bridger, Helen Yee, Wen Yang, Wilson Trevor R, David Bogucki, Christopher Ronald Smith, Erik De Clercq, Krystyna A. Skupinska, Jonathon Langille, Jason M. Crawford, Dana Huskens, Ernie Mceachern
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:262-266
مصطلحات موضوعية: Receptors, CXCR4, Anti-HIV Agents, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Pharmacology, Butylamines, Virus Replication, Biochemistry, Chemical synthesis, CXCR4, Heterocyclic Compounds, 1-Ring, Structure-Activity Relationship, Chemokine receptor, Dogs, Pharmacokinetics, Drug Discovery, Animals, Humans, Structure–activity relationship, Calcium Signaling, Receptor, Molecular Biology, Chemistry, Organic Chemistry, Antagonist, Virology, Rats, Viral replication, Aminoquinolines, HIV-1, Molecular Medicine, Benzimidazoles
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المؤلفون: Wilson Trevor R, Yuanxi Zhou, Zhongren Wang, David Bogucki, Susan Nan, Katrien Princen, Pedro E. Hernandez-Abad, Renato Skerlj, Jason B. Crawford, Dominique Schols, Eva Maria Boehringer, Sigrid Hatse, Gary Bridger, Markus Metz, Erik De Clercq
المصدر: Journal of Medicinal Chemistry. 53:1250-1260
مصطلحات موضوعية: Receptors, CXCR4, Anti-HIV Agents, Pyridines, Stereochemistry, T-Lymphocytes, T cell, HIV Infections, Virus Replication, Chemical synthesis, Virus, Structure-Activity Relationship, Chemokine receptor, Heterocyclic Compounds, Drug Discovery, medicine, Humans, Structure–activity relationship, Receptor, Molecular Structure, Chemistry, In vitro, medicine.anatomical_structure, Models, Chemical, Biochemistry, Viral replication, HIV-1, Molecular Medicine
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المؤلفون: Curtis Harwig, Dominique Schols, Gang Chen, Wen Yang, Duane Veale, Susan Nan, Simon P. Fricker, Alan Kaller, Danielle Guay, Jason M. Crawford, Michael Satori, Markus Metz, Yongbao Zhu, Helen Yee, Maria Krumpak, Elyse Bourque, Wilson Trevor R, David Bogucki, Bryon Carpenter, Michael Bey, David C. Leitch, Ron MacFarland, David Gauthier, Ian Baird, Rebecca Wong, Renato T. Skerlj, Jonathan Langille, Yuanxi Zhou, Gary Bridger, Renee Mosi, Ernest J. McEachern, Tuya Ba, Tong-Shuang Li, Krystyna Vocadlo, Veronique Bodart
المصدر: Journal of medicinal chemistry. 56(20)
مصطلحات موضوعية: Receptors, CCR5, Anti-HIV Agents, Cell Survival, hERG, Human immunodeficiency virus (HIV), CHO Cells, Pharmacology, medicine.disease_cause, Imidazolidines, Virus Replication, Benzoates, Chemokine receptor, Structure-Activity Relationship, Cricetulus, Piperidines, In vivo, Cricetinae, Drug Discovery, medicine, Animals, Humans, Cells, Cultured, Cardiotoxicity, biology, Molecular Structure, Chemistry, Imidazoles, In vitro, Receptor selectivity, HEK293 Cells, Biochemistry, Models, Chemical, Drug Design, Lipophilicity, CCR5 Receptor Antagonists, Host-Pathogen Interactions, biology.protein, HIV-1, Leukocytes, Mononuclear, Molecular Medicine
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المؤلفون: David Bogucki, Renato Skerlj, Gary J. Bridger
المصدر: Synlett. 2000:1488-1490
مصطلحات موضوعية: Thesaurus (information retrieval), Chemistry, Organic Chemistry, Nucleophilic substitution, Combinatorial chemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::d24a90ff28e579fbb70c3724eea9423d
https://doi.org/10.1055/s-2000-7644