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1
المؤلفون: Pamela A. Benfield, Anna-Marie Etzkorn, Anup Vidwans, Catherine R. Burton, Sarah Cox, David A. Nugiel, Karen A. Rossi, Deborah Doleniak, Steven P. Seitz
المصدر: Journal of Medicinal Chemistry. 45:5224-5232
مصطلحات موضوعية: chemistry.chemical_classification, biology, Chemistry, Kinase, Stereochemistry, Cyclin-dependent kinase 2, Serine, Enzyme, Biochemistry, Cyclin-dependent kinase, Enzyme inhibitor, Drug Discovery, biology.protein, Molecular Medicine, Threonine, Protein kinase A
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2
المؤلفون: Angela Smallwood, Dimeo Susan, Carrie Benware, Eddy W. Yue, David J. Carini, C. Anne Higley, Lisa M. Sisk, David A. Nugiel, Chong-Hwan Chang, Catherine R. Burton, Diane M. Sharp, Pamela A. Benfield, Jodi K. Muckelbauer, Sarah Cox, Steven P. Seitz, Haiying Chen, John F. Boylan, Robert H. Grafstrom, George L. Trainor
المصدر: Journal of Medicinal Chemistry. 45:5233-5248
مصطلحات موضوعية: chemistry.chemical_classification, biology, Molecular model, Kinase, medicine.drug_class, Stereochemistry, Carboxamide, Chemical synthesis, chemistry, Enzyme inhibitor, Cyclin-dependent kinase, Drug Discovery, biology.protein, medicine, Molecular Medicine, Transferase, Alkyl
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3
المؤلفون: Carolyn D. Dzierba, David A. Nugiel, Anup Vidwans
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:5489-5491
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Cyclin-dependent kinase, Cell Line, Tumor, Drug Discovery, CDC2-CDC28 Kinases, Combinatorial Chemistry Techniques, Humans, Moiety, Protein kinase A, Molecular Biology, Cyclin-Dependent Kinase Inhibitor p16, chemistry.chemical_classification, Molecular Structure, biology, Chemistry, Cyclin-Dependent Kinase 2, Organic Chemistry, Cyclin-dependent kinase 2, Biological activity, Cyclin-Dependent Kinases, Semicarbazides, Enzyme, Enzyme inhibitor, Colonic Neoplasms, biology.protein, Molecular Medicine, Drug Screening Assays, Antitumor, Signal transduction, Cell Division
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4
المؤلفون: David A. Nugiel, Karl D. Hardman, Robert A. Copeland, David J. Nelson, Carl P. Decicco, Kim Jacobs
المصدر: Bioorganic & Medicinal Chemistry Letters. 5:3053-3056
مصطلحات موضوعية: Piperazic acid, Stereochemistry, fungi, Organic Chemistry, Clinical Biochemistry, Substituent, Pharmaceutical Science, Biochemistry, Acceptor, chemistry.chemical_compound, chemistry, Amide, Drug Discovery, Molecular Medicine, Molecular Biology
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5
المؤلفون: M Wagner Regina, David A. Nugiel, William K. Schmidt
المصدر: Bioorganic & Medicinal Chemistry Letters. 5:1203-1206
مصطلحات موضوعية: chemistry.chemical_classification, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Amino acid, Substituted urea, chemistry.chemical_compound, chemistry, Drug Discovery, Urea, Molecular Medicine, Molecular Biology, Neurotensin
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6
المؤلفون: David A. Nugiel
المصدر: Tetrahedron Letters. 42:3545-3547
مصطلحات موضوعية: chemistry.chemical_classification, Lanthanide, Organic Chemistry, Biochemistry, Combinatorial chemistry, Cycloaddition, Nitrone, chemistry, Lanthanide trifluoromethanesulfonates, Yield (chemistry), Drug Discovery, 1,3-Dipolar cycloaddition, Stereoselectivity, Trifluoromethanesulfonate
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7
المؤلفون: Steven P. Seitz, Anup Vidwans, Deborah Doleniak, Catherine R. Burton, Ana-Marie Etzkorn, Michael Boisclair, Sarah Cox, Pamela A. Benfield, David A. Nugiel, Phillip M. Czerniak
المصدر: Journal of Medicinal Chemistry. 44:1334-1336
مصطلحات موضوعية: Cyclin E, Cyclin D, Transplantation, Heterologous, Cyclin A, Antineoplastic Agents, CDK-activating kinase, Mice, Structure-Activity Relationship, Cyclin-dependent kinase, Drug Discovery, Tumor Cells, Cultured, Animals, Humans, Enzyme Inhibitors, biology, Chemistry, Cyclin-dependent kinase 4, Cyclin-Dependent Kinases, Biochemistry, biology.protein, Cyclin-dependent kinase complex, Cancer research, Pyrazoles, Molecular Medicine, Drug Screening Assays, Antitumor, Cyclin A2
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8
المؤلفون: Joseph Frey, Zvi Rappoport, David A. Nugiel
المصدر: ChemInform. 22
مصطلحات موضوعية: Chemistry, Organic chemistry, General Medicine, Grignard reagent, Medicinal chemistry
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9
المؤلفون: R. M. Wagner, W. K. Schmidt, David A. Nugiel
المصدر: ChemInform. 26
مصطلحات موضوعية: chemistry.chemical_classification, chemistry.chemical_compound, Chemistry, General Medicine, Combinatorial chemistry, Amino acid, Neurotensin
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10
المؤلفون: Lee T. Bacheler, G. V. De Lucca, Dayton T. Meyer, Ronald M. Klabe, Steven P. Seitz, R. F. Iii Kaltenbach, David A. Nugiel, T. Worley, M. M. Rayner, Kim Jacobs, T. E. Smyser, Mona Patel, Prabhakar K. Jadhav
المصدر: ChemInform. 27
مصطلحات موضوعية: chemistry.chemical_compound, Protease, Stereochemistry, Chemistry, medicine.medical_treatment, medicine, Human immunodeficiency virus (HIV), Urea, Structure–activity relationship, General Medicine, medicine.disease_cause