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1
المؤلفون: Samu Melkko, N. Jarousse, David Archer Ellis, Finton Sirockin, A. Bernardi, Aengus Mac Sweeney, Paul Erbel, Paul Ramage, Philipp Grosche, Eva Altmann, Keith D. Combrink, Nicola Hughes
المصدر: Bioorganic & Medicinal Chemistry Letters. 25:438-443
مصطلحات موضوعية: Adenain, Drug, Peptidomimetic, medicine.medical_treatment, media_common.quotation_subject, Clinical Biochemistry, Pharmaceutical Science, Viral Conjunctivitis, Crystallography, X-Ray, Antiviral Agents, Biochemistry, Adenoviridae, Structure-Activity Relationship, Viral Proteins, Drug Discovery, medicine, Humans, Effective treatment, Protease Inhibitors, Molecular Biology, media_common, Binding Sites, Protease, Tetrapeptide, Chemistry, Organic Chemistry, Virology, Protein Structure, Tertiary, Molecular Docking Simulation, Cysteine Endopeptidases, HEK293 Cells, Drug Design, Molecular Medicine, Structure based, Protein Binding
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2
المؤلفون: Eva Altmann, A. Bernardi, Paul Erbel, Aengus Mac Sweeney, N. Jarousse, Paul Ramage, Philipp Grosche, Keith D. Combrink, Nicola Hughes, David Archer Ellis, Samu Melkko, Finton Sirockin
المصدر: ACS Medicinal Chemistry Letters. 5:937-941
مصطلحات موضوعية: Adenain, Protease, Tetrapeptide, Chemistry, medicine.medical_treatment, Organic Chemistry, Drug Discovery, medicine, Structure based, Biochemistry, Cysteine protease, Combinatorial chemistry, Adenoviral infections
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3
المؤلفون: Karen S. MacMillan, Dale L. Boger, Kristopher E. Boyle, William M. Robertson, James P. Lajiness, David Archer Ellis
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:1854-1857
مصطلحات موضوعية: Alkylating Agents, Indoles, Alkylation, Stereochemistry, Protein subunit, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Article, Duocarmycins, chemistry.chemical_compound, chemistry, Duocarmycin SA, Drug Discovery, Molecular Medicine, Pyrroles, Carboxylate, Oxazoles, Molecular Biology, Pyrrole, Oxazole
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4
المؤلفون: Laurie A. LeBrun, Mei Tsan, Yuefen Zhou, Frank Ruebsam, Darian M. Bartkowski, Alan X. Xiang, Ruhi Kamran, Lian-Sheng Li, Richard E. Showalter, Jingjing Zhao, Rupal Patel, Matthew Lardy, Maria V. Sergeeva, Stephen E. Webber, Amit M. Shah, David Archer Ellis, Zhongxiang Sun, Mcguire Helen, Julie Blazel, Leo Kirkovsky, Daniel A. Norris, Tran Chinh Viet, Charles R. Kissinger, Thomas G. Nolan, Peter S. Dragovich, Qing Han
المصدر: Bioorganic & Medicinal Chemistry Letters. 18:4628-4632
مصطلحات موضوعية: Time Factors, Stereochemistry, Chemistry, Pharmaceutical, Clinical Biochemistry, Molecular Conformation, Thiazines, Pharmaceutical Science, Hepacivirus, Viral Nonstructural Proteins, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Inhibitory Concentration 50, Structure-Activity Relationship, chemistry.chemical_compound, Drug Discovery, Humans, Transferase, Replicon, Molecular Biology, chemistry.chemical_classification, biology, Bicyclic molecule, Organic Chemistry, Sulfoxide, In vitro, Pyridazines, Enzyme, Models, Chemical, chemistry, Enzyme inhibitor, Drug Design, Microsomes, Liver, biology.protein, Molecular Medicine, Caco-2 Cells
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5
المؤلفون: Peter S. Dragovich, Tran Chinh Viet, Yuefen Zhou, Kimkim Dao, Julie K. Blazel, Douglas E. Murphy, Frank Ruebsam, Lian-Sheng Li, David Archer Ellis
المصدر: Synthesis. 2008:610-616
مصطلحات موضوعية: Acylation, Chemistry, Organic Chemistry, Condensation, Moiety, Ethyl malonyl chloride, Ring (chemistry), Medicinal chemistry, Catalysis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::ea7ec7b9cbc76581944128acae51456a
https://doi.org/10.1055/s-2008-1032157 -
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المؤلفون: David Archer Ellis, Karen Wolff, Yun He, Donald S. Karanewsky, Baogen Wu, Hong Yin, Jeremy S. Caldwell, Beth Anaclerio, Kelli L. Kuhen, Badry Bursulaya
المصدر: Bioorganic & Medicinal Chemistry Letters. 16:4246-4251
مصطلحات موضوعية: Models, Molecular, Clinical Biochemistry, Pharmaceutical Science, Quinolones, Virus Replication, Biochemistry, Nucleoside Reverse Transcriptase Inhibitor, Structure-Activity Relationship, Drug Resistance, Viral, Drug Discovery, medicine, Structure–activity relationship, Molecular Biology, chemistry.chemical_classification, Binding Sites, Reverse-transcriptase inhibitor, biology, Chemistry, Organic Chemistry, virus diseases, Nucleotidyltransferase, Virology, HIV Reverse Transcriptase, Reverse transcriptase, Enzyme, Models, Chemical, Viral replication, Enzyme inhibitor, Mutation, HIV-1, biology.protein, Reverse Transcriptase Inhibitors, Molecular Medicine, medicine.drug
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7
المؤلفون: Dale L. Boger, Scott E. Wolkenberg, David Archer Ellis
المصدر: Journal of the American Chemical Society. 123:9299-9306
مصطلحات موضوعية: Alkylating Agents, Indoles, Stereochemistry, Quinolones, Alkylation, Leucomycins, Biochemistry, Catalysis, Duocarmycins, chemistry.chemical_compound, Colloid and Surface Chemistry, Animals, Pyrroles, Leukemia L1210, Binding selectivity, Antibiotics, Antineoplastic, Chemistry, Stereoisomerism, DNA, General Chemistry, DNA-binding domain, Kinetics, DNA Alkylation, Enantiomer, Selectivity
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8
المؤلفون: James P. Lajiness, Dale L. Boger, Karen S. MacMillan, David Archer Ellis, Kristopher E. Boyle, William M. Robertson
المصدر: ChemInform. 41
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Duocarmycin SA, Stereochemistry, Protein subunit, General Medicine, Carboxylate, Alkylation
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9
المؤلفون: Ruhi Kamran, Tran Chinh Viet, Laurie A. LeBrun, Alberto Gobbi, Jingjing Zhao, David Archer Ellis, Qiang Zhao, Julie Blazel, Rupal Patel, Matthew Lardy, Maria V. Sergeeva, Thomas G. Nolan, Qing Han, Stephen E. Webber, Amit M. Shah, Yuefen Zhou, Frank Ruebsam, Richard E. Showalter, Darian M. Bartkowski, Leo Kirkovsky, Alan X. Xiang, Lian-Sheng Li, Douglas E. Murphy, Mei Tsan, Mcguire Helen, Charles R. Kissinger, Daniel A. Norris
المصدر: Bioorganicmedicinal chemistry letters. 19(21)
مصطلحات موضوعية: Stereochemistry, Pyridones, Hepatitis C virus, Clinical Biochemistry, Pharmaceutical Science, Hepacivirus, Viral Nonstructural Proteins, medicine.disease_cause, Crystallography, X-Ray, Biochemistry, Antiviral Agents, chemistry.chemical_compound, Structure-Activity Relationship, RNA polymerase, Drug Discovery, medicine, Structure–activity relationship, Animals, Humans, Enzyme Inhibitors, Molecular Biology, NS5B, chemistry.chemical_classification, Binding Sites, biology, Organic Chemistry, virus diseases, RNA-Dependent RNA Polymerase, Small molecule, digestive system diseases, In vitro, Macaca fascicularis, Enzyme, chemistry, Enzyme inhibitor, biology.protein, Microsomes, Liver, Molecular Medicine
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10
المؤلفون: Noble Michael A, Frank Ruebsam, Lian-Sheng Li, Julie Blazel, Yuefen Zhou, Rupal Patel, Stephen E. Webber, Qing Han, Tran Chinh Viet, Peter S. Dragovich, Maria V. Sergeeva, Charles R. Kissinger, Laurie A. LeBrun, Amit M. Shah, David Archer Ellis, Ruhi Kamran, Douglas E. Murphy, Richard E. Showalter, Mei Tsan, Leo Kirkovsky
المصدر: Bioorganicmedicinal chemistry letters. 18(20)
مصطلحات موضوعية: Molecular model, Genotype, Stereochemistry, Chemistry, Pharmaceutical, Clinical Biochemistry, Molecular Conformation, Pharmaceutical Science, Viral Nonstructural Proteins, Crystallography, X-Ray, Biochemistry, Chemical synthesis, Antiviral Agents, chemistry.chemical_compound, Inhibitory Concentration 50, Structure-Activity Relationship, RNA polymerase, Microsomes, Drug Discovery, Humans, Molecular Biology, NS5B, chemistry.chemical_classification, biology, Bicyclic molecule, Thiadiazines, Organic Chemistry, DNA-Directed RNA Polymerases, Nucleotidyltransferase, Cyclic S-Oxides, Pyridazines, Enzyme, chemistry, Models, Chemical, Enzyme inhibitor, Drug Design, biology.protein, Molecular Medicine, Caco-2 Cells