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1دورية أكاديمية
المؤلفون: Florence Ecoeur, Jessica Weiss, Klemens Kaupmann, Samuel Hintermann, David Orain, Christine Guntermann
المصدر: Frontiers in Immunology, Vol 10 (2019)
مصطلحات موضوعية: retinoic acid receptor-related-orphan-receptor-gamma t, nuclear hormone receptor, T helper 17 differentiation, IL-17, autoimmunity, keratinocytes, Immunologic diseases. Allergy, RC581-607
وصف الملف: electronic resource
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2دورية أكاديمية
المؤلفون: Ulf Guendisch, Jessica Weiss, Florence Ecoeur, Julia Christina Riker, Klemens Kaupmann, Joerg Kallen, Samuel Hintermann, David Orain, Janet Dawson, Andreas Billich, Christine Guntermann
المصدر: PLoS ONE, Vol 12, Iss 11, p e0188391 (2017)
وصف الملف: electronic resource
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3دورية أكاديمية
المؤلفون: David Orain, Guido Koch, Rudolf Giger
المصدر: CHIMIA, Vol 57, Iss 5 (2003)
مصطلحات موضوعية: Combinatorial chemistry, Dakin-west, Natural products, Pictet-spengler, Tryptophan, Chemistry, QD1-999
وصف الملف: electronic resource
Relation: https://www.chimia.ch/chimia/article/view/3701; https://doaj.org/toc/0009-4293; https://doaj.org/toc/2673-2424
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4
المؤلفون: Christine Guntermann, Janet Dawson, Anna Vulpetti, Andreas Billich, Rowan Stringer, Johannes Ottl, Samuel Hintermann, Henri Mattes, Eric Vangrevelinghe, Nigel Graham Cooke, Klemens Kaupmann, Romain M. Wolf, Juergen Wagner, Klemens Hoegenauer, Joerg Kallen, David Orain, David Carcache
المصدر: Journal of Medicinal Chemistry. 61:6724-6735
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Drug Inverse Agonism, Inflammation, 01 natural sciences, 03 medical and health sciences, Transcription (biology), In vivo, RAR-related orphan receptor gamma, Catalytic Domain, Drug Discovery, medicine, Animals, Inverse agonist, Transcription factor, 010405 organic chemistry, Drug discovery, Chemistry, Nuclear Receptor Subfamily 1, Group F, Member 3, Rats, 0104 chemical sciences, Cell biology, Disease Models, Animal, 030104 developmental biology, Molecular Medicine, Female, medicine.symptom
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5
المؤلفون: Klaus Weigand, Andrea Vaupel, Roland Feifel, Berndt Oberhauser, Janet Dawson King, Mark Nash, Pius Loetscher, Amanda Littlewood-Evans, David Orain, Wolfgang Miltz, Juraj Velcicky
المصدر: Journal of Medicinal Chemistry. 60:3672-3683
مصطلحات موضوعية: Nociception, 0301 basic medicine, Angiogenesis, hERG, Administration, Oral, Neovascularization, Physiologic, Inflammation, Pharmacology, 01 natural sciences, Receptors, G-Protein-Coupled, Rats, Sprague-Dawley, Neovascularization, 03 medical and health sciences, Drug Discovery, medicine, Animals, Humans, Receptors, Histamine H3, Receptor, biology, 010405 organic chemistry, Chemistry, Antagonist, Rats, 0104 chemical sciences, HEK293 Cells, 030104 developmental biology, Drug Design, Hyperalgesia, biology.protein, Molecular Medicine, Female, medicine.symptom
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6
المؤلفون: Christine Guntermann, Juergen Wagner, David Orain, Andreas Billich, Joerg Kallen, Samuel Hintermann, Janet Dawson, Rowan Stringer, Henri Mattes, Klemens Kaupmann, David Carcache, Anna Vulpetti
المصدر: ChemMedChem. 11:2640-2648
مصطلحات موضوعية: 0301 basic medicine, Imidazopyridine, Drug Inverse Agonism, Pyridines, Receptors, Retinoic Acid, Stereochemistry, medicine.medical_treatment, Plasma protein binding, Pharmacology, Crystallography, X-Ray, Biochemistry, Inhibitory Concentration 50, 03 medical and health sciences, Pharmacokinetics, RAR-related orphan receptor gamma, Drug Discovery, medicine, Animals, Humans, Potency, Inverse agonist, General Pharmacology, Toxicology and Pharmaceutics, Transcription factor, Cells, Cultured, Binding Sites, Molecular Structure, Chemistry, Interleukin-17, Organic Chemistry, Imidazoles, Nuclear Receptor Subfamily 1, Group F, Member 3, Triazoles, Rats, 030104 developmental biology, Cytokine, Molecular Medicine, Protein Binding
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7Design and Synthesis of Selurampanel, a Novel Orally Active and Competitive AMPA Receptor Antagonist
المؤلفون: David Orain, Kurt Lingenhoehl, Sandrine Desrayaud, David Carcache, Joerg Kallen, Anne Picard, Stephan Urwyler, Phillip Floersheim, Engin Tasdelen, Manuel Koller, Celine Dubois, Samuel Haessig, Henri Mattes
المصدر: ChemMedChem. 12:197-201
مصطلحات موضوعية: 0301 basic medicine, Selurampanel, Administration, Oral, AMPA receptor, Molecular Dynamics Simulation, Pharmacology, Crystallography, X-Ray, Binding, Competitive, Biochemistry, Mice, Structure-Activity Relationship, 03 medical and health sciences, Epilepsy, 0302 clinical medicine, Seizures, Drug Discovery, medicine, Animals, Potency, Receptors, AMPA, General Pharmacology, Toxicology and Pharmaceutics, Receptor, Quinazolinones, chemistry.chemical_classification, Electroshock, Sulfonamides, Binding Sites, Organic Chemistry, Glutamate receptor, Antagonist, medicine.disease, Protein Structure, Tertiary, Sulfonamide, Disease Models, Animal, 030104 developmental biology, chemistry, Drug Design, Molecular Medicine, 030217 neurology & neurosurgery
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8
المؤلفون: David Orain, Christine Guntermann, Samuel Hintermann, Jessica Weiss, Florence Ecoeur, Julia Christina Riker, Janet Dawson, Ulf Guendisch, Andreas Billich, Joerg Kallen, Klemens Kaupmann
المصدر: PLoS ONE
PLoS ONE, Vol 12, Iss 11, p e0188391 (2017)مصطلحات موضوعية: 0301 basic medicine, Male, Physiology, Pyridines, Knees, lcsh:Medicine, Gene Expression, Immune Receptors, Biochemistry, White Blood Cells, RAR-related orphan receptor gamma, Animal Cells, Immune Physiology, Medicine and Health Sciences, Enzyme-Linked Immunoassays, lcsh:Science, Receptor, Promoter Regions, Genetic, Musculoskeletal System, Intraepithelial Lymphocytes, Innate Immune System, Multidisciplinary, Immune System Proteins, T Cells, Interleukin-17, Imidazoles, Cell Differentiation, Receptors, Antigen, T-Cell, gamma-delta, Nuclear Receptor Subfamily 1, Group F, Member 3, Cell biology, Cytokines, Legs, Female, Cellular Types, Anatomy, Research Article, Signal Transduction, Protein Binding, Immune Cells, Immunology, Biology, Research and Analysis Methods, 03 medical and health sciences, In vivo, Cell Line, Tumor, Genetics, Inverse agonist, Animals, Humans, Histone H3 acetylation, Immunoassays, Molecular Biology Techniques, Transcription factor, Molecular Biology, Blood Cells, lcsh:R, Limbs (Anatomy), Biology and Life Sciences, Proteins, Cell Biology, Receptors, Interleukin, Molecular Development, Molecular biology, Arthritis, Experimental, Rats, T Cell Receptors, Kinetics, 030104 developmental biology, HEK293 Cells, Pyrimidines, Nuclear receptor, Gene Expression Regulation, Rats, Inbred Lew, Immune System, Immunologic Techniques, Th17 Cells, lcsh:Q, Ex vivo, Developmental Biology, Cloning
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المؤلفون: Samuel Hintermann, David Orain, Maciej Pudelko, Anna Jedrzejczak, Diego Carballa
المصدر: Synlett. 26:1815-1818
مصطلحات موضوعية: chemistry.chemical_compound, chemistry, Organic Chemistry, Organic chemistry, Nonane, Combinatorial chemistry, Octane
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::11b39d4f5f436c6fcd0eea0d83174c47
https://doi.org/10.1055/s-0034-1378722 -
10
المؤلفون: Christine Guntermann, Joerg Kallen, David Orain, Klemens Hoegenauer, Klemens Kaupmann, Celine Be, Samuel Hintermann, Aude Izaac, Luca Arista
المصدر: ChemMedChem. 12(13)
مصطلحات موضوعية: 0301 basic medicine, Agonist, Imidazopyridine, Hydrocarbons, Fluorinated, Stereochemistry, medicine.drug_class, Pyridines, Crystallography, X-Ray, Biochemistry, 03 medical and health sciences, 0302 clinical medicine, Drug Discovery, medicine, Inverse agonist, Humans, Sulfones, General Pharmacology, Toxicology and Pharmaceutics, Binding site, Transcription factor, Adaptor Proteins, Signal Transducing, Pharmacology, Orphan receptor, Sulfonamides, Binding Sites, Chemistry, Organic Chemistry, Imidazoles, Nuclear Proteins, Water, Nuclear Receptor Subfamily 1, Group F, Member 3, Nuclear Receptor Interacting Protein 1, Retinoic acid receptor, 030104 developmental biology, Models, Chemical, 030220 oncology & carcinogenesis, Helix, Molecular Medicine, Cholesterol Esters