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1
المؤلفون: Barbara Hibner, Nancy Kennure, Bernd Riedl, Donald John Wolanin, Wendy Lee, Xiao-Gao Liu, Reina Natero, Donald Bankston, Hong Rong, Uday Khire, Todd Gane, Roger A. Smith, Robert O. Carlson, Jacques Dumas, Ian McAlexander, Jill Kingery-Wood, Sarah Heald, Timothy B. Lowinger, Jeffrey Johnson, Robert Sibley, James Barbosa, Joel Renick, Michael E Katz, Yolanda V Caringal, David R. Brittelli, Mary-Katherine Monahan
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:783-786
مصطلحات موضوعية: biology, medicine.drug_class, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Substituent, Pharmaceutical Science, Carboxamide, Biochemistry, Chemical synthesis, chemistry.chemical_compound, chemistry, Enzyme inhibitor, Amide, Mitogen-activated protein kinase, Drug Discovery, biology.protein, medicine, Molecular Medicine, Structure–activity relationship, Protein kinase A, Molecular Biology
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2
المؤلفون: Dixon Brian R, Jinshan Chen, David R. Brittelli, Jacques Dumas
المصدر: Tetrahedron Letters. 40:9195-9199
مصطلحات موضوعية: Sulfonyl, chemistry.chemical_classification, Organic Chemistry, Cathepsin D, Biochemistry, Solution phase, Combinatorial chemistry, Small molecule, chemistry.chemical_compound, chemistry, Nucleophile, Reagent, Amide, Drug Discovery, Organic chemistry
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3
المؤلفون: Robert Sibley, Dixon Brian R, David R. Brittelli, Gerhard Konig, Stephen K.-F. Wong, Jinshan Chen, Jacques Dumas, James A. Witowsky, Holia Hatoum-Mokdad
المصدر: Bioorganic & Medicinal Chemistry Letters. 9:2531-2536
مصطلحات موضوعية: medicine.drug_class, High-throughput screening, Clinical Biochemistry, Pharmaceutical Science, Cathepsin D, Carboxamide, Biochemistry, Chemical synthesis, Structure-Activity Relationship, Drug Discovery, medicine, Humans, Protease Inhibitors, Molecular Biology, chemistry.chemical_classification, biology, Chemistry, Organic Chemistry, Small molecule, In vitro, Enzyme, Liver, Enzyme inhibitor, biology.protein, Molecular Medicine
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4
المؤلفون: Patricia C. Weber, Robert M. Knabb, Matthew M. Abelman, Charles A. Kettner, David R. Brittelli, John M. Fevig
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:295-300
مصطلحات موضوعية: Cyclohexane, Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Tryptophan, Pharmaceutical Science, Crystal structure, Ring (chemistry), Biochemistry, Pyrrolidine, chemistry.chemical_compound, Thrombin, Drug Discovery, medicine, Side chain, Molecular Medicine, Molecular Biology, medicine.drug, Discovery and development of direct thrombin inhibitors
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5
المؤلفون: Richard S. Alexander, Robert M. Knabb, Joseph Cacciola, John M. Fevig, Patricia C. Weber, David R. Brittelli, Charles A. Kettner
المصدر: Bioorganic & Medicinal Chemistry Letters. 6:301-306
مصطلحات موضوعية: biology, Chemistry, Stereochemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Active site, Biochemistry, Thrombin, Drug Discovery, biology.protein, medicine, Molecular Medicine, Molecular Biology, medicine.drug, Discovery and development of direct thrombin inhibitors
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6
المؤلفون: David R. Brittelli, H. S. Kezar, Walter Adelman Gregory, Peter Franklin Corless, Chung-Ho Park, A M Slee, R. J. Mcripley, V. S. Eberly, M. Forbes, M. A. Wuonola, R. K. Carlson, Chia-Lin J. Wang, S. J. Miller, P. Rajagopalan
المصدر: ChemInform. 22
مصطلحات موضوعية: Substitution reaction, chemistry.chemical_compound, chemistry, Stereochemistry, Group (periodic table), medicine.drug_class, Aryl, Antibiotics, medicine, General Medicine
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7
المؤلفون: Victor Johannes Nickolson, George A. Boswell, Rouxi Lan, Leonard Cook, S. William Tam, Alexander L. Johnson, Robert J. Chorvat, Xusheng Zhang, Chuan Wang, Richard M. Scribner, Richard A. Earl, Hua Wenting, Baoyu Mi, Wendell Wilkie Wilkerson, Robert Zaczek, Melvyn John Myers, M. A. Wuonola, David R. Brittelli
المصدر: Bioorganic & Medicinal Chemistry Letters. 2:851-854
مصطلحات موضوعية: Stereochemistry, Chemistry, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Biochemistry, Drug Discovery, Core (graph theory), medicine, Molecular Medicine, Enhancer, Molecular Biology, Acetylcholine, medicine.drug
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8
المؤلفون: Ronald J. McRipley, Andrew M. Slee, Frank D. Marsh, Virginia S. Eberly, David R. Brittelli, M. A. Wuonola, Chung Ho Park, Martin Forbes, Wang Chia-Lin Jeffrey, Walter Adelman Gregory
المصدر: Journal of Medicinal Chemistry. 35:1156-1165
مصطلحات موضوعية: Staphylococcus aureus, biology, medicine.drug_class, Stereochemistry, Aryl, Carboxamide, Microbial Sensitivity Tests, Electrophilic aromatic substitution, biology.organism_classification, Ring (chemistry), Enterococcus faecalis, Anti-Bacterial Agents, Structure-Activity Relationship, chemistry.chemical_compound, chemistry, Drug Discovery, medicine, Molecular Medicine, Structure–activity relationship, Antibacterial activity, Oxazoles, Antibacterial agent
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::557089b2434c915f304341413cc7222e
https://doi.org/10.1021/jm00084a022 -
9
المؤلفون: James W. Darrow, Aaron Bourret, Robert Desimone, Jin-Ming Xiong, Patricia Maciejewski, Seung H. Lee, David C. Eustice, Mihaela Diana Danca, Douglas A. Pippin, David R. Brittelli, Kropf Jeffrey E, Peter Blomgren, Melissa Hill-Drzewi, Kevin S. Currie, Lisa Elkin, Steven L. Gallion, Scott A. Mitchell
المصدر: Bioorganicmedicinal chemistry letters. 19(24)
مصطلحات موضوعية: animal structures, Angiogenesis, Clinical Biochemistry, Receptor, EphB4, Pharmaceutical Science, Angiogenesis Inhibitors, Biochemistry, Receptor tyrosine kinase, chemistry.chemical_compound, Growth factor receptor, Cell Line, Tumor, Drug Discovery, Humans, Urea, Receptor, Molecular Biology, Protein Kinase Inhibitors, biology, Phenylurea Compounds, Organic Chemistry, Imidazoles, Angiopoietin receptor, Vascular endothelial growth factor, chemistry, Pyrazines, embryonic structures, biology.protein, Cancer research, Molecular Medicine, Signal transduction, Platelet-derived growth factor receptor
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10
المؤلفون: D. C. Eustice, Chia-Lin J. Wang, P. T. Bartholomew, M. Forbes, David R. Brittelli, Andrew M. Slee, M. A. Wuonola, R. J. Mcripley, W. A. Gregory, V. S. Eberly
المصدر: Journal of Medicinal Chemistry. 33:2569-2578
مصطلحات موضوعية: chemistry.chemical_classification, Staphylococcus aureus, Ketone, Chemical Phenomena, Stereochemistry, medicine.drug_class, Aryl, Substituent, Carboxamide, Microbial Sensitivity Tests, Electrophilic aromatic substitution, Anti-Bacterial Agents, Chemistry, Structure-Activity Relationship, chemistry.chemical_compound, Ketyl, chemistry, Drug Discovery, Enterococcus faecalis, medicine, Molecular Medicine, Oxazoles, Alkyl, Antibacterial agent
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::08ae7d5de14ba9bd56c9ab466850c168
https://doi.org/10.1021/jm00171a035