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1دورية أكاديمية
المؤلفون: William N Pappano, Jun Guo, Yupeng He, Debra Ferguson, Sujatha Jagadeeswaran, Donald J Osterling, Wenqing Gao, Julie K Spence, Marina Pliushchev, Ramzi F Sweis, Fritz G Buchanan, Michael R Michaelides, Alexander R Shoemaker, Chris Tse, Gary G Chiang
المصدر: PLoS ONE, Vol 10, Iss 7, p e0131716 (2015)
وصف الملف: electronic resource
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2
المؤلفون: Jonathan Hickson, Letty M Medina, Debra Ferguson, Xin Huang, Susan Bolin, David Frost, Andrew Oleksijew, Natalie A Bratcher
المصدر: Journal of the American Association for Laboratory Animal Science. 58:583-588
مصطلحات موضوعية: Oncology, medicine.medical_specialty, Pain, Mice, SCID, Mice, 03 medical and health sciences, 0302 clinical medicine, Laboratory Animal Science, 030202 anesthesiology, Internal medicine, Ovarian carcinoma, medicine, Carcinoma, Animals, Humans, Pain Management, Bioluminescence imaging, Anesthesia, Ovarian Neoplasms, Pain, Postoperative, business.industry, Cancer, medicine.disease, Buprenorphine, Analgesics, Opioid, Clinical trial, Opioid, 030220 oncology & carcinogenesis, Female, Animal Science and Zoology, Analgesia, business, Ovarian cancer, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::ad33da7922a05f50719c4e2507fab7d4
https://doi.org/10.30802/aalas-jaalas-18-000127 -
3
المؤلفون: Velitchka Bontcheva, Maricel Torrent, David Maag, Anthony Mastracchio, Fritz G. Buchanan, Loren M. Lasko, Debra Ferguson, Thomas D. Penning, Alexander R. Shoemaker, Kenneth D. Bromberg, Chunqiu Lai, Eric F. Johnson
المصدر: Bioorganic & Medicinal Chemistry Letters. 29:1481-1486
مصطلحات موضوعية: biology, 010405 organic chemistry, Chemistry, Kinase, Organic Chemistry, Clinical Biochemistry, Pharmaceutical Science, Cell Cycle Proteins, Protein-Tyrosine Kinases, 01 natural sciences, Biochemistry, Combinatorial chemistry, 0104 chemical sciences, Structure-Activity Relationship, 010404 medicinal & biomolecular chemistry, Wee1, G2/M checkpoint, Heterocyclic Compounds, In vivo, Drug Discovery, biology.protein, Humans, Molecular Medicine, Molecular Biology, Human breast
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4
المؤلفون: Marina Konopleva, Tamar Uziel, Xiaoli Huang, Weiguo Feng, Xiaoyu Lin, Warren M. Kati, Lloyd T. Lam, Vinitha Mary Kuruvilla, Mai H. Bui, Emily J. Faivre, Tianyu Cai, Jenny Rowe, Daniel H. Albert, Richard J. Bellin, Lu Zhang, Zheng Zha, Sriram S. Shanmugavelandy, Paul Hessler, Michael Boyiadzis, Gaurav Mehta, Antonio Cavazos, Keith F. McDaniel, Joshua P. Plotnik, Terrance J. Magoc, Xin Lu, Debra Ferguson, Yu Shen, Lina Han, Neal Goodwin, Qi Zhang, Kathleen A. Dorritie
المصدر: Molecular cancer therapeutics. 20(10)
مصطلحات موضوعية: Cancer Research, BRD4, Pyridines, Androgen Receptor Positive, Antineoplastic Agents, Apoptosis, Mice, SCID, BET inhibitor, Prostate cancer, chemistry.chemical_compound, Mice, Therapeutic index, Mice, Inbred NOD, medicine, Tumor Cells, Cultured, Animals, Humans, Pyrroles, Cell Proliferation, Sulfonamides, Venetoclax, business.industry, Myeloid leukemia, Proteins, medicine.disease, Bridged Bicyclo Compounds, Heterocyclic, Xenograft Model Antitumor Assays, Bromodomain, Leukemia, Myeloid, Acute, Oncology, chemistry, Proto-Oncogene Proteins c-bcl-2, Cancer research, Drug Therapy, Combination, Female, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8076aa78b9f6209f8ff644313a95c59b
https://pubmed.ncbi.nlm.nih.gov/34253595 -
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المؤلفون: Loren M. Lasko, Clarissa G. Jakob, Rohinton P. Edalji, Wei Qiu, Debra Montgomery, Enrico L. Digiammarino, T. Matt Hansen, Roberto M. Risi, Robin Frey, Vlasios Manaves, Bailin Shaw, Mikkel Algire, Paul Hessler, Lloyd T. Lam, Tamar Uziel, Emily Faivre, Debra Ferguson, Fritz G. Buchanan, Ruth L. Martin, Maricel Torrent, Gary G. Chiang, Kannan Karukurichi, J. William Langston, Brian T. Weinert, Chunaram Choudhary, Peter de Vries, Arthur F. Kluge, Michael A. Patane, John H. Van Drie, Ce Wang, David McElligott, Ed Kesicki, Ronen Marmorstein, Chaohong Sun, Philip A. Cole, Saul H. Rosenberg, Michael R. Michaelides, Albert Lai, Kenneth D. Bromberg
المصدر: Nature. 550:128-132
مصطلحات موضوعية: Male, Models, Molecular, 0301 basic medicine, Protein Conformation, Antineoplastic Agents, Mice, SCID, P300-CBP Transcription Factors, Crystallography, X-Ray, Binding, Competitive, Heterocyclic Compounds, 4 or More Rings, Mice, 03 medical and health sciences, Acetyl Coenzyme A, Catalytic Domain, Cell Line, Tumor, Neoplasms, Animals, Humans, Cell Lineage, p300-CBP Transcription Factors, Epigenetics, Enzyme Inhibitors, Cell Proliferation, Histone Acetyltransferases, Regulation of gene expression, Multidisciplinary, biology, Chemistry, Histone acetyltransferase, Xenograft Model Antitumor Assays, Gene Expression Regulation, Neoplastic, Prostatic Neoplasms, Castration-Resistant, 030104 developmental biology, Histone, Receptors, Androgen, Acetylation, Hematologic Neoplasms, Biocatalysis, biology.protein, Cancer research, Histone deacetylase
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6
المؤلفون: Chunqiu Lai, Alexander R. Shoemaker, Fritz G. Buchanan, Eric F. Johnson, David Maag, Anthony Mastracchio, Velitchka Bontcheva, Kenneth D. Bromberg, Thomas D. Penning, Debra Ferguson, Maricel Torrent, Loren M. Lasko
المصدر: Bioorganic & Medicinal Chemistry Letters. 30:126895
مصطلحات موضوعية: Wee1, biology, Stereochemistry, Kinase, Chemistry, Organic Chemistry, Clinical Biochemistry, Drug Discovery, biology.protein, Pharmaceutical Science, Molecular Medicine, Molecular Biology, Biochemistry
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7
المؤلفون: Philip J. Merta, Amanda M. Olson, Fritz G. Buchanan, Nirupama B. Soni, Donald J. Osterling, Alan S. Florjancic, Debra Ferguson, David Maag, Eric F. Johnson, Yunsong Tong, Alexander R. Shoemaker, Maricel Torrent, Kenneth D. Bromberg, Thomas D. Penning, Loren M. Lasko
المصدر: ACS Medicinal Chemistry Letters. 6:58-62
مصطلحات موضوعية: chemistry.chemical_classification, Molecular model, biology, Pyrimidine, Chemistry, Kinase, Organic Chemistry, Pharmacology, Biochemistry, Wee1, chemistry.chemical_compound, Pharmacokinetics, Drug Discovery, biology.protein, Pharmacophore, Cytotoxicity, Tricyclic
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8
المؤلفون: Xiaoli Huang, Terrance J. Magoc, Debra Ferguson, Emily J. Faivre, Xiaoyu Lin, Paul Hessler, Richard J. Bellin, Warren M. Kati, Daniel H. Albert, Lloyd T. Lam, Mai Ha Bui, Tamar Uziel, Denise Wilcox, Keith F. McDaniel, Yu Shen
المصدر: Cancer Research. 78:800-800
مصطلحات موضوعية: 0301 basic medicine, Cancer Research, BRD4, business.industry, Cancer, medicine.disease, Bromodomain, BET inhibitor, 03 medical and health sciences, Leukemia, Myelogenous, Prostate cancer, 030104 developmental biology, Oncology, Tolerability, Cancer research, Medicine, business
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::fec401590f04fd2752ba7e2f5ca2352b
https://doi.org/10.1158/1538-7445.am2018-800 -
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المؤلفون: Ruth L. Martin, Peter de Vries, Rohinton Edalji, T. Matt Hansen, Mikkel Algire, Fritz G. Buchanan, Wei Qiu, Brian T. Weinert, John H. Van Drie, Debra Ferguson, Kesicki Edward A, Ronen Marmorstein, Enrico L. Digiammarino, Philip A. Cole, Lloyd T. Lam, Chunaram Choudhary, Robin R. Frey, Loren M. Lasko, Roberto M. Risi, Kannan R. Karukurichi, Michael A. Patane, Debra Montgomery, Kenneth D. Bromberg, Bailin Shaw, Michael R. Michaelides, David L. McElligott, Arthur F. Kluge, J. William Langston, Ce Wang, Chaohong Sun, Vlasios Manaves, Emily J. Faivre, Maricel Torrent, Gary G. Chiang, Paul Hessler, Albert Lai, Saul H. Rosenberg, Clarissa G. Jakob, Tamar Uziel
المصدر: Nature. 558:E1-E1
مصطلحات موضوعية: 0301 basic medicine, 03 medical and health sciences, Lineage specific, 030104 developmental biology, 0302 clinical medicine, Multidisciplinary, History, 030220 oncology & carcinogenesis, Interpretation (philosophy), Published Erratum, Cancer therapy, Library science, Article
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المؤلفون: Roberto M. Risi, Todd M. Hansen, Clarissa G. Jakob, Mikkel Algire, Tamar Uziel, Lloyd T. Lam, Kenneth D. Bromberg, Vlasios Manaves, Loren M. Lasko, Robin R. Frey, Maricel Torrent, Saul H. Rosenberg, Ruth L. Martin, Debra Montgomery, Bailin Shaw, Michael R. Michaelides, Enrico L. Digiammarino, Wei Qiu, Albert Lai, Paul Hessler, Emily Favire, Fritz G. Buchanan, Debra Ferguson
المصدر: Molecular Cancer Therapeutics. 17:LB-A23
مصطلحات موضوعية: Histone Acetyltransferases, Cancer Research, biology, medicine.drug_class, Chemistry, Cancer, Androgen, medicine.disease, Androgen receptor, Prostate cancer, Histone, Oncology, Acetylation, Cancer research, medicine, biology.protein, Epigenetics
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::16f9918b04e2fa27f6f2e3b6b4a3f001
https://doi.org/10.1158/1535-7163.targ-17-lb-a23