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المؤلفون: Deborah W. Knapp, Deepika Dhawan, Alexander W. Enstrom, Lindsey M. Fourez, Sagar M. Utturkar, Noel Dybdal, Elaine Murray, Uma K. Aryal, Matthew Breen, Ketaki P. Bhide, Christopher M. Fulkerson, Jackeline Franco, Mark Merchant, Rodrigo Mohallem, Liling Liu, José A. Ramos-Vara, Dietrich Tuerck, Audrey Ruple, Tanja S. Zabka, Paul Rossman
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::09e7ae2e500d87ca6f391e089070a4cd
https://doi.org/10.1158/1535-7163.22522869.v1 -
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المؤلفون: Deborah W. Knapp, Deepika Dhawan, Alexander W. Enstrom, Lindsey M. Fourez, Sagar M. Utturkar, Noel Dybdal, Elaine Murray, Uma K. Aryal, Matthew Breen, Ketaki P. Bhide, Christopher M. Fulkerson, Jackeline Franco, Mark Merchant, Rodrigo Mohallem, Liling Liu, José A. Ramos-Vara, Dietrich Tuerck, Audrey Ruple, Tanja S. Zabka, Paul Rossman
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::8f37959f372c1b7d271e50d8816599d6
https://doi.org/10.1158/1535-7163.22522854.v1 -
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المؤلفون: Deborah W. Knapp, Deepika Dhawan, Alexander W. Enstrom, Lindsey M. Fourez, Sagar M. Utturkar, Noel Dybdal, Elaine Murray, Uma K. Aryal, Matthew Breen, Ketaki P. Bhide, Christopher M. Fulkerson, Jackeline Franco, Mark Merchant, Rodrigo Mohallem, Liling Liu, José A. Ramos-Vara, Dietrich Tuerck, Audrey Ruple, Tanja S. Zabka, Paul Rossman
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::1c1c60f2e19eca00cad7cad9a5b7a25c
https://doi.org/10.1158/1535-7163.c.6543510.v1 -
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المؤلفون: Kenichi Umehara, Yumi Cleary, Stephen Fowler, Neil Parrott, Dietrich Tuerck
المصدر: Drug Metabolism and Disposition. 50:214-223
مصطلحات موضوعية: Isoenzymes, Pharmacology, Leukemia, Myeloid, Acute, Pyrrolidines, para-Aminobenzoates, Cytochrome P-450 CYP3A, Cytochrome P-450 CYP3A Inhibitors, Humans, Pharmaceutical Science, Drug Interactions, Models, Biological, Risk Assessment
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2ba778aa8ad3f0b7d543d3c6a7fc42f7
https://doi.org/10.1124/dmd.121.000720 -
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المؤلفون: Agnès Poirier, Heidemarie Kletzl, Cordula Stillhart, Stephen Fowler, Kenichi Umehara, Andreas Guenther, Andreas Brink, Nicole A. Kratochwil, Dietrich Tuerck, Christophe Husser, Mark Savage, Mohammed Ullah, Lutz Mueller, Yumi Cleary, Katja Heinig
المصدر: Drug Metabolism and Disposition. 50:65-75
مصطلحات موضوعية: Pharmacology, Drug, Chemistry, In silico, media_common.quotation_subject, Pharmaceutical Science, Computational biology, Small molecule, Drug development, Pharmacokinetics, In vivo, Distribution (pharmacology), ADME, media_common
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::a42eb9cb10d47b49d0cb86fb0a1206ac
https://doi.org/10.1124/dmd.121.000563 -
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المؤلفون: Uma K. Aryal, Paul M Rossman, Christopher M. Fulkerson, Noel Dybdal, Mark Merchant, Jackeline Franco, Deepika Dhawan, Sagar M. Utturkar, Audrey Ruple, Matthew Breen, Alexander W. Enstrom, Elaine R Murray, Dietrich Tuerck, Lindsey M. Fourez, José A. Ramos-Vara, Deborah W. Knapp, Tanja S. Zabka, Rodrigo Mohallem, Ketaki Bhide, Liling Liu
المصدر: Molecular Cancer Therapeutics. 20:2177-2188
مصطلحات موضوعية: Cancer Research, business.industry, Invasive urothelial carcinoma, Cancer, Drug resistance, medicine.disease, Immune system, Oncology, Pharmacokinetics, Pharmacodynamics, Cancer research, Medicine, business, Adverse effect, Vemurafenib, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::f2d3dbfca305640309f510cd29c85567
https://doi.org/10.1158/1535-7163.mct-20-0893 -
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المؤلفون: Stephen, Fowler, Andreas, Brink, Yumi, Cleary, Andreas, Günther, Katja, Heinig, Christophe, Husser, Heidemarie, Kletzl, Nicole, Kratochwil, Lutz, Mueller, Mark, Savage, Cordula, Stillhart, Dietrich, Tuerck, Mohammed, Ullah, Kenichi, Umehara, Agnès, Poirier
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 50(1)
مصطلحات موضوعية: Survival of Motor Neuron 2 Protein, Pyrimidines, Pharmaceutical Preparations, RNA Splicing, Animals, Humans, Tissue Distribution, RNA, Messenger, In Vitro Techniques, Azo Compounds
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::4530dce338c940f32f354504129eb183
https://pubmed.ncbi.nlm.nih.gov/34620695 -
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المؤلفون: Paul, Rossman, Tanja S, Zabka, Audrey, Ruple, Dietrich, Tuerck, José A, Ramos-Vara, Liling, Liu, Rodrigo, Mohallem, Mark, Merchant, Jackeline, Franco, Christopher M, Fulkerson, Ketaki P, Bhide, Matthew, Breen, Uma K, Aryal, Elaine, Murray, Noel, Dybdal, Sagar M, Utturkar, Lindsey M, Fourez, Alexander W, Enstrom, Deepika, Dhawan, Deborah W, Knapp
المصدر: Molecular cancer therapeutics. 20(11)
مصطلحات موضوعية: Proto-Oncogene Proteins B-raf, Carcinoma, Transitional Cell, Disease Models, Animal, Dogs, Adolescent, Vemurafenib, Mutation, Animals, Humans, Child
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::c8de518ec5c08d0dfebb3b62019c95ab
https://pubmed.ncbi.nlm.nih.gov/34433660 -
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المؤلفون: Jürgen Bachl, Michael Hettich, Bruno Gomes, Maria Amann, Greg Dugan, Mark A. Cline, Sai Kumar Solingapuram Kiran, Wouter H. P. Driessen, Estelle Marrer-Berger, Jason M. Grayson, David L. Caudell, Volker Teichgräber, Flavio Crameri, Christina Claus, Christian Klein, Oliver Krieter, Stefan Evers, Dietrich Tuerck, Maurizio Ceppi
المصدر: Cancer Research. 80:6135-6135
مصطلحات موضوعية: Agonist, Cancer Research, medicine.drug_class, business.industry, Immunogenicity, medicine.medical_treatment, Translational medicine, Immune system, Oncology, Cancer immunotherapy, Pharmacodynamics, Cancer research, medicine, Endocrine system, business, Cancer immunology
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::3e97a769ec05daeff3e989059f66ae0a
https://doi.org/10.1158/1538-7445.am2020-6135 -
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المؤلفون: Tianle Yang, Hasane Ratni, Emmanuel Pinard, Nanjing Zhang, Hongyan Qi, Nikolai Naryshkin, Priya Vazirani, Stephan Kirchner, Xiaoyan Zhang, Karen S. Chen, Amal Dakka, Lutz Mueller, Friedrich Metzger, Woll Matthew G, Sergey Paushkin, Xin Zhao, Marla Weetall, Gary Mitchell Karp, Kathleen D. McCarthy, Agnès Poirier, Wolfgang Muster, Pascale David-Pierson, Luke Green, Irene Gerlach, Anthony Turpoff, Dietrich Tuerck
المصدر: Journal of Medicinal Chemistry. 59:6086-6100
مصطلحات موضوعية: 0301 basic medicine, Pyrimidinones, SMN1, Biology, medicine.disease_cause, Muscular Atrophy, Spinal, Mice, 03 medical and health sciences, Exon, 0302 clinical medicine, Drug Discovery, medicine, Animals, Humans, RNA, Messenger, Genetics, Messenger RNA, Mutation, Alternative splicing, Exons, Spinal muscular atrophy, medicine.disease, SMA, nervous system diseases, Survival of Motor Neuron 2 Protein, Alternative Splicing, 030104 developmental biology, RNA splicing, Cancer research, Molecular Medicine, 030217 neurology & neurosurgery