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1دورية أكاديمية
المؤلفون: Hanan S. Anbar, Mohammed I. El-Gamal, Hamadeh Tarazi, Bong S. Lee, Hong R. Jeon, Dow Kwon, Chang-Hyun Oh
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 35, Iss 1, Pp 1712-1726 (2020)
مصطلحات موضوعية: apoptosis, imidazothiazole, melanoma, modelling, v600e-b-raf, Therapeutics. Pharmacology, RM1-950
وصف الملف: electronic resource
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2
المؤلفون: Bong Sang Lee, Hong R. Jeon, Dow Kwon, Chang-Hyun Oh, Mohammed I. El-Gamal, Hanan S. Anbar, Hamadeh Tarazi
المصدر: Journal of Enzyme Inhibition and Medicinal Chemistry, Vol 35, Iss 1, Pp 1712-1726 (2020)
Journal of Enzyme Inhibition and Medicinal Chemistry
article-version (VoR) Version of Recordمصطلحات موضوعية: Proto-Oncogene Proteins B-raf, Imidazothiazole, Quantitative Structure-Activity Relationship, Antineoplastic Agents, RM1-950, Molecular Dynamics Simulation, 01 natural sciences, modelling, chemistry.chemical_compound, Cell Line, Tumor, Drug Discovery, Oximes, medicine, melanoma, Humans, Protein Kinase Inhibitors, v600e-b-raf, Cell Proliferation, Pharmacology, Sulfonamides, 010405 organic chemistry, Chemistry, Melanoma, Imidazoles, apoptosis, imidazothiazole, Raf kinase, General Medicine, Sorafenib, medicine.disease, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, Thiazoles, Vemurafenib, Apoptosis, Cancer research, Molecular mechanism, Carbamates, Therapeutics. Pharmacology, Drug Screening Assays, Antitumor, Imidazothiazole derivatives, V600E, Research Article, Research Paper
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3
المؤلفون: Eslam M.H. Ali, Garam Kim, Young Jik Kwon, Usama M. Ammar, Dong Keun Han, Mahmoud M. Gamal El-Din, Karim I. Mersal, Hong R. Jeon, Bong Sang Lee, Kyung-Tae Lee, Kyung Ho Yoo, Jae Kyun Lee, Mohammed I. El-Gamal, Kwan Hyi Lee, Hong Seok Choi, Chang Hyun Oh, Dow Kwon, Mohammed S. Abdel-Maksoud
مصطلحات موضوعية: MAPK/ERK pathway, Kinase, Cellular Assay, chemistry.chemical_compound, chemistry, Biochemistry, In vivo, Drug Discovery, Cancer cell, Molecular Medicine, Thiazole, RB, Sulfamide, V600E
وصف الملف: application/pdf
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4
المؤلفون: Mohammed S, Abdel-Maksoud, Mohammed I, El-Gamal, Bong S, Lee, Mahmoud M, Gamal El-Din, Hong R, Jeon, Dow, Kwon, Usama M, Ammar, Karim I, Mersal, Eslam M H, Ali, Kyung-Tae, Lee, Kyung Ho, Yoo, Dong Keun, Han, Jae Kyun, Lee, Garam, Kim, Hong Seok, Choi, Young Jik, Kwon, Kwan Hyi, Lee, Chang Hyun, Oh
المصدر: Journal of medicinal chemistry. 64(10)
مصطلحات موضوعية: Mitogen-Activated Protein Kinase Kinases, Proto-Oncogene Proteins B-raf, Sulfonamides, Binding Sites, Transplantation, Heterologous, Drug Evaluation, Preclinical, Imidazoles, Molecular Docking Simulation, Mice, Structure-Activity Relationship, Thiazoles, Drug Stability, Cell Line, Tumor, Animals, Humans, Drug Screening Assays, Antitumor, Phosphorylation, Melanoma, Protein Kinase Inhibitors, Cell Proliferation, Half-Life
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5
المؤلفون: Seung Mok Lee, Dow Kwon, Eun Ju Kim, Chan Wong Park, Yong Sik Kim, Joo Byung Chae, Kil Do Cho, In Hoi Huh, Dong Yeun Kim
المصدر: Arzneimittelforschung. 51:204-213
مصطلحات موضوعية: Male, Antiulcer drug, medicine.drug_class, Proton-pump inhibitor, In Vitro Techniques, Pharmacology, 2-Pyridinylmethylsulfinylbenzimidazoles, Gastric Acid, Rats, Sprague-Dawley, chemistry.chemical_compound, Oral administration, Drug Discovery, medicine, Animals, Enzyme Inhibitors, Aminopyrine, Omeprazole, Parietal cell, Stomach, Proton Pump Inhibitors, Anti-Ulcer Agents, Rats, medicine.anatomical_structure, chemistry, Biochemistry, Gastric Mucosa, Sulfoxides, Gastric acid, Benzimidazoles, Pentagastrin, Rabbits, Histamine, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2365dfd53eb0a0c34b276c8383e70fd0
https://doi.org/10.1055/s-0031-1300026 -
6
المؤلفون: Bong Sang Lee, Ji Yun Moon, Mohammed I. El-Gamal, Dong Jin Lee, Won-Jai Choi, Hyun-Il Kim, Dow Kwon, Sun Ahe Lee, Chang-Hyun Oh, Young-Jin Cho, Hanan S. Anbar, Hong-Ryeol Jeon, Hye Jin Chung
المصدر: Bioorganicmedicinal chemistry letters. 23(5)
مصطلحات موضوعية: Male, Clinical Biochemistry, Cmax, Pharmaceutical Science, Biological Availability, Tetrazoles, Pharmacology, Biochemistry, Rats, Sprague-Dawley, Rat liver microsomes, Pharmacokinetics, Ester prodrug, Drug Stability, Drug Discovery, medicine, Animals, Prodrugs, Molecular Biology, Antihypertensive Agents, Gastric Juice, Chemistry, Organic Chemistry, Imidazoles, Esters, Prodrug, In vitro, Bioavailability, Rats, Microsomes, Liver, Molecular Medicine, Olmesartan, Angiotensin II Type 1 Receptor Blockers, medicine.drug