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1
المؤلفون: Renato Skerlj, Tuya Ba, Ernest J. McEachern, Elyse Bourque, Ian Baird, Dominique Schols, Wilson Trevor R, Renee Mosi, Jonathan Langille, Yuanxi Zhou, Bryon Carpenter, Michael Bey, Simon P. Fricker, Dana Huskens, Duane Veale, Rebecca S.Y. Wong, Gary Bridger, Curtis Harwig, Veronique Bodart, Ron MacFarland, Markus Metz, Sanjay Danthi
المصدر: ACS Medicinal Chemistry Letters. 3:216-221
مصطلحات موضوعية: congenital, hereditary, and neonatal diseases and abnormalities, biology, business.industry, Purkinje fibers, Organic Chemistry, hERG, Human immunodeficiency virus (HIV), Pharmacology, medicine.disease_cause, Biochemistry, Bioavailability, Chemokine receptor, medicine.anatomical_structure, Drug Discovery, Lipophilicity, biology.protein, Medicine, Action potential duration, cardiovascular diseases, business, Ion channel
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2
المؤلفون: Renato Skerlj, Gary Bridger, Yuanxi Zhou, Elyse Bourque, Ernest McEachern, Jonathan Langille, Curtis Harwig, Duane Veale, Wen Yang, Tongshong Li, Yongbao Zhu, Michael Bey, Ian Baird, Michael Sartori, Markus Metz, Renee Mosi, Kim Nelson, Veronique Bodart, Rebecca Wong, Simon Fricker, Ron Mac Farland, Dana Huskens, Dominique Schols
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:6950-6954
مصطلحات موضوعية: Tertiary amine, Anti-HIV Agents, Pyridines, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, CCR5 receptor antagonist, Pharmacology, Virus Replication, Biochemistry, Peripheral blood mononuclear cell, Chemical synthesis, Inhibitory Concentration 50, Dogs, Piperidines, Drug Discovery, medicine, Animals, Humans, Structure–activity relationship, Molecular Biology, Molecular Structure, Chemistry, Organic Chemistry, virus diseases, Amides, In vitro, Rats, Viral replication, Drug Design, CCR5 Receptor Antagonists, HIV-1, Leukocytes, Mononuclear, Molecular Medicine
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3
المؤلفون: Curtis Harwig, Rossana Wauthy, Renato Skerlj, Fluri Maria Di, Yongbao Zhu, Duane Veale, Dominique Schols, Gary Bridger, Helen Yee, Wen Yang, Wilson Trevor R, David Bogucki, Christopher Ronald Smith, Erik De Clercq, Krystyna A. Skupinska, Jonathon Langille, Jason M. Crawford, Dana Huskens, Ernie Mceachern
المصدر: Bioorganic & Medicinal Chemistry Letters. 21:262-266
مصطلحات موضوعية: Receptors, CXCR4, Anti-HIV Agents, Clinical Biochemistry, Administration, Oral, Pharmaceutical Science, Pharmacology, Butylamines, Virus Replication, Biochemistry, Chemical synthesis, CXCR4, Heterocyclic Compounds, 1-Ring, Structure-Activity Relationship, Chemokine receptor, Dogs, Pharmacokinetics, Drug Discovery, Animals, Humans, Structure–activity relationship, Calcium Signaling, Receptor, Molecular Biology, Chemistry, Organic Chemistry, Antagonist, Virology, Rats, Viral replication, Aminoquinolines, HIV-1, Molecular Medicine, Benzimidazoles
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4
المصدر: Canadian Journal of Chemistry. 82:240-253
مصطلحات موضوعية: Aqueous solution, Proton, 1-Naphthol, Organic Chemistry, General Chemistry, Photochemistry, Catalysis, Naphthoquinone, Quinone, chemistry.chemical_compound, chemistry, Intramolecular force, Excited state, Phenol
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5
المؤلفون: Curtis Harwig, Dominique Schols, Gang Chen, Wen Yang, Duane Veale, Susan Nan, Simon P. Fricker, Alan Kaller, Danielle Guay, Jason M. Crawford, Michael Satori, Markus Metz, Yongbao Zhu, Helen Yee, Maria Krumpak, Elyse Bourque, Wilson Trevor R, David Bogucki, Bryon Carpenter, Michael Bey, David C. Leitch, Ron MacFarland, David Gauthier, Ian Baird, Rebecca Wong, Renato T. Skerlj, Jonathan Langille, Yuanxi Zhou, Gary Bridger, Renee Mosi, Ernest J. McEachern, Tuya Ba, Tong-Shuang Li, Krystyna Vocadlo, Veronique Bodart
المصدر: Journal of medicinal chemistry. 56(20)
مصطلحات موضوعية: Receptors, CCR5, Anti-HIV Agents, Cell Survival, hERG, Human immunodeficiency virus (HIV), CHO Cells, Pharmacology, medicine.disease_cause, Imidazolidines, Virus Replication, Benzoates, Chemokine receptor, Structure-Activity Relationship, Cricetulus, Piperidines, In vivo, Cricetinae, Drug Discovery, medicine, Animals, Humans, Cells, Cultured, Cardiotoxicity, biology, Molecular Structure, Chemistry, Imidazoles, In vitro, Receptor selectivity, HEK293 Cells, Biochemistry, Models, Chemical, Drug Design, Lipophilicity, CCR5 Receptor Antagonists, Host-Pathogen Interactions, biology.protein, HIV-1, Leukocytes, Mononuclear, Molecular Medicine
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6
المؤلفون: Dana Huskens, Ernest J. McEachern, Yongbao Zhu, Helen Yee, Krystyna A. Skupinska, Michael Sartori, Alan Kaller, Gary Bridger, Renato Skerlj, Erik De Clercq, Duane Veale, Ian Baird, Letian Wang, Kate Burrage, Dominique Schols, Wen Yang, Christopher Ronald Smith, Curtis Harwig, Rossana Wauthy
المصدر: Bioorganicmedicinal chemistry letters. 21(5)
مصطلحات موضوعية: DNA Replication, Receptors, CXCR4, Tertiary amine, Anti-HIV Agents, Clinical Biochemistry, Pharmaceutical Science, Butylamines, Virus Replication, Biochemistry, CXCR4, Virus, Heterocyclic Compounds, 1-Ring, Dogs, Pharmacokinetics, Drug Discovery, Structure–activity relationship, Animals, Molecular Biology, biology, Molecular Structure, Chemistry, Organic Chemistry, biology.organism_classification, Virology, humanities, In vitro, Rats, Viral replication, Drug Design, Lentivirus, Aminoquinolines, HIV-1, Molecular Medicine, Benzimidazoles
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7
المؤلفون: Duane Veale, Jason B. Crawford, Gary Bridger, Erik De Clercq, Dominique Schols, Ernest J. McEachern, Bem Atsma, Katrien Princen, Jonathon Langille, Renato Skerlj, Yuanxi Zhou, Al Kaller, Curtis Harwig, Sigrid Hatse, Susan Nan, Wilson Trevor R
المصدر: Journal of medicinal chemistry. 53(8)
مصطلحات موضوعية: Receptors, CXCR4, Cell Membrane Permeability, Anti-HIV Agents, Administration, Oral, Biological Availability, CCR5 receptor antagonist, Pharmacology, Butylamines, Virus Replication, Cell Line, Chemokine receptor, Heterocyclic Compounds, 1-Ring, Radioligand Assay, Structure-Activity Relationship, Dogs, Drug Discovery, Structure–activity relationship, Animals, Humans, Receptor, CXCR4 antagonist, Chemistry, Stereoisomerism, Small molecule, Rats, Viral replication, Cell culture, Aminoquinolines, HIV-1, Leukocytes, Mononuclear, Molecular Medicine, Benzimidazoles, Calcium