-
1دورية أكاديمية
المؤلفون: Dung DTM; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Vietnam., Park EJ; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Cheongju, Chungbuk, 28160, Republic of Korea., Anh DT; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Vietnam., Phan DTP; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Vietnam., Na IH; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Cheongju, Chungbuk, 28160, Republic of Korea., Kwon JH; Korea Research Institute of Bioscience and Biotechnology, Cheongju, Chungbuk, Republic of Korea., Kang JS; Korea Research Institute of Bioscience and Biotechnology, Cheongju, Chungbuk, Republic of Korea., Tung TT; Faculty of Pharmacy, PHENIKAA University, Hanoi, 12116, Vietnam.; PHENIKAA Institute for Advanced Study (PIAS), PHENIKAA University, Hanoi, 12116, Vietnam., Han SB; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Cheongju, Chungbuk, 28160, Republic of Korea. shan@chungbuk.ac.kr., Nam NH; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Vietnam. doctornam@gmail.com.
المصدر: Scientific reports [Sci Rep] 2022 Feb 21; Vol. 12 (1), pp. 2886. Date of Electronic Publication: 2022 Feb 21.
نوع المنشور: Journal Article; Research Support, Non-U.S. Gov't
بيانات الدورية: Publisher: Nature Publishing Group Country of Publication: England NLM ID: 101563288 Publication Model: Electronic Cited Medium: Internet ISSN: 2045-2322 (Electronic) Linking ISSN: 20452322 NLM ISO Abbreviation: Sci Rep Subsets: MEDLINE
مواضيع طبية MeSH: Antineoplastic Agents* , Drug Design* , Enzyme Activators*, Hydrazines/*chemical synthesis , Hydrazines/*pharmacology, Apoptosis/drug effects ; Caspase 3/metabolism ; Cell Cycle/drug effects ; Cell Line, Tumor ; Colonic Neoplasms/pathology ; Drug Screening Assays, Antitumor/methods ; Humans ; Lung Neoplasms/pathology ; Male ; Prostatic Neoplasms/pathology
-
2دورية أكاديمية
المؤلفون: Dung DTM; Department of Pharmaceutical Chemistry, Hanoi University of Pharmacy, Hanoi, Vietnam., Park EJ; College of Pharmacy, Chungbuk National University, Cheongju, Chungbuk, Republic of Korea., Anh DT; Department of Pharmaceutical Chemistry, Hanoi University of Pharmacy, Hanoi, Vietnam., Hai PT; Department of Pharmaceutical Chemistry, Hanoi University of Pharmacy, Hanoi, Vietnam., Huy LD; Department of Pharmaceutical Chemistry, Hanoi University of Pharmacy, Hanoi, Vietnam., Jun HW; College of Pharmacy, Chungbuk National University, Cheongju, Chungbuk, Republic of Korea., Kwon JH; Korea Research Institute of Bioscience and Biotechnology, Cheongju, Chungbuk, Republic of Korea., Young Ji A; College of Pharmacy, Chungbuk National University, Cheongju, Chungbuk, Republic of Korea., Kang JS; Korea Research Institute of Bioscience and Biotechnology, Cheongju, Chungbuk, Republic of Korea., Tung TT; Faculty of Pharmacy, PHENIKAA University, Hanoi, Vietnam.; PHENIKAA Institute for Advanced Study (PIAS), PHENIKAA University, Hanoi, Vietnam., Dung PTP; Department of Pharmaceutical Chemistry, Hanoi University of Pharmacy, Hanoi, Vietnam., Han SB; College of Pharmacy, Chungbuk National University, Cheongju, Chungbuk, Republic of Korea., Nam NH; Department of Pharmaceutical Chemistry, Hanoi University of Pharmacy, Hanoi, Vietnam.
المصدر: Archiv der Pharmazie [Arch Pharm (Weinheim)] 2022 Jan; Vol. 355 (1), pp. e2100216. Date of Electronic Publication: 2021 Oct 21.
نوع المنشور: Comparative Study; Journal Article
بيانات الدورية: Publisher: Wiley-VCH Verlag GmbH & Co. KGaA Country of Publication: Germany NLM ID: 0330167 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1521-4184 (Electronic) Linking ISSN: 03656233 NLM ISO Abbreviation: Arch Pharm (Weinheim) Subsets: MEDLINE
مواضيع طبية MeSH: Antineoplastic Agents/*pharmacology , Benzylidene Compounds/*pharmacology , Hydrazines/*pharmacology , Quinolones/*pharmacology, Antineoplastic Agents/chemical synthesis ; Antineoplastic Agents/chemistry ; Benzylidene Compounds/chemical synthesis ; Benzylidene Compounds/chemistry ; Cell Line, Tumor ; Colonic Neoplasms/drug therapy ; Fluorouracil/pharmacology ; Humans ; Hydrazines/chemical synthesis ; Hydrazines/chemistry ; Lung Neoplasms/drug therapy ; Male ; Molecular Docking Simulation ; PC-3 Cells ; Prostatic Neoplasms/drug therapy ; Quinolones/chemical synthesis ; Quinolones/chemistry ; Structure-Activity Relationship
-
3دورية أكاديمية
المؤلفون: Dung DTM; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, 10000, Vietnam., Park EJ; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Chungbuk, 28160, Republic of Korea., Anh DT; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, 10000, Vietnam., Hai PT; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, 10000, Vietnam., Bao LQ; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, 10000, Vietnam., Ji AY; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Chungbuk, 28160, Republic of Korea., Kang JS; Korea Research Institute of Bioscience and Biotechnology, Cheongju, Chungbuk, 28116, Republic of Korea., Tung TT; Faculty of Pharmacy, Phenikaa University, Hanoi 12116, Vietnam.; PHENIKAA Institute for Advanced Study (PIAS), Phenikaa University, Hanoi 12116, Vietnam., Han SB; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Chungbuk, 28160, Republic of Korea., Nam NH; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, 10000, Vietnam.
المصدر: Anti-cancer agents in medicinal chemistry [Anticancer Agents Med Chem] 2022; Vol. 22 (14), pp. 2586-2598.
نوع المنشور: Journal Article; Research Support, Non-U.S. Gov't
بيانات الدورية: Publisher: Bentham Science Publishers Country of Publication: Netherlands NLM ID: 101265649 Publication Model: Print Cited Medium: Internet ISSN: 1875-5992 (Electronic) Linking ISSN: 18715206 NLM ISO Abbreviation: Anticancer Agents Med Chem Subsets: MEDLINE
مواضيع طبية MeSH: Antineoplastic Agents*/chemistry, Caspase 3/metabolism ; Caspases/metabolism ; Cell Line, Tumor ; Cell Proliferation ; Drug Screening Assays, Antitumor ; Humans ; Hydrazines ; Molecular Docking Simulation ; Structure-Activity Relationship
-
4دورية أكاديمية
المؤلفون: Anh DT; Department of Pharmaceutical Chemistry, Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi 10000, Vietnam., Hai PT; Department of Pharmaceutical Chemistry, Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi 10000, Vietnam., Huy LD; Department of Pharmaceutical Chemistry, Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi 10000, Vietnam., Ngoc HB; Department of Pharmaceutical Chemistry, Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi 10000, Vietnam., Ngoc TTM; Department of Pharmaceutical Chemistry, Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi 10000, Vietnam., Dung DTM; Department of Pharmaceutical Chemistry, Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi 10000, Vietnam., Park EJ; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Cheongju, Chungbuk 28160, Republic of Korea., Song IK; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Cheongju, Chungbuk 28160, Republic of Korea., Kang JS; Laboratory Animal Resource Center, Korea Research Institute of Bioscience and Biotechnology, Cheongju, Chungbuk 28116, Republic of Korea., Kwon JH; Laboratory Animal Resource Center, Korea Research Institute of Bioscience and Biotechnology, Cheongju, Chungbuk 28116, Republic of Korea., Tung TT; Faculty of Pharmacy, PHENIKAA University, Hanoi 12116, Vietnam.; PHENIKAA Institute for Advanced Study (PIAS), PHENIKAA University, Hanoi 12116, Vietnam., Han SB; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Cheongju, Chungbuk 28160, Republic of Korea., Nam NH; Department of Pharmaceutical Chemistry, Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi 10000, Vietnam.
المصدر: ACS omega [ACS Omega] 2021 Feb 08; Vol. 6 (7), pp. 4907-4920. Date of Electronic Publication: 2021 Feb 08 (Print Publication: 2021).
نوع المنشور: Journal Article
بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101691658 Publication Model: eCollection Cited Medium: Internet ISSN: 2470-1343 (Electronic) Linking ISSN: 24701343 NLM ISO Abbreviation: ACS Omega Subsets: PubMed not MEDLINE
-
5دورية أكاديمية
المؤلفون: Huan LC; Hanoi University of Pharmacy, Hanoi, Vietnam.; Thai Binh University of Medicine and Pharmacy, Thai Binh City, Vietnam., Anh DT; Hanoi University of Pharmacy, Hanoi, Vietnam., Hai PT; Hanoi University of Pharmacy, Hanoi, Vietnam., Anh LD; Hanoi University of Pharmacy, Hanoi, Vietnam., Park EJ; College of Pharmacy, Chungbuk National University, Cheongju, Republic of Korea., Ji AY; College of Pharmacy, Chungbuk National University, Cheongju, Republic of Korea., Kang JS; Bio-Evaluation Center, Korea Research Institute of Bioscience and Biotechnology, Cheongju, Republic of Korea., Dung DTM; Hanoi University of Pharmacy, Hanoi, Vietnam., Oanh DTK; Hanoi University of Pharmacy, Hanoi, Vietnam., Tung TT; Faculty of Pharmacy, PHENIKAA University, Hanoi, Vietnam.; PHENIKAA Institute for Advanced Study (PIAS), PHENIKAA University, Hanoi, Vietnam., Hai DTT; Hanoi University of Pharmacy, Hanoi, Vietnam., Han SB; College of Pharmacy, Chungbuk National University, Cheongju, Republic of Korea., Nam NH; Hanoi University of Pharmacy, Hanoi, Vietnam.
المصدر: Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2020 Dec; Vol. 35 (1), pp. 1854-1865.
نوع المنشور: Journal Article
بيانات الدورية: Publisher: Taylor & Francis Country of Publication: England NLM ID: 101150203 Publication Model: Print Cited Medium: Internet ISSN: 1475-6374 (Electronic) Linking ISSN: 14756366 NLM ISO Abbreviation: J Enzyme Inhib Med Chem Subsets: MEDLINE
مواضيع طبية MeSH: Antineoplastic Agents/*chemical synthesis , Caspase Inhibitors/*chemical synthesis , Caspases, Initiator/*metabolism , Hydrazines/*chemical synthesis, Antineoplastic Agents/pharmacology ; Apoptosis/drug effects ; Caspase Inhibitors/pharmacology ; Cell Line, Tumor ; Cell Proliferation/drug effects ; Drug Screening Assays, Antitumor ; Humans ; Hydrazines/pharmacology ; Isatin/chemistry ; Molecular Docking Simulation ; Structure-Activity Relationship
-
6دورية أكاديمية
المؤلفون: Anh DT; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Viet Nam., Hai PT; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Viet Nam., Dung DTM; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Viet Nam., Dung PTP; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Viet Nam., Huong LT; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Viet Nam., Park EJ; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Cheongju, Chungbuk 28160, Republic of Korea., Jun HW; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Cheongju, Chungbuk 28160, Republic of Korea., Kang JS; Laboratory Animal Resource Center, Korea Research Institute of Bioscience and Biotechnology, Cheongju, Chungbuk, Republic of Korea., Kwon JH; Laboratory Animal Resource Center, Korea Research Institute of Bioscience and Biotechnology, Cheongju, Chungbuk, Republic of Korea., Tung TT; Faculty of Pharmacy, PHENIKAA University, Hanoi 12116, Viet Nam; PHENIKAA Institute for Advanced Study (PIAS), PHENIKAA University, Hanoi 12116, Viet Nam., Han SB; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Cheongju, Chungbuk 28160, Republic of Korea. Electronic address: shan@chungbuk.ac.kr., Nam NH; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Viet Nam. Electronic address: namnh@hup.edu.vn.
المصدر: Bioorganic & medicinal chemistry letters [Bioorg Med Chem Lett] 2020 Nov 15; Vol. 30 (22), pp. 127537. Date of Electronic Publication: 2020 Sep 08.
نوع المنشور: Journal Article; Research Support, Non-U.S. Gov't
بيانات الدورية: Publisher: Elsevier Science Ltd Country of Publication: England NLM ID: 9107377 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1464-3405 (Electronic) Linking ISSN: 0960894X NLM ISO Abbreviation: Bioorg Med Chem Lett Subsets: MEDLINE
مواضيع طبية MeSH: Amides/*pharmacology , Antineoplastic Agents/*pharmacology , Histone Deacetylase 2/*antagonists & inhibitors , Histone Deacetylase 6/*antagonists & inhibitors , Histone Deacetylase Inhibitors/*pharmacology, Amides/chemical synthesis ; Amides/chemistry ; Antineoplastic Agents/chemical synthesis ; Antineoplastic Agents/chemistry ; Cell Line, Tumor ; Cell Proliferation/drug effects ; Dose-Response Relationship, Drug ; Drug Design ; Drug Screening Assays, Antitumor ; Histone Deacetylase 2/metabolism ; Histone Deacetylase 6/metabolism ; Histone Deacetylase Inhibitors/chemical synthesis ; Histone Deacetylase Inhibitors/chemistry ; Humans ; Indoles/chemistry ; Indoles/pharmacology ; Molecular Structure ; Structure-Activity Relationship
-
7دورية أكاديمية
المؤلفون: Anh DT; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Viet Nam., Hai PT; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Viet Nam., Huong LT; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Viet Nam., Park EJ; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Cheongju, Chungbuk 28160, Republic of Korea., Jun HW; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Cheongju, Chungbuk 28160, Republic of Korea., Kang JS; Laboratory Animal Resource Center, Korea Research Institute of Bioscience and Biotechnology, Cheongju, Chungbuk, Republic of Korea., Kwon JH; Laboratory Animal Resource Center, Korea Research Institute of Bioscience and Biotechnology, Cheongju, Chungbuk, Republic of Korea., Dung DTM; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Viet Nam., Anh VT; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Viet Nam., Hue VTM; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Viet Nam. Electronic address: namnh@hup.edu.vn., Han SB; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Cheongju, Chungbuk 28160, Republic of Korea., Nam NH; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Viet Nam. Electronic address: shan@chungbuk.ac.kr.
المصدر: Bioorganic chemistry [Bioorg Chem] 2020 Aug; Vol. 101, pp. 103988. Date of Electronic Publication: 2020 Jun 01.
نوع المنشور: Journal Article; Research Support, Non-U.S. Gov't
بيانات الدورية: Publisher: Elsevier Country of Publication: United States NLM ID: 1303703 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1090-2120 (Electronic) Linking ISSN: 00452068 NLM ISO Abbreviation: Bioorg Chem Subsets: MEDLINE
مواضيع طبية MeSH: Antineoplastic Agents/*pharmacology , Histone Deacetylase Inhibitors/*pharmacology , Hydroxamic Acids/*pharmacology , Oxazoles/*chemistry , Thiazoles/*chemistry, Antineoplastic Agents/chemistry ; Apoptosis/drug effects ; Cell Line, Tumor ; Drug Screening Assays, Antitumor ; Histone Deacetylase Inhibitors/chemistry ; Humans ; Hydroxamic Acids/chemistry ; Molecular Docking Simulation ; Spectrum Analysis/methods ; Structure-Activity Relationship
-
8دورية أكاديمية
المؤلفون: Lan TT; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, 10000, Vietnam., Anh DT; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, 10000, Vietnam., Pham-The H; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, 10000, Vietnam., Dung DTM; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, 10000, Vietnam., Park EJ; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Cheongju, Chungbuk, 28160, Republic of, Korea., Jang SD; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Cheongju, Chungbuk, 28160, Republic of, Korea., Kwon JH; Bio-Evaluation Center, Korea Research Institute of Bioscience and Biotechnology, Cheongju, Chungbuk, 28116, Republic of, Korea., Kang JS; Bio-Evaluation Center, Korea Research Institute of Bioscience and Biotechnology, Cheongju, Chungbuk, 28116, Republic of, Korea., Thuan NT; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, 10000, Vietnam., Han SB; College of Pharmacy, Chungbuk National University, 194-31, Osongsaengmyung-1, Heungdeok, Cheongju, Chungbuk, 28160, Republic of, Korea., Nam NH; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, 10000, Vietnam.
المصدر: Chemistry & biodiversity [Chem Biodivers] 2020 Jul; Vol. 17 (7), pp. e2000290. Date of Electronic Publication: 2020 Jun 23.
نوع المنشور: Journal Article
بيانات الدورية: Publisher: Verlag Helvetica Chimica Acta Country of Publication: Switzerland NLM ID: 101197449 Publication Model: Print-Electronic Cited Medium: Internet ISSN: 1612-1880 (Electronic) Linking ISSN: 16121872 NLM ISO Abbreviation: Chem Biodivers Subsets: MEDLINE
مواضيع طبية MeSH: Drug Design*, Acetylcholinesterase/*metabolism , Antineoplastic Agents/*pharmacology , Cholinesterase Inhibitors/*pharmacology, Antineoplastic Agents/chemical synthesis ; Antineoplastic Agents/chemistry ; Biphenyl Compounds/antagonists & inhibitors ; Cell Cycle/drug effects ; Cell Proliferation/drug effects ; Cholinesterase Inhibitors/chemical synthesis ; Cholinesterase Inhibitors/chemistry ; Dose-Response Relationship, Drug ; Drug Screening Assays, Antitumor ; Humans ; Molecular Docking Simulation ; Molecular Structure ; Picrates/antagonists & inhibitors ; Structure-Activity Relationship ; Tumor Cells, Cultured
-
9دورية أكاديمية
المؤلفون: Dung DTM; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Vietnam., Huan NV; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Vietnam., Cam DM; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Vietnam., Hieu DC; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Vietnam., Hai PT; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Vietnam., Huong LT; School of Medicine and Pharmacy, Hanoi National University, Hanoi, Vietnam., Kim J; College of Pharmacy, Chungbuk National University, Cheongju, Chungbuk 28160, Korea., Choi JE; College of Pharmacy, Chungbuk National University, Cheongju, Chungbuk 28160, Korea., Kang JS; Bio-Evaluation Center, Korea Research Institute of Bioscience and Biotechnology, Cheongju, Chungbuk, Korea., Han SB; College of Pharmacy, Chungbuk National University, Cheongju, Chungbuk 28160, Korea., Nam NH; Hanoi University of Pharmacy, 13-15 Le Thanh Tong, Hanoi, Vietnam.
المصدر: Medicinal chemistry (Shariqah (United Arab Emirates)) [Med Chem] 2018; Vol. 14 (8), pp. 831-850.
نوع المنشور: Journal Article
بيانات الدورية: Publisher: Bentham Science Publishers Country of Publication: Netherlands NLM ID: 101240303 Publication Model: Print Cited Medium: Internet ISSN: 1875-6638 (Electronic) Linking ISSN: 15734064 NLM ISO Abbreviation: Med Chem Subsets: MEDLINE
مواضيع طبية MeSH: Antineoplastic Agents/*pharmacology , Histone Deacetylase Inhibitors/*pharmacology , Hydroxamic Acids/*pharmacology , Indoles/*pharmacology , Triazoles/*pharmacology, Antineoplastic Agents/chemical synthesis ; Antineoplastic Agents/chemistry ; Catalytic Domain ; Cell Line, Tumor ; Histone Deacetylase Inhibitors/chemical synthesis ; Histone Deacetylase Inhibitors/chemistry ; Humans ; Hydroxamic Acids/chemical synthesis ; Hydroxamic Acids/chemistry ; Indoles/chemical synthesis ; Indoles/chemistry ; Molecular Docking Simulation ; Structure-Activity Relationship ; Triazoles/chemical synthesis ; Triazoles/chemistry ; Vorinostat/pharmacology