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1
المؤلفون: Qian Wang, Sybil O'Connor, Alan Roberts, Brian W. Metcalf, Leslie Hall, Maxim Soloviev, Michael Hansbury, Greg Hollis, Xin He, Matthew C. Stubbs, Niu Shin, Wenqing Yao, Kamna Katiyar, Phillip C.C. Liu, Kathy Wang, Sharon Diamond, Brent Douty, Gengjie Yang, Dana Shuey, Maryanne B. Covington, Paul Collier, Mingming Gao, Patricia Feldman, Peggy Scherle, Timothy Burn, Andrew P. Combs, Yun-Long Li, Lynn Leffet, Robert C. Newton, Paul Waeltz, Holly Koblish, Jin Lu, Swamy Yeleswaram, Yanlong Li, Reid Huber, Robert Collins, Eddy W. Yue
المصدر: Journal of Pharmacology and Experimental Therapeutics. 374:211-222
مصطلحات موضوعية: 0301 basic medicine, Pharmacology, Phosphoinositide 3-kinase, biology, Cell growth, business.industry, medicine.disease, In vitro, Lymphoma, 03 medical and health sciences, 030104 developmental biology, 0302 clinical medicine, Mechanism of action, In vivo, Cell culture, biology.protein, Cancer research, Molecular Medicine, Medicine, medicine.symptom, business, 030217 neurology & neurosurgery, PI3K/AKT/mTOR pathway
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::450ddea425cecfdf40bf1184c7e8c723
https://doi.org/10.1124/jpet.120.265538 -
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المؤلفون: Andrew P Combs, Niu Shin, Laurine Galya, James Hall, Sharon Diamond, Kevin Baptiste, Jason Boer, Yan-ou Yang, Kevin J Bowman, Maryanne B Covington, Yanlong Li, Xin He, Daniel Levy, Brent D Douty, Padmaja Polam, David M Burns, Artem Shvartsbart, Eddy W Yue, Rick Sparks, Nikoo Falahatpisheh, Lixin Shao, Stacey Shepard, Andrew W Buesking
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::68d9b46276e455cc32362364091e1119
https://doi.org/10.1021/scimeetings.0c06483 -
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المؤلفون: Niu, Shin, Matthew, Stubbs, Holly, Koblish, Eddy W, Yue, Maxim, Soloviev, Brent, Douty, Kathy He, Wang, Qian, Wang, Mingming, Gao, Patricia, Feldman, Gengjie, Yang, Leslie, Hall, Michael, Hansbury, Sybil, O'Connor, Lynn, Leffet, Robert, Collins, Kamna, Katiyar, Xin, He, Paul, Waeltz, Paul, Collier, Jin, Lu, Yun-Long, Li, Yanlong, Li, Phillip C C, Liu, Timothy, Burn, Maryanne, Covington, Sharon, Diamond, Dana, Shuey, Alan, Roberts, Swamy, Yeleswaram, Greg, Hollis, Brian, Metcalf, Wenqing, Yao, Reid, Huber, Andrew, Combs, Robert, Newton, Peggy, Scherle
المصدر: The Journal of pharmacology and experimental therapeutics. 374(1)
مصطلحات موضوعية: Pyrrolidines, Lymphoma, Antineoplastic Agents, Xenograft Model Antitumor Assays, Disease Models, Animal, Mice, Phosphatidylinositol 3-Kinases, Pyrimidines, Liver, Cell Line, Tumor, Animals, Humans, Immunologic Factors, Pyrazoles, Female, Phosphoinositide-3 Kinase Inhibitors
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::14a526e7b4c814d8f260a1bead68f92f
https://pubmed.ncbi.nlm.nih.gov/32345620 -
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المؤلفون: Brian M. Glass, Padmaja Polam, Tom Emm, Kevin Bowman, Jordan S. Fridman, Holly Koblish, Richard Wynn, Michael Hansbury, Yanlong Li, Eddy W. Yue, Brian Metcalf, Michael J. Bower, Min Wei, Richard B. Sparks, Peggy Scherle, Xiangdong Liu, Andrew P. Combs, Timothy Burn, Dilip P. Modi, Brian Wayland, Qian Wang, Lynn Leffet, Brent Douty, Wenyu Zhu, Amy Takvorian, Joseph Glenn
المصدر: ACS Medicinal Chemistry Letters
مصطلحات موضوعية: 0301 basic medicine, Letter, Organic Chemistry, data-centric medicinal chemistry, Pembrolizumab, Pharmacology, Furazan, Biochemistry, Small molecule, In vitro, Bioavailability, 03 medical and health sciences, chemistry.chemical_compound, 030104 developmental biology, 0302 clinical medicine, IDO1, chemistry, INCB24360, 030220 oncology & carcinogenesis, Drug Discovery, Epacadostat, Indoleamine 2,3-dioxygenase, immuno-oncology, Sulfamide, ADME
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المؤلفون: Swamy Yeleswaram, Thomas Maduskuie, Brian Wayland, Hao Feng, Patricia Feldman, Niu Shin, Yanlong Li, Chu-Biao Xue, Peggy Scherle, Song Mei, Kathy Wang, Maryanne Covington, Wenqing Yao, Padmaja Polam, Richard B. Sparks, Wenyu Zhu, Xin He, Sharon Diamond, Eddy W. Yue, Chunhong He, Brian Metcalf, Holly Koblish, Ke Zhang, Nikoo Falahatpisheh, Brent Douty, Leslie Hall, Yu Li, Andrew P. Combs, Joseph Glenn, Kamna Katiyar, Yun-Long Li
المصدر: ACS Med Chem Lett
مصطلحات موضوعية: Purine, Phosphoinositide 3-kinase, biology, 010405 organic chemistry, Organic Chemistry, Pharmacology, 01 natural sciences, Biochemistry, Duvelisib, Pyrazolopyrimidine, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, chemistry.chemical_compound, chemistry, Pharmacokinetics, In vivo, Drug Discovery, biology.protein, Idelalisib, ADME
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المؤلفون: Niu Shin, Yan-Ou Yang, Eddy W. Yue, Monika Scuron, Eduardo Huarte, Paul Smith, Melissa Parker, Brittany Fay, Andrew P. Combs
المصدر: Poster Presentations.
مصطلحات موضوعية: Autoimmune disease, biology, business.industry, T cell, Lupus nephritis, Autoantibody, medicine.disease, Pathogenesis, medicine.anatomical_structure, Shareholder, Immunology, medicine, biology.protein, Antibody, business, B cell
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::ae312724c779bf38bc75a0e1bf42ac91
https://doi.org/10.1136/annrheumdis-2019-eular.4990 -
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المؤلفون: Paul Waeltz, Liang-Chuan S. Wang, Gregory Hollis, Yue Zhang, Eddy W. Yue, Nikoo Falahatpisheh, Reid Huber, Peggy Scherle, Timothy Burn, Thomas Maduskuie, Brent Douty, Yun-Long Li, Gengjie Yang, Andrew P. Combs, Holly Koblish, Mark Rupar, Michael Hansbury
المصدر: Journal for Immunotherapy of Cancer
مصطلحات موضوعية: Pharmacology, Cancer Research, Tumor microenvironment, T cell, medicine.medical_treatment, Immunology, FOXP3, Immunotherapy, Biology, Immune system, medicine.anatomical_structure, Oncology, Poster Presentation, medicine, Molecular Medicine, Immunology and Allergy, Cytotoxic T cell, IL-2 receptor, CD8
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المؤلفون: Qian Wang, Holly Koblish, Andrew P. Combs, Richard Wynn, Lynn Leffet, Robert C. Newton, Padmaja Polam, Kevin Bowman, Xiangdong Liu, Eddy W. Yue, Richard B. Sparks, Paul Waeltz, Peggy Scherle, Timothy Burn, Niu Shin, Gengjie Yang, Mark Rupar, Michael Hansbury, Jordan S. Fridman, Beth Thomas, Yanlong Li, Kathy Wang
المصدر: Blood. 115:3520-3530
مصطلحات موضوعية: Cellular immunity, T-Lymphocytes, medicine.medical_treatment, Immunology, Mice, Nude, Apoptosis, Biology, Biochemistry, Mice, chemistry.chemical_compound, Immune system, Neoplasms, medicine, Animals, Humans, Indoleamine-Pyrrole 2,3,-Dioxygenase, Enzyme Inhibitors, CD86, Immunity, Cellular, Mice, Inbred BALB C, Dose-Response Relationship, Drug, Cell growth, Dendritic Cells, Cell Biology, Hematology, Coculture Techniques, Tryptophan Oxygenase, In vitro, Cytokine, chemistry, Cancer research, B7-2 Antigen, Kynurenine, HeLa Cells
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::d1d22827acb3bc70083e41ba10ba8e88
https://doi.org/10.1182/blood-2009-09-246124 -
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المؤلفون: Maria Rafalski, Wei Han, Swamy Yeleswaram, Charles F. Albright, Melody Diamond, George L. Trainor, Nilsa R. Graciani, Randine Dowling, Xiang-Jun Jiang, Zilun Hu, Steven P. Seitz, Eddy W. Yue, Robert Bruckner, Mingzhu Zhang, Shu-Yun Zhang
المصدر: Bioorganic & Medicinal Chemistry Letters. 20:853-856
مصطلحات موضوعية: Clinical Biochemistry, Pharmaceutical Science, Antineoplastic Agents, macromolecular substances, Matrix metalloproteinase, Biochemistry, Mice, Therapeutic index, In vivo, Cell Line, Tumor, Drug Discovery, polycyclic compounds, medicine, Animals, Humans, Prodrugs, Doxorubicin, Molecular Biology, Neprilysin, Chemistry, organic chemicals, Organic Chemistry, technology, industry, and agriculture, Prodrug, Xenograft Model Antitumor Assays, Matrix Metalloproteinases, carbohydrates (lipids), Cancer research, Molecular Medicine, HT1080, Ex vivo, medicine.drug
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المؤلفون: Jordan S. Fridman, Michael Hansbury, Richard B. Sparks, Andrew P. Combs, Gengjie Yang, Kevin Bowman, Holly Koblish, Paul Waeltz, Patrick J. Haley, Peggy Scherle, Timothy Burn, Kris Vaddi, Eddy W. Yue, Claire L. Neilan
المصدر: Molecular Cancer Therapeutics. 9:489-498
مصطلحات موضوعية: Cancer Research, Amidines, Pharmacology, Biology, Mice, chemistry.chemical_compound, Dogs, Immune system, In vivo, Cell Line, Tumor, Neoplasms, medicine, Animals, Humans, Indoleamine-Pyrrole 2,3,-Dioxygenase, Lymphocytes, Enzyme Inhibitors, Indoleamine 2,3-dioxygenase, Kynurenine, Mice, Inbred BALB C, Catabolism, Tryptophan, Cancer, medicine.disease, In vitro, Oncology, chemistry, Immune System, Female, Immunotherapy, Lymph Nodes, Lymph
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::58dd4aaafcf4e05d0076d4a647cde251
https://doi.org/10.1158/1535-7163.mct-09-0628