-
1
المؤلفون: Melissa C. Holt, Zahra Assar, Reza Beheshti Zavareh, Lin Lin, Justin Anglin, Oksana Mashadova, Daniel Haldar, Edouard Mullarky, Daniel M. Kremer, Lewis C. Cantley, Alec C. Kimmelman, Adam J. Stein, Luke L. Lairson, Costas A. Lyssiotis
المصدر: Biochemistry. 57:6604-6614
مصطلحات موضوعية: Models, Molecular, 0301 basic medicine, Binding Sites, 010304 chemical physics, Protein Conformation, Crystallography, X-Ray, 01 natural sciences, Biochemistry, Article, High-Throughput Screening Assays, Pancreatic Neoplasms, Structure-Activity Relationship, 03 medical and health sciences, 030104 developmental biology, Colonic Neoplasms, Mutation, 0103 physical sciences, Tumor Cells, Cultured, Humans, Metabolomics, Enzyme Inhibitors, Aspartate Aminotransferase, Cytoplasmic, Cell Proliferation
-
2
المؤلفون: Lewis C. Cantley, Rafael de Cabo, Ana P. Gomes, Julie Han, Anders P. Mutvei, Charles Kinzig, Jennifer E. Endress, Mélanie Planque, Noah Dephoure, Didem Ilter, Vivien Low, John Blenis, John M. Asara, Tanya Schild, Sarah-Maria Fendt, Edouard Mullarky, Adnan Ahmed, Ilaria Elia, Juan Fernández-García, Adam Rosenzweig, Dorien Broekaert
مصطلحات موضوعية: business.industry, Methylmalonic acid, food and beverages, Cancer, medicine.disease, SOX4, chemistry.chemical_compound, Mediator, chemistry, Tumor progression, Cancer cell, Cancer research, medicine, Propionate metabolism, business, Reprogramming
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::3cf4462822fb091fe9b09e5db2d9c920
https://doi.org/10.1101/2020.06.04.135087 -
3
المؤلفون: Lewis C. Cantley, Roozbeh Eskandari, Vipin Suri, Roger Liang, Nello Mainolfi, Edward R. Kastenhuber, Diane Kang, Min Yu, Matthew G. Vander Heiden, Ariana Plasger, Jing Ni, Alba Luengo, Victoria Osorio-Vasquez, Ahmed Ali, Rakesh K. Jain, David M. Sabatini, Edouard Mullarky, Eugenie Kim, Shawn M. Davidson, Samuel F. Bakhoum, Matija Snuderl, Bryan Ngo, Eva Hernando, Sophia Doll, Jean J. Zhao, Mark Manfredi, Matthias Mann, Sarah Bacha, Michael E. Pacold, Roshan K. Siriam, Gino D. Ferraro, Paolo Cotzia, Sophia Bustraan, Adam Friedman, Drew R. Jones
مصطلحات موضوعية: 0303 health sciences, Biology, medicine.disease, 3. Good health, Metastasis, Serine, 03 medical and health sciences, 0302 clinical medicine, Downregulation and upregulation, Cell culture, Glycine, medicine, Cancer research, Gene silencing, Phosphoglycerate dehydrogenase, 030217 neurology & neurosurgery, 030304 developmental biology, Brain metastasis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::4e114c3b878bf679b40fc5a4320aca66
https://doi.org/10.1101/2020.03.03.974980 -
4
المؤلفون: Mélanie Planque, Didem Ilter, Noah Dephoure, Lewis C. Cantley, Juan Fernández-García, Adam Rosenzweig, Adnan Ahmed, Ilaria Elia, Charles Kinzig, Edouard Mullarky, John Blenis, Tanya Schild, Dorien Broekaert, Vivien Low, Jennifer E. Endress, Sarah-Maria Fendt, John M. Asara, Rafael de Cabo, Ana P. Gomes, Julie Han, Anders P. Mutvei
المصدر: Nature
مصطلحات موضوعية: 0301 basic medicine, Male, Aging, Methylmalonic acid, chemistry.chemical_compound, Mice, 0302 clinical medicine, Transforming Growth Factor beta, Neoplasms, GLUTATHIONE, Medicine, Neoplasm Metastasis, ONCOGENESIS, Multidisciplinary, food and beverages, Middle Aged, EPITHELIAL-MESENCHYMAL TRANSITION, 3. Good health, PROSTATE-CANCER, Gene Expression Regulation, Neoplastic, Multidisciplinary Sciences, 030220 oncology & carcinogenesis, Disease Progression, Science & Technology - Other Topics, Female, SOX4, Signal transduction, Signal Transduction, Adult, EXPRESSION, GENES, METABOLISM, Article, SOXC Transcription Factors, 03 medical and health sciences, Mediator, Downregulation and upregulation, Cell Line, Tumor, Animals, Humans, Neoplasm Invasiveness, Aged, Science & Technology, business.industry, Cancer, medicine.disease, 030104 developmental biology, chemistry, Ageing, Cancer cell, METASTASIS, CELLS, Cancer research, business, Transcriptome, Methylmalonic Acid
وصف الملف: Print-Electronic
-
5
المؤلفون: Daniel Haldar, Justin L. Anglin, Reza Beheshti Zavareh, Costas A. Lyssiotis, Alec C. Kimmelman, Philipp N. Sander, Luke L. Lairson, Lewis C. Cantley, Edouard Mullarky
المصدر: Bioorganic & Medicinal Chemistry Letters. 28:2675-2678
مصطلحات موضوعية: 0301 basic medicine, Indoles, Clinical Biochemistry, Cell, Pharmaceutical Science, Malignancy, Biochemistry, Piperazines, Article, Transaminase, Mice, Structure-Activity Relationship, 03 medical and health sciences, 0302 clinical medicine, Drug Stability, Pharmacokinetics, Drug Discovery, medicine, Animals, Potency, Aspartate Aminotransferases, Enzyme Inhibitors, Molecular Biology, Transaminases, Chemistry, Phenylurea Compounds, Organic Chemistry, Cancer, medicine.disease, Small molecule, Metabolic pathway, 030104 developmental biology, medicine.anatomical_structure, 030220 oncology & carcinogenesis, Cancer research, Molecular Medicine, Female, Aspartate Aminotransferase, Cytoplasmic, Carcinoma, Pancreatic Ductal
-
6
المؤلفون: Stacia Kargman, Andrew John Jennings, Michael Miller, Andrew Stamford, Damodharan Lakshminarasimhan, Lewis C. Cantley, Anita D. Robin, Mayako Michino, David J. Huggins, Jiayi Xu, Edouard Mullarky, Andrea Olland, Daisuke Tomita, Naoyoshi Noguchi, Guoan Zhang, Peter T. Meinke, Taojunfeng Su
المصدر: Bioorg Med Chem Lett
مصطلحات موضوعية: Indoles, Clinical Biochemistry, Pharmaceutical Science, Dehydrogenase, Molecular Dynamics Simulation, Crystallography, X-Ray, 01 natural sciences, Biochemistry, Article, Serine, Structure-Activity Relationship, Cell Line, Tumor, Drug Discovery, Humans, Phosphoglycerate dehydrogenase, Enzyme Inhibitors, Molecular Biology, Phosphoglycerate Dehydrogenase, Cell Proliferation, chemistry.chemical_classification, Indole test, Binding Sites, 010405 organic chemistry, Organic Chemistry, Oxidoreductase inhibitor, Amides, 0104 chemical sciences, Protein Structure, Tertiary, 010404 medicinal & biomolecular chemistry, Metabolic pathway, Enzyme, chemistry, Molecular Medicine, NAD+ kinase
-
7
المؤلفون: Sejeong Shin, Noah Dephoure, Edouard Mullarky, Lewis C. Cantley, Sang-Oh Yoon, Paola Cavaliere, Adam Rosenzweig, Vivien Low, Zih-Jie Shen, Ekrem Emrah Er, Joan Massagué, Jessica K. Tyler, Dylan R. McNally, John Blenis, Didem Ilter, Tanya Schild, Michal J. Nagiec, Ana P. Gomes, Julie Han, Anders P. Mutvei, Yi-Hung Ou, Martín A. Rivas, Ari Melnick
المصدر: Cancer Cell
مصطلحات موضوعية: 0301 basic medicine, Male, Cancer Research, Epithelial-Mesenchymal Transition, Carcinogenesis, Chromatin remodeling, Article, Epigenesis, Genetic, Histones, 03 medical and health sciences, Histone H3, Mice, 0302 clinical medicine, Cell Line, Tumor, Animals, Humans, Epigenetics, RNA-Seq, Neoplasm Metastasis, Promoter Regions, Genetic, Transcription factor, CAF-1 complex, Regulation of gene expression, biology, Carcinoma, Cell Biology, Xenograft Model Antitumor Assays, Chromatin, Cell biology, Gene Expression Regulation, Neoplastic, Chromatin Assembly Factor-1, 030104 developmental biology, Histone, Oncology, 030220 oncology & carcinogenesis, biology.protein, Disease Progression, Female, Transcription Factors
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::12264f5d2a1ddfe7ce67b10259df1913
https://pubmed.ncbi.nlm.nih.gov/31564638 -
8
المؤلفون: Jing Ni, Roozbeh Eskandari, Matija Snuderl, Edward R. Kastenhuber, Sophia Doll, Roshan K. Sriram, Rakesh K. Jain, Jean J. Zhao, Sophia Bustraan, Michael E. Pacold, Ahmed Ali, Eugenie Kim, Samuel F. Bakhoum, Edouard Mullarky, Bryan Ngo, Adam Friedman, Nello Mainolfi, Matthias Mann, Drew R. Jones, David M. Sabatini, Vipin Suri, Ariana Plasger, Roger Liang, Shawn M. Davidson, Lewis C. Cantley, Diane Kang, Min Yu, Alba Luengo, Benjamin D. Stein, Sarah Bacha, Mark Manfredi, Gino D. Ferraro, Matthew G. Vander Heiden
المصدر: Cancer Research. 80:5712-5712
مصطلحات موضوعية: Serine, Cancer Research, Breast cancer, Oncology, business.industry, medicine, Cancer research, medicine.disease, business, Brain metastasis
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::04d87cb3ec58463388bfa48ef3dc155c
https://doi.org/10.1158/1538-7445.am2020-5712 -
9
المؤلفون: Quentin Spillier, Lewis C. Cantley, Anita D. Robin, Alice Dutu, Edouard Mullarky, Séverine Ravez, Raphaël Frédérick, Cyril Corbet, Olivier Feron
مصطلحات موضوعية: 0301 basic medicine, Drug Evaluation, Preclinical, Context (language use), Antineoplastic Agents, Article, 03 medical and health sciences, 0302 clinical medicine, Cell Line, Tumor, Neoplasms, Drug Discovery, High-Throughput Screening Assays, Humans, Phosphoglycerate dehydrogenase, Enzyme Inhibitors, Phosphoglycerate Dehydrogenase, Cell Proliferation, chemistry.chemical_classification, Chemistry, Extramural, In vitro, Thioamides, 030104 developmental biology, Enzyme, Biochemistry, 030220 oncology & carcinogenesis, Molecular Medicine, Pharmacophore, Function (biology)
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::83923eb21d42f4aef1c6ef102fab580a
https://europepmc.org/articles/PMC5603230/ -
10
المؤلفون: Alec C. Kimmelman, Ya'an Kang, Xiaoxu Wang, Lewis C. Cantley, Rushika M. Perera, John M. Asara, Jason B. Fleming, Matteo Ligorio, Jaekyoung Son, Costas A. Lyssiotis, Marcia C. Haigis, Edouard Mullarky, Ronald A. DePinho, Nabeel Bardeesy, Ng Shyh-Chang, Cristina R. Ferrone, Haoqiang Ying, Sujun Hua
المصدر: Nature
مصطلحات موضوعية: 0303 health sciences, Multidisciplinary, Glutaminolysis, endocrine system diseases, Glutamate dehydrogenase, Biology, Mitochondrion, GOT2, Article, 3. Good health, Glutamine, Citric acid cycle, 03 medical and health sciences, Metabolic pathway, 0302 clinical medicine, Biochemistry, 030220 oncology & carcinogenesis, Cancer cell, 030304 developmental biology