-
1
المؤلفون: Adrian Liam Gill, Severin K. Thompson, Alexander G. Dossetter, Edward Jolyon Griffen, Andreas Buckl
المصدر: Expert Opinion on Therapeutic Patents. 31:1189-1204
مصطلحات موضوعية: Patent literature, Son of Sevenless, Antineoplastic Agents, Bioinformatics, Patents as Topic, Drug Development, Neoplasms, Drug Discovery, Animals, Humans, Medicine, Pharmacology, biology, business.industry, Drug discovery, Cancer, General Medicine, medicine.disease, Small molecule, Clinical trial, Mutation, ras Proteins, biology.protein, SOS1, Signal transduction, SOS1 Protein, business, Signal Transduction
-
2
المصدر: Burger's Medicinal Chemistry and Drug Discovery
مصطلحات موضوعية: Quantitative structure–activity relationship, Computer science, business.industry, Artificial intelligence, business, CASP
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::6dad82e4dcff9e7b8e8b110d17da8fc9
https://doi.org/10.1002/0471266949.bmc267 -
3
المؤلفون: Stephen J. Messham, Andrew G. Leach, Steven J. Enoch, Francesco Coppola, Alhusein Hussin, Joanna Zarnecka, Alexander G. Dossetter, Iva Lukac, Edward Jolyon Griffen
المصدر: Zarnecka, J, Lukac, I, Messham, S J, Hussin, A, Coppola, F, Enoch, S J, Dossetter, A G, Griffen, E J & Leach, A G 2021, ' Mapping Ligand-Shape Space for Protein–Ligand Systems: Distinguishing Key-in-Lock and Hand-in-Glove Proteins ', Journal of Chemical Information and Modeling, vol. 61, no. 4, pp. 1859–1874 . https://doi.org/10.1021/acs.jcim.1c00089
مصطلحات موضوعية: Physics, Binding Sites, Record locking, 010304 chemical physics, Protein Conformation, General Chemical Engineering, Molecular Conformation, Proteins, General Chemistry, Library and Information Sciences, Type (model theory), Ligands, Ligand (biochemistry), 01 natural sciences, 0104 chemical sciences, Computer Science Applications, Set (abstract data type), 010404 medicinal & biomolecular chemistry, Molecular geometry, 0103 physical sciences, Key (cryptography), Molecule, Biological system, Algorithms, Protein ligand
وصف الملف: application/pdf
-
4
المصدر: Griffen, E J, Dossetter, A G & Leach, A G 2020, ' Chemists: AI Is Here; Unite To Get the Benefits ', Journal of Medicinal Chemistry . https://doi.org/10.1021/acs.jmedchem.0c00163
مصطلحات موضوعية: 0303 health sciences, Chemistry, Management science, Chemistry, Pharmaceutical, Quantitative Structure-Activity Relationship, 01 natural sciences, 0104 chemical sciences, 010404 medicinal & biomolecular chemistry, 03 medical and health sciences, Computational Chemistry, Artificial Intelligence, Drug Discovery, Molecular Medicine, Humans, Interdisciplinary communication, Cooperative behavior, Chemistry (relationship), Cooperative Behavior, 030304 developmental biology
وصف الملف: application/pdf
-
5
المؤلفون: Andrew G. Leach, Edward Jolyon Griffen, Alexander Dossetter
مصطلحات موضوعية: Computer science, Component (UML), Scale (chemistry), Data mining, Matched molecular pair analysis, computer.software_genre, computer, Analysis method, Field (computer science)
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::153d972ffc2649cd076296af91cf5114
https://doi.org/10.1039/9781788016841-00250 -
6
المصدر: Griffen, E J, Dossetter, A G, Leach, A G & Montague, S 2018, ' Can we accelerate medicinal chemistry by augmenting the chemist with Big Data and artificial intelligence? ', Drug discovery today, vol. 23, no. 7, pp. 1373-1384 . https://doi.org/10.1016/j.drudis.2018.03.011
مصطلحات موضوعية: QA75, 0301 basic medicine, RM, Chemistry, Pharmaceutical, Big data, Intellectual property, Chemist, Task (project management), Structure-Activity Relationship, 03 medical and health sciences, Artificial Intelligence, Drug Discovery, Animals, Data Mining, Humans, Chemistry (relationship), Set (psychology), Pharmacology, Molecular Structure, business.industry, Drug discovery, High-Throughput Screening Assays, Knowledge sharing, 030104 developmental biology, Pharmaceutical Preparations, Artificial intelligence, business, Databases, Chemical
وصف الملف: application/pdf
-
7
المؤلفون: Dennis Norman, Helen E. Colley, Munitta Muthana, Lynne Williams, Joanne Harrison, Sean F. Coole, Mark J. Thompson, Edward Jolyon Griffen, Matthew L. Brett, Sarah Danson, Vamshi Tulasi, Lucinda V. Jackson, Peter Lockey, Melanie Wong, Daniel P. Mason, Luke Jennings, Alexander G. Dossetter
المصدر: Journal of Medicinal Chemistry. 58:9309-9333
مصطلحات موضوعية: Male, Indoles, Mice, Nude, Antineoplastic Agents, Microtubules, Mice, Structure-Activity Relationship, Tubulin, Microtubule, Drug Discovery, Animals, Humans, Cytotoxic T cell, Structure–activity relationship, Cell Proliferation, biology, Tubulin Modulators, Cell growth, Chemistry, Molecular biology, Head and Neck Neoplasms, Caco-2, Cell culture, Cancer research, biology.protein, Heterografts, Molecular Medicine, Caco-2 Cells, Drug Screening Assays, Antitumor, Neoplasm Transplantation
-
8
المؤلفون: Andrew G. Leach, Iva Lukac, Alexander G. Dossetter, Joanna Zarnecka, Edward Jolyon Griffen
مصطلحات موضوعية: Cheminformatics, Drug discovery, Chemistry, Computational biology, Matched molecular pair analysis, Combinatorial chemistry
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_________::f081cb2a3dc011fbe2da44161cf99f74
https://doi.org/10.1016/b978-0-12-409547-2.12347-9 -
9
المصدر: Drug Discovery Today. 18:724-731
مصطلحات موضوعية: Pharmacology, Molecular Structure, Computer science, Process (engineering), Drug discovery, Matched-Pair Analysis, computer.software_genre, Yield design, Structure-Activity Relationship, Drug Design, Drug Discovery, Animals, Humans, Data mining, Matched molecular pair analysis, computer
-
10
المصدر: Journal of Medicinal Chemistry. 54:7739-7750
مصطلحات موضوعية: Chemistry, Drug Discovery, Molecular Medicine, Matched molecular pair analysis, Medicinal chemistry