-
1
المؤلفون: Brian M. Arnold, Miriam del Prado, Smriti Iyengar, Edward L. Mattiuz, Zhipei Wu, Mark A. Winter, David Bleakman, Ken H. Ho, Ann Marie L. Ogden, Paul L. Ornstein, Carrie K. Jones, Sandra Ann Filla, Brian Michael Mathes, Michael Gregory Bell, Douglas Richard Stack, Ana Maria Escribano, Thomas J. Bleisch, Ana I. Mateo, Kevin John Hudziak, Andrew Alt, Rosa Maria A. Simmons, Harlan E. Shannon, Robert E. Stratford, Jose A. Martinez-Perez, Esteban Dominguez, Ana M. Castaño
المصدر: Bioorganic & Medicinal Chemistry Letters. 23:6459-6462
مصطلحات موضوعية: Molecular Sequence Data, Clinical Biochemistry, Administration, Oral, Pain, Pharmaceutical Science, Pharmacology, Biochemistry, Structure-Activity Relationship, chemistry.chemical_compound, Receptors, Kainic Acid, Oral administration, In vivo, Drug Discovery, Animals, Prodrugs, Amino Acid Sequence, Molecular Biology, Benzoic acid, chemistry.chemical_classification, Chemistry, Organic Chemistry, Haplorhini, Prodrug, Isoquinolines, Amino acid, Disease Models, Animal, Molecular Medicine
-
2
المؤلفون: Edward L. Mattiuz, Ann Marie L. Ogden, Ana M. Castaño, Zhipei Wu, Robert E. Stratford, E. Dominguez, Thomas J. Bleisch, Brian Michael Mathes, Brian M. Arnold, David Bleakman, Smriti Iyengar, Rosa Maria A. Simmons, Harlan E. Shannon, Sandra Ann Filla, Jose A. Martinez-Perez, Douglas Richard Stack, Ana I. Mateo, Miriam del Prado, Kevin John Hudziak, Andrew Alt, Michael Gregory Bell, Carrie K. Jones, Paul L. Ornstein, Jennifer L. Buckmaster, Ana Maria Escribano, Mark A. Winter, Ken H. Ho
المصدر: Journal of Medicinal Chemistry. 48:4200-4203
مصطلحات موضوعية: Analgesic, Biological Availability, Pain, Kainate receptor, Pharmacology, Cell Line, Receptors, Kainic Acid, Drug Discovery, Animals, Humans, Receptors, AMPA, Amino Acids, Receptor, alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid, chemistry.chemical_classification, Analgesics, Chemistry, Glutamate receptor, Antagonist, Prodrug, Recombinant Proteins, Rats, Amino acid, Disease Models, Animal, Spinal Cord, Biochemistry, Hyperalgesia, Molecular Medicine, Licking
-
3
المؤلفون: Amanda J. Long, Jennifer Witcher, Edward L. Mattiuz, John-Michael Sauer, Holly R. Thomasson, Karl A. Desante, G. Douglas Ponsler
المصدر: Drug Metabolism and Disposition. 31:98-107
مصطلحات موضوعية: Adult, Male, Pharmacology, CYP2D6, Propylamines, Metabolite, Atomoxetine, Pharmaceutical Science, Middle Aged, Atomoxetine Hydrochloride, Excretion, Hydroxylation, chemistry.chemical_compound, Cytochrome P-450 CYP2D6, chemistry, Pharmacokinetics, Oral administration, medicine, Humans, Biotransformation, Atomoxetine hydrochloride, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::9637f5478fba6df030f42b65abba078a
https://doi.org/10.1124/dmd.31.1.98 -
4
المؤلفون: Ken H. Ho, Edward L. Mattiuz, Ann Marie L. Ogden, Brian Michael Mathes, Ana I. Mateo, David Bleakman, Kevin John Hudziak, Donna K. Dieckman, Sandra Ann Filla, Mark A. Winter, Thomas J. Bleisch, Ana Maria Escribano, Paul L. Ornstein, Kirk W. Johnson, Douglas Richard Stack, Amy Clemens-Smith, Miriam del Prado, Ana M. Castaño, Mary A. Katofiasc, Robert E. Stratford, E. Dominguez, Michael Gregory Bell, Lee A. Phebus, Jose A. Martinez-Perez
المصدر: Journal of Medicinal Chemistry. 45:4383-4386
مصطلحات موضوعية: Stereochemistry, Migraine Disorders, Carboxylic Acids, Administration, Oral, Biological Availability, Kainate receptor, Pharmacology, Cell Line, Radioligand Assay, Receptors, Kainic Acid, Drug Discovery, medicine, Animals, Humans, Prodrugs, Rats, Wistar, Receptor, Dose-Response Relationship, Drug, Chemistry, Antagonist, Glutamate receptor, Esters, Biological activity, Prodrug, Isoquinolines, Rats, Disease Models, Animal, Mechanism of action, Competitive antagonist, Acute Disease, Molecular Medicine, Calcium, medicine.symptom, Excitatory Amino Acid Antagonists
-
5
المؤلفون: Miriam del Prado, Ken H. Ho, Brian Michael Mathes, Smriti Iyengar, Mark A. Winter, Harlan E. Shannon, Carrie K. Jones, David K. Clawson, Ana Maria Escribano, Douglas Richard Stack, Esteban Dominguez, Paul L. Ornstein, Ana I. Mateo, Jose A. Martinez-Perez, Kevin John Hudziak, Andrew Alt, Edward L. Mattiuz, Brian M. Arnold, Sandra Ann Filla, Thomas J. Bleisch, Ana M. Castaño, Michael Gregory Bell, Rosa Maria A. Simmons, Robert E. Stratford, Ann Marie L. Ogden, Zhipei Wu, David Bleakman
المصدر: Bioorganicmedicinal chemistry letters. 23(23)
مصطلحات موضوعية: Male, Stereochemistry, Clinical Biochemistry, Analgesic, Molecular Sequence Data, Pharmaceutical Science, Administration, Oral, Pain, Tetrazoles, Biochemistry, Rats, Sprague-Dawley, chemistry.chemical_compound, Structure-Activity Relationship, Receptors, Kainic Acid, In vivo, Drug Discovery, Animals, Tetrazole, Prodrugs, Amino Acid Sequence, Receptor, Molecular Biology, Organic Chemistry, Prodrug, Isoquinolines, In vitro, Rats, Disease Models, Animal, chemistry, Molecular Medicine, Selectivity, Linker
-
6
المؤلفون: Palaniappan Kulanthaivel, Robert J. Barbuch, William J. Wheeler, Anthony G. Borel, Timothy M. Jones, Valentine J. Klimkowski, Edward L. Mattiuz, David A. Jackson, Gregory A. Rener
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 39(5)
مصطلحات موضوعية: Male, Stereochemistry, Pyridines, Metabolite, Pharmaceutical Science, Tandem mass spectrometry, chemistry.chemical_compound, Dogs, Bathochromic shift, Animals, Receptors, Ghrelin, Structural analog, Pharmacology, Chromatography, Human Growth Hormone, Aromatization, Imidazoles, Dipeptides, Rats, Inbred F344, Rats, chemistry, Lipophilicity, Female, Quantitative analysis (chemistry), Heterocyclic Compounds, 3-Ring, Conjugate
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::66aad7994ceadaaf07c6971089063b82
https://pubmed.ncbi.nlm.nih.gov/21346003 -
7
المؤلفون: David O. Calligaro, Amy Clemens-Smith, Ken H. Ho, Darryle D. Schoepp, Marlene L. Cohen, Mary Gates, Robert E. Stratford, Paul L. Ornstein, K.R Jarvie, Ann Marie L. Ogden, Sandra Ann Filla, Rebecca A. Wright, Mary A. Katofiasc, Brianne Weiss, Bryan G. Johnson, Geihan Rizkalla, Andrew Alt, Craig R. Salhoff, Kathryn W. Schenck, David Bleakman, Donna K. Dieckman, Kirk W. Johnson, Edward L. Mattiuz, Lee A. Phebus
المصدر: The Journal of pharmacology and experimental therapeutics. 318(2)
مصطلحات موضوعية: Male, medicine.drug_class, Migraine Disorders, Phencyclidine, Kainate receptor, AMPA receptor, Pharmacology, In Vitro Techniques, Motor Activity, Ligands, Transfection, Binding, Competitive, Muscle, Smooth, Vascular, Trigeminal ganglion, Benzodiazepines, Dorsal root ganglion, Receptors, Kainic Acid, medicine, Animals, Humans, Saphenous Vein, Receptors, AMPA, Receptor, Neurons, Chemistry, Glutamate receptor, Antagonist, Blood Proteins, Receptor antagonist, Isoquinolines, Rats, Electrophysiology, medicine.anatomical_structure, Molecular Medicine, Calcium, Rabbits, Excitatory Amino Acid Antagonists, Proto-Oncogene Proteins c-fos, Muscle Contraction
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::5211cdf990741fc3ac26cc363aeecbe0
https://pubmed.ncbi.nlm.nih.gov/16690725 -
8
المؤلفون: Palaniappan, Kulanthaivel, Robert J, Barbuch, Rita S, Davidson, Ping, Yi, Gregory A, Rener, Edward L, Mattiuz, Chad E, Hadden, Lawrence A, Goodwin, William J, Ehlhardt
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 32(9)
مصطلحات موضوعية: Time Factors, Siloxanes, Drug Evaluation, Preclinical, Hydroxylation, Catalysis, Mass Spectrometry, Cyclic N-Oxides, Dogs, Isomerism, Animals, Amines, Furans, Vinca Alkaloids, Serum Albumin, Titanium, Molecular Structure, Temperature, Water, Isoquinolines, Rats, Pyridazines, Pharmaceutical Preparations, Sulfoxides, Female, Oxidation-Reduction, Palladium, Chromatography, Liquid
URL الوصول: https://explore.openaire.eu/search/publication?articleId=pmid________::9e887b1b44310fe6ff04f5c0030b8818
https://pubmed.ncbi.nlm.nih.gov/15319338 -
9
المؤلفون: M. G. Gadberry, William J. Wheeler, Edward L. Mattiuz, Nagy A. Farid, K. C. Cassidy, E. J. Perkins, D. D. O'Bannon, Paul G. Wood, David A. Jackson, J. W. Cramer, H. J. Weiss
المصدر: Drug metabolism and disposition: the biological fate of chemicals. 31(11)
مصطلحات موضوعية: Male, Metabolite, Glucuronidation, Drug Evaluation, Preclinical, Pharmaceutical Science, Ether, Benzoates, chemistry.chemical_compound, Mice, Species Specificity, In vivo, Animals, Humans, Benzoic acid, Pharmacology, Metabolism, Middle Aged, Blood proteins, Macaca mulatta, Rats, Inbred F344, Rats, Macaca fascicularis, chemistry, Biochemistry, Liver, Female, Glucuronide
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::7a4d32b7976ade8f159a6d2829756459
https://pubmed.ncbi.nlm.nih.gov/14570771 -
10
المؤلفون: Steven A. Wrighton, Edward L. Mattiuz, William J. Ehlhardt, Matthew G. Soars, David A. Jackson, Palaniappan Kulanthaivel
المصدر: Journal of pharmacological and toxicological methods. 47(3)
مصطلحات موضوعية: Bioanalysis, Magnetic Resonance Spectroscopy, Glucuronidation, Anthraquinones, Toxicology, Ethinyl Estradiol, Xenobiotics, chemistry.chemical_compound, Dogs, Glucuronides, In vivo, Ethinylestradiol, Gallic Acid, medicine, Animals, Humans, Glucuronosyltransferase, Propofol, Chromatography, High Pressure Liquid, Pharmacology, Chromatography, Haplorhini, Reference Standards, Glucuronic acid, Buprenorphine, Rats, chemistry, Biochemistry, Microsome, Microsomes, Liver, Xenobiotic, Glucuronide, medicine.drug