المؤلفون: Abdelgawad MA, Al-Sanea MM, Musa A, Elmowafy M, El-Damasy AK, Azouz AA, Ghoneim MM, Bakr RR

المصدر: Journal of Inflammation Research, Vol Volume 15, Pp 451-463 (2022)

مصطلحات موضوعية: cyclooxygenase inhibitors, anti-inflammatory activity, ulcerogenic effects, tricyclic pyridopyrimidines, Pathology, RB1-214, Therapeutics. Pharmacology, RM1-950

وصف الملف: electronic resource

Relation: https://www.dovepress.com/docking-study-synthesis-and-anti-inflammatory-potential-of-some-new-py-peer-reviewed-fulltext-article-JIR; https://doaj.org/toc/1178-7031

URL الوصول: https://doaj.org/article/4ab2aeeb54f3482fa4da464477e8831f

المؤلفون: Bae SH; Department of Medical and Biological Sciences, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea.; BK Four Department of Biotechnology, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea., Yoo S; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, 02792, Republic of Korea., Lee J; Department of Medical and Biological Sciences, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea., Park HJ; Department of Medical and Biological Sciences, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea.; BK Four Department of Biotechnology, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea., Kwon SP; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, 02792, Republic of Korea., Jin H; Center for Advanced Biomolecular Recognition, Korea Institute of Science and Technology (KIST), Seoul, 02792, Republic of Korea.; Division of Bio-Medical Science and Technology, KIST School, University of Science and Technology (UST), Seoul, Republic of Korea., Park SI; SML Biopharm, Gwangmyeong, 14353, Republic of Korea., Lee YS; Department of Medical and Biological Sciences, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea.; BK Four Department of Biotechnology, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea., Bang YJ; Department of Medical and Biological Sciences, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea.; BK Four Department of Biotechnology, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea., Roh G; Department of Medical and Biological Sciences, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea.; BK Four Department of Biotechnology, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea., Lee S; Department of Medical and Biological Sciences, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea.; BK Four Department of Biotechnology, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea., Youn SB; Department of Medical and Biological Sciences, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea.; BK Four Department of Biotechnology, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea., Kim IW; Cancer Research Institute, Seoul National University College of Medicine, Seoul, 03080, Republic of Korea., Oh HR; Cancer Research Institute, Seoul National University College of Medicine, Seoul, 03080, Republic of Korea., El-Damasy AK; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, 02792, Republic of Korea., Keum G; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, 02792, Republic of Korea., Kim H; Center for Advanced Biomolecular Recognition, Korea Institute of Science and Technology (KIST), Seoul, 02792, Republic of Korea.; Division of Bio-Medical Science and Technology, KIST School, University of Science and Technology (UST), Seoul, Republic of Korea., Youn H; Cancer Research Institute, Seoul National University College of Medicine, Seoul, 03080, Republic of Korea.; Department of Nuclear Medicine, Cancer Imaging Center, Seoul National University Hospital, Seoul, 03080, Republic of Korea., Nam JH; Department of Medical and Biological Sciences, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea.; BK Four Department of Biotechnology, The Catholic University of Korea, Gyeonggi-do, Bucheon, Republic of Korea., Bang EK; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, 02792, Republic of Korea.; KHU-KIST Department of Converging Science and Technology, Graduate School, Kyung Hee University, Seoul, 02447, Republic of Korea.

المصدر: Bioactive materials [Bioact Mater] 2024 May 14; Vol. 38, pp. 486-498. Date of Electronic Publication: 2024 May 14 (Print Publication: 2024).

نوع المنشور: Journal Article

بيانات الدورية: Publisher: Ke Ai Publishing Country of Publication: China NLM ID: 101685294 Publication Model: eCollection Cited Medium: Internet ISSN: 2452-199X (Electronic) Linking ISSN: 2452199X NLM ISO Abbreviation: Bioact Mater Subsets: PubMed not MEDLINE

المؤلفون: El-Damasy AK; Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea.; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura 35516, Egypt., Kim HJ; Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea., Al-Karmalawy AA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Horus University-Egypt, New Damietta 34518, Egypt.; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Ahram Canadian University, 6th of October City 12566, Egypt., Alnajjar R; CADD Unit, Faculty of Pharmacy, Libyan International Medical University, Benghazi 16063, Libya.; Department of Chemistry, Faculty of Science, University of Benghazi, Benghazi 16063, Libya.; Department of Chemistry, University of Cape Town, Rondebosch 7700, South Africa., Khalifa MM; Department of Pharmaceutical Medicinal Chemistry & Drug Design, Faculty of Pharmacy (Boys), Al-Azhar University, Cairo 11884, Egypt., Bang EK; Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea., Keum G; Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea.

المصدر: Pharmaceuticals (Basel, Switzerland) [Pharmaceuticals (Basel)] 2024 Mar 27; Vol. 17 (4). Date of Electronic Publication: 2024 Mar 27.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101238453 Publication Model: Electronic Cited Medium: Print ISSN: 1424-8247 (Print) Linking ISSN: 14248247 NLM ISO Abbreviation: Pharmaceuticals (Basel) Subsets: PubMed not MEDLINE

المؤلفون: El-Damasy AK; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, South Korea.; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt., Kim HJ; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, South Korea., Nocentini A; Section of Pharmaceutical and Nutraceutical Sciences, Department of NEUROFARBA, University of Florence, Florence, Italy.; Laboratory of Molecular Modeling Cheminformatics & QSAR, Department of NEUROFARBA-Pharmaceutical and Nutraceutical Section, University of Firenze, Florence, Italy., Seo SH; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, South Korea., Eldehna WM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafr El Sheikh, Egypt., Bang EK; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, South Korea., Supuran CT; Section of Pharmaceutical and Nutraceutical Sciences, Department of NEUROFARBA, University of Florence, Florence, Italy., Keum G; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, South Korea.; Division of Bio-Medical Science & Technology, KIST School, Korea University of Science and Technology (UST), Seoul, South Korea.

المصدر: Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2023 Dec; Vol. 38 (1), pp. 2154603.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: Taylor & Francis Country of Publication: England NLM ID: 101150203 Publication Model: Print Cited Medium: Internet ISSN: 1475-6374 (Electronic) Linking ISSN: 14756366 NLM ISO Abbreviation: J Enzyme Inhib Med Chem Subsets: MEDLINE

مواضيع طبية MeSH: Carbonic Anhydrases*/metabolism, Humans ; Structure-Activity Relationship ; Carbonic Anhydrase Inhibitors/pharmacology ; Carbonic Anhydrase IX ; Antigens, Neoplasm ; MCF-7 Cells ; Coumarins/pharmacology ; Molecular Structure

المؤلفون: El-Damasy AK; Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, Republic of Korea.; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt., Kim HJ; Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, Republic of Korea., Park JW; Supercomputing Application Center, Div. of National Supercomputing, Korea Institute of Science and Technology Information, Daejeon, Republic of Korea., Nam Y; Medicinal Materials Research Center, Korea Institute of Science and Technology (KIST), Seoul, Republic of Korea., Hur W; Medicinal Materials Research Center, Korea Institute of Science and Technology (KIST), Seoul, Republic of Korea., Bang EK; Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, Republic of Korea., Keum G; Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, Republic of Korea.; Division of Bio-Medical Science & Technology, KIST School, Korea University of Science and Technology (UST), Seoul, Republic of Korea.

المصدر: Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2023 Dec; Vol. 38 (1), pp. 2228515.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: Taylor & Francis Country of Publication: England NLM ID: 101150203 Publication Model: Print Cited Medium: Internet ISSN: 1475-6374 (Electronic) Linking ISSN: 14756366 NLM ISO Abbreviation: J Enzyme Inhib Med Chem Subsets: MEDLINE

مواضيع طبية MeSH: Indazoles*/pharmacology , Leukemia, Myelogenous, Chronic, BCR-ABL Positive*/drug therapy , Leukemia, Myelogenous, Chronic, BCR-ABL Positive*/genetics , Leukemia, Myelogenous, Chronic, BCR-ABL Positive*/metabolism, Humans ; Drug Resistance, Neoplasm ; Imatinib Mesylate/pharmacology ; Imatinib Mesylate/therapeutic use ; Protein Kinase Inhibitors/pharmacology ; Protein Kinase Inhibitors/therapeutic use ; Fusion Proteins, bcr-abl/genetics ; Fusion Proteins, bcr-abl/metabolism ; Benzamides/pharmacology ; Cell Line, Tumor ; Mutation ; Cell Proliferation ; Apoptosis

المؤلفون: El-Damasy AK; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, Republic of Korea.; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt., Jin H; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, Republic of Korea., Park JW; Center for Supercomputing Applications, Div. of National Supercomputing R&D, Korea Institute of Science and Technology Information, Daejeon, Republic of Korea., Kim HJ; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, Republic of Korea., Khojah H; Department of Pharmacognosy, College of Pharmacy, Jouf University, Sakaka, Saudi Arabia., Seo SH; Center for Brain Disorders, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, Republic of Korea., Lee JH; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, Republic of Korea., Bang EK; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, Republic of Korea., Keum G; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul, Republic of Korea.; Division of Bio-Medical Science & Technology, KIST School, Korea University of Science and Technology (UST), Seoul, Republic of Korea.

المصدر: Journal of enzyme inhibition and medicinal chemistry [J Enzyme Inhib Med Chem] 2023 Dec; Vol. 38 (1), pp. 2189097.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: Taylor & Francis Country of Publication: England NLM ID: 101150203 Publication Model: Print Cited Medium: Internet ISSN: 1475-6374 (Electronic) Linking ISSN: 14756366 NLM ISO Abbreviation: J Enzyme Inhib Med Chem Subsets: MEDLINE

مواضيع طبية MeSH: Fusion Proteins, bcr-abl*/genetics , Pyrimidines*/pharmacology, Imatinib Mesylate/pharmacology ; Piperazines/pharmacology ; Benzamides/pharmacology ; Apoptosis

المؤلفون: El-Damasy AK; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea.; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura 35516, Egypt., Jin H; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea., Sabry MA; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura 35516, Egypt., Kim HJ; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea., Alanazi MM; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh 11451, Saudi Arabia., Seo SH; Center for Brain Disorders, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea., Bang EK; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea., Keum G; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea.; Division of Bio-Medical Science & Technology, KIST School, Korea University of Science and Technology (UST), Seoul 02792, Republic of Korea.

المصدر: Medicina (Kaunas, Lithuania) [Medicina (Kaunas)] 2023 Jun 02; Vol. 59 (6). Date of Electronic Publication: 2023 Jun 02.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: MDPI Country of Publication: Switzerland NLM ID: 9425208 Publication Model: Electronic Cited Medium: Internet ISSN: 1648-9144 (Electronic) Linking ISSN: 1010660X NLM ISO Abbreviation: Medicina (Kaunas) Subsets: MEDLINE

مواضيع طبية MeSH: Thiazoles*/pharmacology , Thiazoles*/therapeutic use , Antineoplastic Agents*/pharmacology , Antineoplastic Agents*/therapeutic use, Humans ; Structure-Activity Relationship ; Drug Screening Assays, Antitumor ; Cell Proliferation ; Cell Line, Tumor ; Pyrimidines/pharmacology ; Pyrimidines/therapeutic use ; Dose-Response Relationship, Drug

المؤلفون: Kim HJ; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea., Park JW; Supercomputing Application Center, Division of National Supercomputing, Korea Institute of Science and Technology Information, Daejeon 34141, Republic of Korea., Seo S; Supercomputing Application Center, Division of National Supercomputing, Korea Institute of Science and Technology Information, Daejeon 34141, Republic of Korea., Cho KH; School of Systems Biomedical Science, Soongsil University, Seoul 06978, Republic of Korea., Alanazi MM; Department of Pharmaceutical Chemistry, College of Pharmacy, King Saud University, Riyadh 11421, Saudi Arabia., Bang EK; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea., Keum G; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea.; Division of Bio-Medical Science & Technology, KIST School, Korea University of Science and Technology (UST), Seoul 02792, Republic of Korea., El-Damasy AK; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea.

المصدر: International journal of molecular sciences [Int J Mol Sci] 2023 Feb 06; Vol. 24 (4). Date of Electronic Publication: 2023 Feb 06.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101092791 Publication Model: Electronic Cited Medium: Internet ISSN: 1422-0067 (Electronic) Linking ISSN: 14220067 NLM ISO Abbreviation: Int J Mol Sci Subsets: MEDLINE

مواضيع طبية MeSH: Antineoplastic Agents*/pharmacology , Melanoma*/drug therapy , Quinolones*/pharmacology, Humans ; Cell Line, Tumor ; Cell Proliferation ; Drug Screening Assays, Antitumor ; Molecular Docking Simulation ; Protein Kinase Inhibitors/pharmacology ; Proto-Oncogene Proteins B-raf/metabolism ; Structure-Activity Relationship

المؤلفون: El-Damasy AK; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea.; Department of Medicinal Chemistry, Faculty of Pharmacy, Mansoura University, Mansoura 35516, Egypt., Park JE; Department of Pharmacy, and Research Institute of Life Pharmaceutical Sciences, Sunchon National University, Suncheon 57922, Republic of Korea., Kim HJ; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea., Lee J; Disease Target Structure Research Center, Korea Research Institute of Bioscience and Biotechnology (KRIBB), Daejeon 34141, Republic of Korea.; Department of Bioinformatics, KRIBB School of Bioscience, University of Science and Technology (UST), Daejeon 34113, Republic of Korea., Bang EK; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea., Kim H; Department of Pharmacy, and Research Institute of Life Pharmaceutical Sciences, Sunchon National University, Suncheon 57922, Republic of Korea., Keum G; Center for Brain Technology, Brain Science Institute, Korea Institute of Science and Technology (KIST), Seoul 02792, Republic of Korea.

المصدر: Pharmaceuticals (Basel, Switzerland) [Pharmaceuticals (Basel)] 2023 Jan 06; Vol. 16 (1). Date of Electronic Publication: 2023 Jan 06.

نوع المنشور: Journal Article

بيانات الدورية: Publisher: MDPI Country of Publication: Switzerland NLM ID: 101238453 Publication Model: Electronic Cited Medium: Print ISSN: 1424-8247 (Print) Linking ISSN: 14248247 NLM ISO Abbreviation: Pharmaceuticals (Basel) Subsets: PubMed not MEDLINE

المؤلفون: El-Abd AO; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Delta University for Science and Technology, 11152 Gamasa, Egypt., Bayomi SM; Department of Medicinal Chemistry, Faculty of Pharmacy, University of Mansoura, 35516 Mansoura, Egypt., El-Damasy AK; Department of Medicinal Chemistry, Faculty of Pharmacy, University of Mansoura, 35516 Mansoura, Egypt., Mansour B; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Delta University for Science and Technology, 11152 Gamasa, Egypt., Abdel-Aziz NI; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Delta University for Science and Technology, 11152 Gamasa, Egypt.; Department of Medicinal Chemistry, Faculty of Pharmacy, University of Mansoura, 35516 Mansoura, Egypt., El-Sherbeny MA; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Delta University for Science and Technology, 11152 Gamasa, Egypt.; Department of Medicinal Chemistry, Faculty of Pharmacy, University of Mansoura, 35516 Mansoura, Egypt.

المصدر: ACS omega [ACS Omega] 2022 Sep 07; Vol. 7 (37), pp. 33599-33613. Date of Electronic Publication: 2022 Sep 07 (Print Publication: 2022).

نوع المنشور: Journal Article

بيانات الدورية: Publisher: American Chemical Society Country of Publication: United States NLM ID: 101691658 Publication Model: eCollection Cited Medium: Internet ISSN: 2470-1343 (Electronic) Linking ISSN: 24701343 NLM ISO Abbreviation: ACS Omega Subsets: PubMed not MEDLINE