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1
المؤلفون: Elaine Ryan, Qi Gao, Cathy D. Mahle, Dedong Wu, Lawrence G. Iben, Stephen R. Bertenshaw, Li-Qiang Sun, Jie Chen, Cen Xu, Katherine S. Takaki
المصدر: Bioorganic & Medicinal Chemistry Letters. 15:1345-1349
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Ligands, Biochemistry, Chemical synthesis, Melatonin receptor, Mice, Structure-Activity Relationship, Drug Discovery, medicine, Animals, Humans, Vasoconstrictor Agents, Cloning, Molecular, Receptor, Molecular Biology, Benzofurans, Melatonin, Rat tail artery, Molecular Structure, Bicyclic molecule, Receptor, Melatonin, MT2, Chemistry, Receptor, Melatonin, MT1, Organic Chemistry, General Medicine, Ligand (biochemistry), Recombinant Proteins, In vitro, Rats, Vasoconstriction, NIH 3T3 Cells, Molecular Medicine, Aliphatic compound, Protein Binding
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2
المؤلفون: Anthony J. Gentile, Jeffrey A. Deskus, Nathan S. Sarbin, James R. Epperson, Elaine Ryan, Lawrence G. Iben
المصدر: Bioorganic & Medicinal Chemistry Letters. 14:1023-1026
مصطلحات موضوعية: Agonist, medicine.drug_class, Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Carboxamide, Binding, Competitive, Biochemistry, Chemical synthesis, Melatonin, Structure-Activity Relationship, Drug Discovery, medicine, Humans, Anilides, Receptor, Molecular Biology, Molecular Structure, Receptor, Melatonin, MT2, Chemistry, Organic Chemistry, In vitro, Melatonergic, Molecular Medicine, Selectivity, medicine.drug
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3
المؤلفون: Amit G. Gulwadi, Subramaniam Krishnananthan, Matthew T. Taber, Henry Wong, Thaddeus F. Molski, Carolyn D. Korpinen, Kai Xie, Cen Xu, Qi Gao, Elaine Ryan, Graham Johnson, Swanee Jacutin-Porte, Juliang Zhu, Todd A. Verdoorn, Kevin D. Burris, Sing-Yuen Sit
المصدر: Journal of Medicinal Chemistry. 45:3660-3668
مصطلحات موضوعية: Agonist, Stereochemistry, medicine.drug_class, Molecular Conformation, Convergent synthesis, Dinapsoline, Naphthols, In Vitro Techniques, Crystallography, X-Ray, Chemical synthesis, Dopamine agonist, Cell Line, Rats, Sprague-Dawley, Radioligand Assay, chemistry.chemical_compound, Drug Discovery, Cyclic AMP, medicine, Animals, Isoquinoline, Receptors, Dopamine D2, Receptors, Dopamine D1, Stereoisomerism, Isoquinolines, Corpus Striatum, Rats, chemistry, Dopamine Agonists, Molecular Medicine, Pharmacophore, Enantiomer, medicine.drug
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4
المؤلفون: Kevin D. Burris, Frank D. Yocca, Perry B. Molinoff, Cen Xu, Katsura Tottori, Thaddeus F. Molski, Tetsuro Kikuchi, Elaine Ryan
المصدر: Journal of Pharmacology and Experimental Therapeutics. 302:381-389
مصطلحات موضوعية: Agonist, medicine.medical_specialty, medicine.drug_class, Bifeprunox, Aripiprazole, Atypical antipsychotic, CHO Cells, Quinolones, Pharmacology, Partial agonist, Piperazines, Radioligand Assay, GTP-Binding Proteins, 1-Methyl-3-isobutylxanthine, Cricetinae, Internal medicine, Dopamine receptor D2, Cyclic AMP, medicine, Animals, Humans, Receptors, Dopamine D2, Chemistry, Colforsin, Dopaminergic, Dopamine D2 Receptor Antagonists, Endocrinology, Spiperone, Dopamine Agonists, Dopamine Antagonists, Molecular Medicine, Endogenous agonist, Antipsychotic Agents, Signal Transduction, medicine.drug
URL الوصول: https://explore.openaire.eu/search/publication?articleId=doi_dedup___::2744104acf9b25b331d41051008ca48b
https://doi.org/10.1124/jpet.102.033175 -
5
المؤلفون: Cathy D. Mahle, Katherine S. Takaki, Cen Xu, Jay O. Knipe, Lori Pajor, Jie Chen, Lawrence G. Iben, Li-Qiang Sun, Elaine Ryan
المصدر: Bioorganicmedicinal chemistry letters. 14(20)
مصطلحات موضوعية: Agonist, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Pharmaceutical Science, Administration, Oral, Biological Availability, Pharmacology, In Vitro Techniques, Biochemistry, Chemical synthesis, Melatonin receptor, Muscle, Smooth, Vascular, Melatonin, chemistry.chemical_compound, Mice, Radioligand Assay, Structure-Activity Relationship, Drug Discovery, Acetamides, medicine, Cyclic AMP, Animals, Humans, Benzofuran, Receptor, Molecular Biology, Melatonin receptor agonist, Benzofurans, Dose-Response Relationship, Drug, Receptor, Melatonin, MT2, Receptor, Melatonin, MT1, Organic Chemistry, General Medicine, Bioavailability, Rats, chemistry, NIH 3T3 Cells, Molecular Medicine, Acetamide, medicine.drug, Muscle Contraction
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6
المؤلفون: Nathan S. Sarbin, Anthony J. Gentile, Lawrence G. Iben, Jeffrey A. Deskus, Elaine Ryan, James R. Epperson
المصدر: ChemInform. 35
مصطلحات موضوعية: Melatonin, Chemistry, Stereochemistry, Mt1 receptor, medicine, General Medicine, Selectivity, Receptor, Melatonergic, medicine.drug
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7
المؤلفون: Jie Chen, Cen Xu, Lawrence G. Iben, Katherine S. Takaki, Cathy D. Mahle, James R. Epperson, Jeffrey A. Deskus, Graham Johnson, Elaine Ryan, Li-Qiang Sun, Marc Bruce
المصدر: Bioorganicmedicinal chemistry letters. 14(14)
مصطلحات موضوعية: Agonist, Stereochemistry, medicine.drug_class, Clinical Biochemistry, Receptors, Melatonin, Pharmaceutical Science, Receptors, Cell Surface, Ligands, Biochemistry, Chemical synthesis, Melatonin receptor, Cell Line, chemistry.chemical_compound, Radioligand Assay, Structure-Activity Relationship, Drug Discovery, Radioligand, medicine, Structure–activity relationship, Humans, Receptor, Molecular Biology, Melatonin, Benzoxazoles, Binding Sites, Bicyclic molecule, Chemistry, Organic Chemistry, Benzoxazole, Drug Design, Molecular Medicine
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8كتاب
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9
المؤلفون: Li-Qiang Sun, Jie Chen, Ronald J. Mattson, James R. Epperson, Jeffrey A. Deskus, Wen-Sen Li, Katherine Takaki, Donald B. Hodges, Lawrence Iben, Cathy D. Mahle, Astrid Ortiz, David Molstad, Elaine Ryan, Krishnaswamy Yeleswaram, Cen Xu, Guanglin Luo
المصدر: Bioorganicmedicinal chemistry letters. 13(24)
مصطلحات موضوعية: Stereochemistry, Clinical Biochemistry, Pharmaceutical Science, Ligands, Biochemistry, Melatonin receptor, Chemical synthesis, Pyrrole derivatives, Mice, Structure-Activity Relationship, Heterocyclic Compounds, Drug Discovery, Cyclic AMP, Animals, Humans, Cloning, Molecular, Molecular Biology, Melatonin, Bicyclic molecule, Chemistry, Receptor, Melatonin, MT2, Receptor, Melatonin, MT1, Organic Chemistry, Colforsin, 3T3 Cells, Recombinant Proteins, Melatonergic, Kinetics, Aminoquinolines, Molecular Medicine
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10
المؤلفون: Graham Johnson, Jie Chen, Cathy D. Mahle, Cen Xu, Elaine Ryan, Katherine S. Takaki, Lawrence G. Iben, Li-Qiang Sun
المصدر: Bioorganicmedicinal chemistry letters. 14(5)
مصطلحات موضوعية: medicine.drug_class, Stereochemistry, Clinical Biochemistry, Receptors, Melatonin, Pharmaceutical Science, Carboxamide, Ligands, Biochemistry, Chemical synthesis, chemistry.chemical_compound, Drug Discovery, medicine, Radioligand, Humans, Receptor, Molecular Biology, Melatonin, Benzoxazoles, Bicyclic molecule, Organic Chemistry, General Medicine, Benzoxazole, Ligand (biochemistry), Affinities, chemistry, Drug Design, Molecular Medicine, Pharmacophore, Protein Binding